Target Details
| UniProt AC | P49354 |
|---|---|
| Gene Symbol | FNTA |
| Protein Name | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01239 (PPTA) |
Summary
- Multi-target molecules 1,421
- Clinical molecules 1125
- Avg pChEMBL 7.75
KEGG Pathways (1)
Active Molecules (1,421)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UQRQADYTKHCQGV
|
9.0 | pIC50 | 2 | Yes | |
VBOYISMKUMBEJC
|
9.0 | pIC50 | 3 | Yes | |
BBVMIKDYONNPSU
|
9.0 | pIC50 | 2 | Yes | |
HPTPUWFOBXCUAN
|
9.0 | pIC50 | 3 | Yes | |
BHKKLGROGAROGK
|
9.0 | pIC50 | 3 | Yes | |
AIOFERITDFXPBZ
|
9.0 | pIC50 | 2 | Yes | |
AIZAXCJJFKTNIA
|
9.0 | pIC50 | 2 | Yes | |
ASJFFPIKUVTYEV
|
9.0 | IC50 | 2 | — | |
ASJFFPIKUVTYEV
|
9.0 | pIC50 | 2 | Yes | |
BICXECMCJCNEDG
|
9.0 | pIC50 | 2 | Yes | |
CJOWDGQKVQMHOD
|
9.0 | pIC50 | 2 | Yes | |
GYHJYVOLUAYUGE
|
9.0 | pIC50 | 2 | Yes | |
HKGUHEGKBLYKHY
|
9.0 | pIC50 | 3 | Yes | |
IEVQWJGNVJGOPG
|
9.0 | pIC50 | 2 | Yes | |
JJQTVXNPRRSENU
|
9.0 | pIC50 | 2 | Yes | |
JRTOBKVVIBBEQD
|
9.0 | pIC50 | 2 | Yes | |
KISBCVMWQAXCRV
|
9.0 | pIC50 | 2 | Yes | |
KKJPSAVOCOHZGT
|
9.0 | pIC50 | 2 | Yes | |
NAEYWVZYJOIXPA
|
9.0 | pIC50 | 3 | Yes | |
OCGBVMDVBLYKEO
|
9.0 | pIC50 | 2 | Yes | |
OUQYWOOMZNKZCC
|
9.0 | pIC50 | 2 | Yes | |
PBRQCWRYSWNUKC
|
9.0 | IC50 | 2 | — | |
QFVRKKGXFGGVET
|
9.0 | pIC50 | 3 | Yes | |
RFDWGJYINANKTJ
|
9.0 | pIC50 | 2 | Yes | |
RZOJUYACASNMGU
|
9.0 | pIC50 | 2 | Yes | |
VEZHVPLIKFFIOV
|
9.0 | pIC50 | 2 | Yes | |
YHIHBFWTEDMUPR
|
9.0 | pIC50 | 2 | Yes | |
ARZMSIQUIDXWHZ
|
9.0 | pIC50 | 2 | Yes | |
BCNAPHWOUDETDR
|
9.0 | IC50 | 2 | — | |
BECWPNYJZIVGFM
|
9.0 | pIC50 | 3 | Yes | |
BHBPTTBKKZBFIQ
|
9.0 | pIC50 | 2 | Yes | |
GAQHYZNOMLXSEA
|
9.0 | pIC50 | 2 | Yes | |
GDPDFNXDSFOTHH
|
9.0 | pIC50 | 3 | Yes | |
MNUNZZHRDOMTJY
|
9.0 | pIC50 | 3 | Yes | |
OBXLXUGOZZWQOW
|
9.0 | IC50 | 2 | — | |
VLQSBTGRKZOYFJ
|
9.0 | pIC50 | 4 | Yes | |
WISKOZINSNUMIP
|
9.0 | pIC50 | 2 | Yes | |
XIVVAPJAZVPZQR
|
9.0 | pIC50 | 2 | Yes | |
ZGQAAHNNGHYZAB
|
9.0 | pIC50 | 2 | Yes | |
PPSUJYUXOZCAFU
|
8.9 | pIC50 | 3 | Yes | |
ADDOXKIOPBTSEG
|
8.9 | pIC50 | 2 | Yes | |
AVEYRMOKDFXVLL
|
8.9 | pIC50 | 2 | Yes | |
BIHDOYKIKJUQTP
|
8.9 | pIC50 | 2 | Yes | |
FBXAUVHISXRYSQ
|
8.9 | IC50 | 2 | — | |
GRKGCIUUSLKRTB
|
8.9 | pIC50 | 2 | Yes | |
KHPPZVJYPAXFML
|
8.9 | pIC50 | 2 | Yes | |
NIACYCIOHPNBOW
|
8.9 | pIC50 | 2 | Yes | |
OAOJLQIBUMOZQL
|
8.9 | pIC50 | 2 | Yes | |
YBYDQOIAYNOCOH
|
8.9 | pIC50 | 2 | Yes | |
YCUWEXRMZLDWND
|
8.9 | pIC50 | 3 | Yes |