Target Details
| UniProt AC | P49354 |
|---|---|
| Gene Symbol | FNTA |
| Protein Name | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01239 (PPTA) |
Summary
- Multi-target molecules 1,421
- Clinical molecules 1125
- Avg pChEMBL 7.75
KEGG Pathways (1)
Active Molecules (1,421)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZCCICPFBBPENMT
|
8.9 | pIC50 | 3 | Yes | |
ZGBJQRVUJIKBSE
|
8.9 | pIC50 | 2 | Yes | |
AHPUIZQTTZGXBJ
|
8.9 | pIC50 | 3 | Yes | |
CMJUYLXTUMAMFB
|
8.9 | pIC50 | 2 | Yes | |
CXKCBVJOXUNDSU
|
8.9 | pIC50 | 2 | Yes | |
IGCORMDACWRGMB
|
8.9 | pIC50 | 3 | Yes | |
UZMOGBCVDQWRFX
|
8.9 | pIC50 | 2 | Yes | |
VXSSQHPMYCZWRC
|
8.9 | pIC50 | 2 | Yes | |
XEYVAVWLDJJMQX
|
8.9 | pIC50 | 2 | Yes | |
XHIISTKHRQWJJN
|
8.9 | pIC50 | 3 | Yes | |
YDQQLXXIRZYPPK
|
8.9 | pIC50 | 3 | Yes | |
YIHOJJQZGPJKGV
|
8.9 | pIC50 | 3 | Yes | |
ZEIRRWOZIKZYIO
|
8.9 | pIC50 | 3 | Yes | |
OLUZMRATNLVQMT
|
8.9 | IC50 | 2 | — | |
AYVGITDSDRJQKI
|
8.8 | pIC50 | 3 | Yes | |
BAHABGBETCGAQD
|
8.8 | IC50 | 3 | — | |
CKADUCCMLBGQGD
|
8.8 | pIC50 | 3 | Yes | |
FZJOMPQKENNHGD
|
8.8 | pIC50 | 3 | Yes | |
KMNYYAJYASNHCC
|
8.8 | pIC50 | 3 | Yes | |
KPRXKFKHZVTBIT
|
8.8 | pIC50 | 2 | Yes | |
KUHZXPPLZCMGNF
|
8.8 | pIC50 | 2 | Yes | |
KULAYTGUTXCHSV
|
8.8 | IC50 | 2 | — | |
NAUDEXJEXLGXTN
|
8.8 | pIC50 | 2 | Yes | |
STZJDNIOWZMUJX
|
8.8 | pIC50 | 2 | Yes | |
WBCIUSMPAYCADE
|
8.8 | IC50 | 2 | — | |
DLASOUKHRBZNDA
|
8.8 | pIC50 | 2 | Yes | |
HMTOSAULPVTKEX
|
8.8 | pIC50 | 2 | Yes | |
HOOMWYSTEWJDOS
|
8.8 | pIC50 | 2 | Yes | |
KICVKKMBSGOHAY
|
8.8 | pIC50 | 3 | Yes | |
VWNBOOIWICWEPL
|
8.8 | IC50 | 2 | — | |
XFLDZCZKAVQGOE
|
8.8 | IC50 | 2 | — | |
YSZYMWKMFGGIQP
|
8.8 | pIC50 | 2 | Yes | |
ZBVRAORJUFNDAX
|
8.8 | pIC50 | 2 | Yes | |
ZQIKAKSHLZASKW
|
8.8 | pIC50 | 2 | Yes | |
MASXKDVYFMKYRW
|
8.8 | pIC50 | 2 | Yes | |
UNEVEWKTGHFQJP
|
8.8 | pIC50 | 2 | Yes | |
USPFJPDEADLGIG
|
8.8 | IC50 | 2 | — | |
XJVUCSNFEJKWBV
|
8.8 | pIC50 | 2 | Yes | |
YIZSZHVXFHAUCR
|
8.8 | pIC50 | 3 | Yes | |
FARRVZOQABGAGC
|
8.8 | pIC50 | 2 | Yes | |
HGDNILFTURGNIL
|
8.8 | pIC50 | 3 | Yes | |
HQDNURJWABRGRP
|
8.8 | pIC50 | 2 | Yes | |
JBTVOWMPTOMYFD
|
8.8 | pIC50 | 2 | Yes | |
SCQNETOOVNYIJP
|
8.8 | pIC50 | 2 | Yes | |
SJOPIYABUQAMST
|
8.8 | IC50 | 2 | — | |
WBCIUSMPAYCADE
|
8.8 | IC50 | 2 | — | |
WOYOASASOHZEDR
|
8.8 | pIC50 | 2 | Yes | |
RHXLRBJBYOPEAL
|
8.8 | pIC50 | 2 | Yes | |
WDIWKDRZXKMPAH
|
8.8 | pIC50 | 2 | Yes | |
AYMOTDQQAAKWQI
|
8.7 | pIC50 | 2 | Yes |