Target Details
| UniProt AC | P49354 |
|---|---|
| Gene Symbol | FNTA |
| Protein Name | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01239 (PPTA) |
Summary
- Multi-target molecules 1,421
- Clinical molecules 1125
- Avg pChEMBL 7.75
KEGG Pathways (1)
Active Molecules (1,421)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OMODHEKCMZABQT
|
7.3 | pIC50 | 2 | Yes | |
SCRKEDSZWRHMLN
|
7.3 | IC50 | 2 | — | |
SKECBVYVVSSXSD
|
7.3 | pIC50 | 2 | Yes | |
PALNUDJZQNISFV
|
7.3 | pIC50 | 2 | Yes | |
GERFWDRHAJVQRY
|
7.3 | pIC50 | 2 | Yes | |
NIWAAOQMMJIQQE
|
7.3 | IC50 | 2 | — | |
UHGZCRVPTZSYOB
|
7.3 | pIC50 | 2 | Yes | |
WLPWQYIANXQUAR
|
7.3 | pIC50 | 2 | Yes | |
DOOYRJLMWIPDFF
|
7.3 | pIC50 | 2 | Yes | |
KGKPSDXDDIJGRA
|
7.3 | IC50 | 2 | — | |
QXMXLXMWARQWNN
|
7.3 | pIC50 | 2 | Yes | |
VRSNOOISIRFSDW
|
7.3 | pIC50 | 2 | Yes | |
WAHSFNMXOHAFIQ
|
7.3 | pIC50 | 2 | Yes | |
YZXGVUSIYCGRQI
|
7.3 | pIC50 | 2 | Yes | |
QXMXLXMWARQWNN
|
7.3 | pIC50 | 2 | Yes | |
XFLDZCZKAVQGOE
|
7.3 | IC50 | 2 | — | |
CKUHCKCWOOAQKN
|
7.3 | pIC50 | 2 | Yes | |
DWTFHVQGFAMPIJ
|
7.3 | pIC50 | 2 | Yes | |
JZSBUEWWLNHSPY
|
7.3 | pIC50 | 2 | Yes | |
KGSICNXNFOBMJP
|
7.3 | pIC50 | 2 | Yes | |
MMVLVRLMGLVJPZ
|
7.3 | pIC50 | 2 | Yes | |
QIQWUVXAQGNSCR
|
7.3 | pIC50 | 2 | Yes | |
XWCMUCOWDZOIAS
|
7.3 | pIC50 | 2 | Yes | |
YJNGMDBYFVYMGU
|
7.3 | IC50 | 2 | — | |
NGWHQWBIMKMHDC
|
7.3 | pIC50 | 3 | Yes | |
OOTPGGWGGFGWFC
|
7.3 | IC50 | 2 | — | |
VAIBMLXNEIEZII
|
7.3 | pIC50 | 2 | Yes | |
ZJDKIZWSAPCYLY
|
7.3 | pIC50 | 2 | Yes | |
QCDHQOJQZWJDKD
|
7.3 | pIC50 | 2 | Yes | |
QFRFAEZUAFKYNV
|
7.3 | pIC50 | 3 | Yes | |
UJBRGSBCWPZFDZ
|
7.3 | pIC50 | 2 | Yes | |
ATJPCVSJAZCTKM
|
7.3 | pIC50 | 2 | Yes | |
BBJDHKUNEILAOY
|
7.3 | IC50 | 2 | — | |
FFALBTXIOBRXDI
|
7.3 | pIC50 | 2 | Yes | |
MHNMEERHZSPWFL
|
7.3 | IC50 | 3 | — | |
MMVLVRLMGLVJPZ
|
7.3 | pIC50 | 2 | Yes | |
PCMOPVSFMUOUFR
|
7.3 | IC50 | 2 | — | |
PKMVDYSKPDHRLR
|
7.3 | pIC50 | 3 | Yes | |
UTKUPTTVIYDTLT
|
7.3 | pIC50 | 2 | Yes | |
VLPFBBPLGMITHP
|
7.3 | pIC50 | 2 | Yes | |
XVWPFYDMUFBHBF
|
7.3 | IC50 | 2 | — | |
BQMDSBZYLBSEIH
|
7.3 | pIC50 | 2 | Yes | |
BWBARWMGJYTEDQ
|
7.3 | pIC50 | 2 | Yes | |
GNEPJAOLPFUJSS
|
7.3 | pIC50 | 2 | Yes | |
VFMUHVILDDZEAG
|
7.3 | pIC50 | 2 | Yes | |
IDHGAQOVWWBGFK
|
7.2 | IC50 | 4 | — | |
GDBOJNVAFLVGKR
|
7.2 | pIC50 | 2 | Yes | |
MYRBTMFPTMIADC
|
7.2 | pIC50 | 2 | Yes | |
MZKNCHCTZBSPNY
|
7.2 | pIC50 | 2 | Yes | |
NNWWMMNANLBUAQ
|
7.2 | pIC50 | 2 | Yes |