Target Details
| UniProt AC | P49354 |
|---|---|
| Gene Symbol | FNTA |
| Protein Name | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01239 (PPTA) |
Summary
- Multi-target molecules 1,421
- Clinical molecules 1125
- Avg pChEMBL 7.75
KEGG Pathways (1)
Active Molecules (1,421)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WPZXABAVFMGYIS
|
8.1 | pIC50 | 2 | Yes | |
ZMPPPCWXZUURIX
|
8.1 | pIC50 | 2 | Yes | |
CJIVZNOHIDIINJ
|
8.1 | pIC50 | 2 | Yes | |
FCTWBCRRJCWKTE
|
8.1 | pIC50 | 2 | Yes | |
ICFXMOZSPFIDAS
|
8.1 | pIC50 | 2 | Yes | |
SWZGYZRZEHXDAJ
|
8.1 | pIC50 | 2 | Yes | |
UXDWHSLPIYXEQA
|
8.1 | pIC50 | 3 | Yes | |
PBMKCIIZEGBJQL
|
8.1 | IC50 | 2 | — | |
CRZFJHYKXXQOID
|
8.1 | pIC50 | 2 | Yes | |
GZHDTPNNJPPQMX
|
8.1 | Ki | 2 | — | |
MMYMFHIOHNIUSB
|
8.1 | pIC50 | 2 | Yes | |
DEBGEDXBSMFDAS
|
8.1 | IC50 | 2 | — | |
HLPQICVVEMSECL
|
8.1 | pIC50 | 2 | Yes | |
QKWVXFYKJWTMMF
|
8.1 | pIC50 | 2 | Yes | |
QMBOMETUAPMBFM
|
8.1 | pIC50 | 3 | Yes | |
SUHLJVHSQCIBRD
|
8.1 | pIC50 | 3 | Yes | |
RCCUCHCLRYWOAS
|
8.0 | pIC50 | 2 | Yes | |
YZPIHUPBGVJAAS
|
8.0 | pIC50 | 2 | Yes | |
BRCCXAUQKZKZAB
|
8.0 | pIC50 | 2 | Yes | |
COLCNDRDBCLVOC
|
8.0 | IC50 | 2 | — | |
DBWZOKRHHKZPJP
|
8.0 | IC50 | 3 | — | |
MCCIFKLDYHXXJP
|
8.0 | IC50 | 2 | — | |
RMXCVAFRLLKAJD
|
8.0 | pIC50 | 3 | Yes | |
DKBCPWSPMZLASX
|
8.0 | pIC50 | 2 | Yes | |
BVDBXZCOEACWLX
|
8.0 | IC50 | 2 | — | |
CBDOEMKELXJEST
|
8.0 | pIC50 | 2 | Yes | |
FPVFNTHWCRWGPI
|
8.0 | pIC50 | 2 | Yes | |
FQELRMKFQZFXCH
|
8.0 | pIC50 | 2 | Yes | |
GOYDJMAPJITTBZ
|
8.0 | IC50 | 2 | — | |
ISLPXYUADRUJGE
|
8.0 | pIC50 | 2 | Yes | |
IZYCQMKDUPSJSI
|
8.0 | pIC50 | 3 | Yes | |
KMCSNINJDQEUSB
|
8.0 | IC50 | 2 | — | |
LMBPTRXCFXWLRW
|
8.0 | IC50 | 2 | — | |
MDHIWABIFRJJQN
|
8.0 | pIC50 | 2 | Yes | |
PWWOCBOJXZIMPZ
|
8.0 | pIC50 | 2 | Yes | |
QQBJGMOFEGWNEB
|
8.0 | pIC50 | 2 | Yes | |
SPULWNYHMWGKTL
|
8.0 | pIC50 | 2 | Yes | |
UEBNHTSMTQUOQB
|
8.0 | pIC50 | 2 | Yes | |
UQPBEYBGEYZEHF
|
8.0 | IC50 | 4 | — | |
ZORLZQLLRSELQH
|
8.0 | pIC50 | 2 | Yes | |
YDXZCFLYIHUBSR
|
8.0 | pIC50 | 2 | Yes | |
YMZZCTYMIDSJJQ
|
8.0 | pIC50 | 2 | Yes | |
AHPUIZQTTZGXBJ
|
8.0 | pIC50 | 2 | Yes | |
DIDRALNGAJEZDV
|
8.0 | pIC50 | 4 | Yes | |
DLKRWIGCXANSMO
|
8.0 | IC50 | 2 | — | |
DXJRWWRZZPRGJB
|
8.0 | pIC50 | 3 | Yes | |
IPRQDTJTDYDPBX
|
8.0 | pIC50 | 2 | Yes | |
UHGZCRVPTZSYOB
|
8.0 | pIC50 | 2 | Yes | |
VKLQBYODSYOXOK
|
8.0 | pIC50 | 3 | Yes | |
VTTUTHTUYFRALO
|
8.0 | IC50 | 2 | — |