Target Details
| UniProt AC | P49354 |
|---|---|
| Gene Symbol | FNTA |
| Protein Name | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01239 (PPTA) |
Summary
- Multi-target molecules 1,421
- Clinical molecules 1125
- Avg pChEMBL 7.75
KEGG Pathways (1)
Active Molecules (1,421)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DJVTZQIKKLGURV
|
9.3 | pIC50 | 3 | Yes | |
DJYOAYPWIWACRH
|
9.3 | pIC50 | 3 | Yes | |
GKFPROVOIQKYTO
|
9.3 | IC50 | 2 | — | |
ORYMXHUFOAZSNG
|
9.3 | pIC50 | 2 | Yes | |
QKFHVTMTAUFWNT
|
9.3 | pIC50 | 3 | Yes | |
WJLNAPDUWBBQHL
|
9.3 | pIC50 | 3 | Yes | |
WQCSBRZKGIGNTL
|
9.3 | pIC50 | 2 | Yes | |
XPKOMAYTINMMOL
|
9.3 | pIC50 | 2 | Yes | |
ZIXDDEATQSBHHL
|
9.3 | pIC50 | 5 | Yes | |
VXVRUWALANZFFN
|
9.3 | pIC50 | 2 | Yes | |
VYLMFRUDZGQCNT
|
9.3 | pIC50 | 6 | Yes | |
JGIGBEKDNKBDDC
|
9.3 | pIC50 | 2 | Yes | |
FWWJGHORTZMPHN
|
9.3 | pIC50 | 2 | Yes | |
ITOOXSJDSBTQNY
|
9.3 | pIC50 | 3 | Yes | |
SFSVYOSUWJRGTM
|
9.2 | pIC50 | 2 | Yes | |
LMXZFNUEMHAYLD
|
9.2 | pIC50 | 3 | Yes | |
PJUKABGUVXKGFB
|
9.2 | pIC50 | 2 | Yes | |
LMGSQMQVUYDBRD
|
9.2 | pIC50 | 2 | Yes | |
GEOWAWJUOWQWJH
|
9.2 | pIC50 | 3 | Yes | |
HQQOMOWVWPBVRR
|
9.2 | pIC50 | 2 | Yes | |
HQQOMOWVWPBVRR
|
9.2 | pIC50 | 3 | Yes | |
KZSBNUBNJHIROE
|
9.2 | pIC50 | 2 | Yes | |
NLCBWQRVYLSINY
|
9.2 | pIC50 | 4 | Yes | |
RYTREGFJFCUMBB
|
9.2 | pIC50 | 2 | Yes | |
TYNOFQUWLFNSFL
|
9.2 | IC50 | 2 | — | |
TYNOFQUWLFNSFL
|
9.2 | IC50 | 2 | — | |
XKBOADWPZLOLCO
|
9.2 | pIC50 | 3 | Yes | |
YYDYJITZGLMMFM
|
9.2 | IC50 | 2 | — | |
KUCIXFHIZYSMOM
|
9.2 | pIC50 | 2 | Yes | |
PVPHNBNJQXLVQM
|
9.2 | pIC50 | 2 | Yes | |
WUBHEKLVWNZHSF
|
9.2 | pIC50 | 3 | Yes | |
XXNOXIHVPUERGU
|
9.2 | pIC50 | 3 | Yes | |
STYWCLSYFHKEDV
|
9.2 | pIC50 | 2 | Yes | |
WHPKJYJVLZBIAP
|
9.2 | pIC50 | 3 | Yes | |
CQCNIBNGGPUKMH
|
9.2 | pIC50 | 3 | Yes | |
MFPPMKRAKTUYMX
|
9.2 | pIC50 | 3 | Yes | |
MRIIEPZJIMUDLC
|
9.2 | pIC50 | 3 | Yes | |
WYJDYTUMUBOENZ
|
9.2 | pIC50 | 2 | Yes | |
RXGGZGACWDLIGX
|
9.2 | pIC50 | 2 | Yes | |
VDAIFUYTPNJOFW
|
9.2 | pIC50 | 2 | Yes | |
XRJFAINHZHMKOK
|
9.2 | pIC50 | 3 | Yes | |
HRCUJSFALQORGR
|
9.2 | pIC50 | 3 | Yes | |
ONSUIKYVBGOGPD
|
9.2 | pIC50 | 2 | Yes | |
BJWFIOSIGHDXLF
|
9.2 | pIC50 | 2 | Yes | |
FPEPZFNRGIPRRN
|
9.2 | pIC50 | 2 | Yes | |
KVCBEZWLSRNJTD
|
9.2 | pIC50 | 2 | Yes | |
OAEIWTGUZXTPAT
|
9.2 | pIC50 | 3 | Yes | |
OKGNJWICJWXHCX
|
9.2 | IC50 | 2 | — | |
OLCWFLWEHWLBTO
|
9.2 | pIC50 | 4 | Yes | |
VRUOPFISMXRWIS
|
9.2 | IC50 | 2 | — |