Target Details
| UniProt AC | P49354 |
|---|---|
| Gene Symbol | FNTA |
| Protein Name | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01239 (PPTA) |
Summary
- Multi-target molecules 1,421
- Clinical molecules 1125
- Avg pChEMBL 7.75
KEGG Pathways (1)
Active Molecules (1,421)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FLNCVWATJBZKRU
|
7.4 | pIC50 | 2 | Yes | |
IXIKCENTAPEJEA
|
7.4 | pIC50 | 2 | Yes | |
PCFMKLVXKKAJSV
|
7.4 | pIC50 | 2 | Yes | |
PCFMKLVXKKAJSV
|
7.4 | pIC50 | 2 | Yes | |
ABTXIAMOBHCWMR
|
7.4 | pIC50 | 2 | Yes | |
BNESXHDPUFELSD
|
7.4 | pIC50 | 2 | Yes | |
DMSCAHDPEYGXKR
|
7.4 | IC50 | 2 | — | |
GBDDVKMRTGPCDF
|
7.4 | pIC50 | 2 | Yes | |
HASNIZLQJKWUHP
|
7.4 | pIC50 | 2 | Yes | |
MDOOQICNCKEHFW
|
7.4 | pIC50 | 3 | Yes | |
ODTFPKNIFYMEHP
|
7.4 | pIC50 | 2 | Yes | |
PCEQFKLIONHDSE
|
7.4 | pIC50 | 2 | Yes | |
XENZKNOSOFDDED
|
7.4 | pIC50 | 2 | Yes | |
DCVOTMAQSRGQLQ
|
7.4 | pIC50 | 2 | Yes | |
GCZIVFMNASXWTO
|
7.4 | pIC50 | 2 | Yes | |
GJOYCZXIAXQQNR
|
7.4 | pIC50 | 2 | Yes | |
KJDFLBHKZQUEFX
|
7.4 | pIC50 | 2 | Yes | |
MOCUABRQFZUWQK
|
7.4 | pIC50 | 2 | Yes | |
UTMZYAWLRIYYGT
|
7.4 | pIC50 | 2 | Yes | |
CPSSWZSRNFSQCV
|
7.4 | IC50 | 2 | — | |
DPUOYNLDETWCLN
|
7.4 | pIC50 | 2 | Yes | |
FSXYFJWXKIMVFY
|
7.4 | pIC50 | 2 | Yes | |
HFDXBAKHDUJSKS
|
7.4 | pIC50 | 2 | Yes | |
KJSMLERTEOUXOK
|
7.4 | pIC50 | 2 | Yes | |
OPJNGFCKISFMLV
|
7.4 | pIC50 | 2 | Yes | |
UNMKLZBYJNBEEK
|
7.4 | pIC50 | 3 | Yes | |
YRCIPCCRRZWPGD
|
7.4 | pIC50 | 2 | Yes | |
AAXGNXOJOSOUQQ
|
7.4 | pIC50 | 3 | Yes | |
BCRBAAGRYPXBFL
|
7.4 | IC50 | 2 | — | |
MLVPMWIOABZTQP
|
7.4 | pIC50 | 2 | Yes | |
NBWCLOAUIPSQPV
|
7.4 | pIC50 | 2 | Yes | |
URFHMEIWBPJSAJ
|
7.4 | pIC50 | 3 | Yes | |
XCASJHOUQCCHSR
|
7.4 | pIC50 | 2 | Yes | |
DXZIXKOCIQSMJW
|
7.4 | pIC50 | 2 | Yes | |
GFLATSMJZZMJPM
|
7.4 | pIC50 | 2 | Yes | |
GMTZBAHJVUECAM
|
7.4 | pIC50 | 2 | Yes | |
JUOFAUOWWKTUIO
|
7.4 | pIC50 | 2 | Yes | |
KDDZVJQCAMDQTB
|
7.4 | pIC50 | 2 | Yes | |
PYJYSZJNKRTPIY
|
7.4 | IC50 | 2 | — | |
QXMXLXMWARQWNN
|
7.4 | pIC50 | 2 | Yes | |
AYJMTZHIZXFBFE
|
7.4 | pIC50 | 2 | Yes | |
AYVOHKUVBAZLSK
|
7.4 | pIC50 | 2 | Yes | |
DFXJFEAHWLUMQK
|
7.4 | IC50 | 2 | — | |
LQNDTMZXYCNVNE
|
7.4 | pIC50 | 2 | Yes | |
WRTWELJAUYNNMB
|
7.4 | pIC50 | 2 | Yes | |
AQFSLYDVQZALJV
|
7.3 | pIC50 | 2 | Yes | |
DBCXWVGNCLNTQP
|
7.3 | pIC50 | 2 | Yes | |
IMZURFDDENFPKW
|
7.3 | IC50 | 2 | — | |
LVZGQJMNYKYGLS
|
7.3 | pIC50 | 2 | Yes | |
MAXWIYONKRGTOX
|
7.3 | pIC50 | 2 | Yes |