Target Details
| UniProt AC | P49354 |
|---|---|
| Gene Symbol | FNTA |
| Protein Name | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01239 (PPTA) |
Summary
- Multi-target molecules 1,421
- Clinical molecules 1125
- Avg pChEMBL 7.75
KEGG Pathways (1)
Active Molecules (1,421)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CHVJSILONSNEQT
|
9.5 | pIC50 | 2 | Yes | |
MDKRCQNLMFYBAJ
|
9.5 | pIC50 | 2 | Yes | |
CKVSFSCNFUEJNJ
|
9.5 | pIC50 | 3 | Yes | |
CXZANANUPGZRRJ
|
9.5 | pIC50 | 2 | Yes | |
JDDIKIAGECJRRO
|
9.5 | pIC50 | 2 | Yes | |
JNJBXYHGNTUTTK
|
9.5 | pIC50 | 4 | Yes | |
XUQVGNQCLMEBOL
|
9.5 | pIC50 | 3 | Yes | |
YZFYPECRJZGSGJ
|
9.5 | IC50 | 2 | — | |
ZBRVJLSHNVWEKS
|
9.5 | pIC50 | 3 | Yes | |
JRJRLAHKHIKIEQ
|
9.5 | pIC50 | 2 | Yes | |
YGJHSCAJBDJRFY
|
9.5 | pIC50 | 3 | Yes | |
NBMZKTWABZIDLO
|
9.5 | pIC50 | 2 | Yes | |
QGPSHWUWMGSFJB
|
9.5 | pIC50 | 3 | Yes | |
QOTXVDPQOVHXPX
|
9.5 | pIC50 | 3 | Yes | |
NKNMRYCDVOOEKZ
|
9.5 | pIC50 | 3 | Yes | |
HWHGRAMVKSPMDJ
|
9.5 | pIC50 | 2 | Yes | |
SRVLVBDYUWMIOB
|
9.4 | pIC50 | 3 | Yes | |
VRUYMJKZIKNSKH
|
9.4 | pIC50 | 3 | Yes | |
DCDYIJATVKPDDB
|
9.4 | pIC50 | 2 | Yes | |
DIBXXBYKQOAPHR
|
9.4 | pIC50 | 2 | Yes | |
IGCOPNHCHHWZNH
|
9.4 | pIC50 | 3 | Yes | |
JQBCZQXINWOHEL
|
9.4 | pIC50 | 2 | Yes | |
KWJJDZYGKXQTJC
|
9.4 | pIC50 | 2 | Yes | |
XWDXWBALIUAPLO
|
9.4 | pIC50 | 2 | Yes | |
IQZCODLAPFPVNS
|
9.4 | IC50 | 2 | — | |
ACXPVQQIYOUAGF
|
9.4 | pIC50 | 3 | Yes | |
HDGVZUWMGHDPLU
|
9.4 | IC50 | 2 | — | |
HGGZKXBVGGKUJC
|
9.4 | IC50 | 2 | — | |
OKLOPBKXGZVBCB
|
9.4 | pIC50 | 4 | Yes | |
XHJYBXKCAUZIFW
|
9.4 | pIC50 | 2 | Yes | |
AQRLDBGCWSEIIY
|
9.4 | pIC50 | 3 | Yes | |
LIRHXIGWHONJAQ
|
9.4 | pIC50 | 3 | Yes | |
QMUSHXFQMCVHRH
|
9.4 | pIC50 | 2 | Yes | |
RCFIBNPHKRATBK
|
9.4 | pIC50 | 2 | Yes | |
UYKAYMDFMOZSIG
|
9.4 | pIC50 | 2 | Yes | |
CRPNIZNJBGVBMQ
|
9.4 | pIC50 | 2 | Yes | |
FSSFYFUDWJPZMF
|
9.4 | pIC50 | 2 | Yes | |
OJEWQHUSLNOLBT
|
9.4 | pIC50 | 3 | Yes | |
AECLAEDYDCKFJG
|
9.4 | pIC50 | 2 | Yes | |
KRDCKLXYBSFBNW
|
9.4 | pIC50 | 2 | Yes | |
BNBSDZRWCCHBOZ
|
9.3 | pIC50 | 2 | Yes | |
DRDJJFGPXROAMP
|
9.3 | pIC50 | 3 | Yes | |
HSMBIOOZBSGLTB
|
9.3 | pIC50 | 2 | Yes | |
NUJXPVZUWBELDZ
|
9.3 | pIC50 | 2 | Yes | |
QRWYVPGOSHKJPP
|
9.3 | pIC50 | 3 | Yes | |
SHPJZFRGYYTFJF
|
9.3 | pIC50 | 3 | Yes | |
LONOBJYLFFURAI
|
9.3 | pIC50 | 3 | Yes | |
ROYSOBXGDVHDTQ
|
9.3 | pIC50 | 5 | Yes | |
INXLLPVQCSRCGC
|
9.3 | pIC50 | 2 | Yes | |
ABMQIHFTAMGDJE
|
9.3 | pIC50 | 3 | Yes |