Target Details
| UniProt AC | P49354 |
|---|---|
| Gene Symbol | FNTA |
| Protein Name | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01239 (PPTA) |
Summary
- Multi-target molecules 1,421
- Clinical molecules 1125
- Avg pChEMBL 7.75
KEGG Pathways (1)
Active Molecules (1,421)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VSZXKSCVZMOQFB
|
9.2 | pIC50 | 3 | Yes | |
YHZAWDJTCMTRQA
|
9.2 | pIC50 | 2 | Yes | |
ZPHPMNJCCXXCGX
|
9.2 | pIC50 | 3 | Yes | |
ZXEBGRLCZDOCAL
|
9.2 | pIC50 | 2 | Yes | |
AXIVWWPYPSYJLD
|
9.1 | pIC50 | 7 | Yes | |
LFTRQPMHZNHIDH
|
9.1 | pIC50 | 2 | Yes | |
PPUPMAFZXZRFPN
|
9.1 | pIC50 | 2 | Yes | |
YREMCUVJCPALAV
|
9.1 | pIC50 | 2 | Yes | |
BGKFZODPGHMODV
|
9.1 | pIC50 | 2 | Yes | |
SWLCOFSBLYLWEQ
|
9.1 | pIC50 | 2 | Yes | |
ZLNNDPISKMQXCE
|
9.1 | pIC50 | 2 | Yes | |
BLEVYVOQEISZIT
|
9.1 | pIC50 | 3 | Yes | |
OUAONGDGIKMGQT
|
9.1 | pIC50 | 2 | Yes | |
BXRDSFHISHNZJF
|
9.1 | pIC50 | 2 | Yes | |
DJZAMXRHXDPZOJ
|
9.1 | IC50 | 2 | — | |
GTURWVWPNOUBNH
|
9.1 | pIC50 | 3 | Yes | |
GUUIRIMAQGOLHT
|
9.1 | IC50 | 2 | — | |
MWUKOHOBDTWNMQ
|
9.1 | IC50 | 2 | — | |
OEMBXAJIJLOISQ
|
9.1 | pIC50 | 2 | Yes | |
PLHJCIYEEKOWNM
|
9.1 | pIC50 | 4 | Yes | |
RDECPKAPXFKZRQ
|
9.1 | pIC50 | 3 | Yes | |
RHTSWGZKPCQUKZ
|
9.1 | pIC50 | 3 | Yes | |
SFJJHGCGXLUQLC
|
9.1 | pIC50 | 2 | Yes | |
YRBSHYLIBVCREO
|
9.1 | pIC50 | 2 | Yes | |
ZGXXVZOEOVXKNI
|
9.1 | pIC50 | 2 | Yes | |
KIJGRUQPENRVQJ
|
9.1 | pIC50 | 2 | Yes | |
PCCXFDJNOPAWDJ
|
9.1 | pIC50 | 2 | Yes | |
DUORQQSLNAGSSQ
|
9.1 | pIC50 | 3 | Yes | |
SHUCBLWUZXSRAC
|
9.1 | pIC50 | 3 | Yes | |
XIPVCWJXWJDNCA
|
9.1 | pIC50 | 2 | Yes | |
ASUWZCFQGVUVGX
|
9.1 | pIC50 | 3 | Yes | |
HYDRIOWWHJJSSW
|
9.1 | pIC50 | 3 | Yes | |
KULAYTGUTXCHSV
|
9.1 | pIC50 | 4 | Yes | |
GOQKNURHCDAYKJ
|
9.1 | pIC50 | 3 | Yes | |
DIAXSDUMDSLTMQ
|
9.1 | pIC50 | 2 | Yes | |
FLBYMAWUXCWVAF
|
9.1 | pIC50 | 2 | Yes | |
FUQQEQIALYIXCF
|
9.1 | pIC50 | 2 | Yes | |
GLENTBWEHGHDCL
|
9.1 | pIC50 | 2 | Yes | |
GSZHIOCIMUCGFD
|
9.1 | pIC50 | 2 | Yes | |
HWLBLFBLGGVDBT
|
9.1 | pIC50 | 3 | Yes | |
NIKJJDARCUJOSC
|
9.1 | pIC50 | 3 | Yes | |
OCODFFZNRDTKIQ
|
9.1 | IC50 | 2 | — | |
PTNBPPZVBINDKZ
|
9.1 | pIC50 | 3 | Yes | |
PZCCBYWNHZAHAG
|
9.1 | pIC50 | 2 | Yes | |
VHSNTJWPNYCXNM
|
9.1 | pIC50 | 2 | Yes | |
VRUOPFISMXRWIS
|
9.1 | IC50 | 2 | — | |
VZFHWZARTPYKEO
|
9.1 | pIC50 | 2 | Yes | |
XEOVKXSFYIXXCT
|
9.1 | pIC50 | 2 | Yes | |
CCWBGSWFGJGKBW
|
9.0 | pIC50 | 2 | Yes | |
JHFMJRWJSSLDJT
|
9.0 | pIC50 | 2 | Yes |