Target Details
| UniProt AC | P49354 |
|---|---|
| Gene Symbol | FNTA |
| Protein Name | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01239 (PPTA) |
Summary
- Multi-target molecules 1,421
- Clinical molecules 1125
- Avg pChEMBL 7.75
KEGG Pathways (1)
Active Molecules (1,421)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PUYMVXRERWLXDU
|
8.2 | pIC50 | 2 | Yes | |
AQTMMHDZTUQGJD
|
8.2 | pIC50 | 3 | Yes | |
DEXSDZQNSUQUAY
|
8.2 | IC50 | 2 | — | |
JVAQVSBUXYDHFX
|
8.2 | pIC50 | 2 | Yes | |
NOCAUXIJQHYHJE
|
8.2 | IC50 | 2 | — | |
OBXLXUGOZZWQOW
|
8.2 | IC50 | 2 | — | |
XRDQKSAFYWAWJI
|
8.2 | IC50 | 2 | — | |
XWUNACODWZDLMP
|
8.2 | pIC50 | 3 | Yes | |
COPRVKYDYTZHGW
|
8.2 | pIC50 | 2 | Yes | |
DDTGELIOCFLYLI
|
8.2 | pIC50 | 2 | Yes | |
MKWMDDYXJPKBRA
|
8.2 | pIC50 | 2 | Yes | |
QJAYXHNDUQQSPN
|
8.2 | pIC50 | 2 | Yes | |
RJMUYANIARJTKU
|
8.2 | pIC50 | 2 | Yes | |
PHGAACKWQSAJHR
|
8.2 | pIC50 | 2 | Yes | |
WLEUBRYSZJGDFY
|
8.2 | IC50 | 4 | — | |
WLEUBRYSZJGDFY
|
8.2 | IC50 | 3 | — | |
BAQAZCQBLRUMRU
|
8.2 | pIC50 | 2 | Yes | |
CGJFRYFIVOQHJK
|
8.2 | pIC50 | 2 | Yes | |
DRIXLVGOZDWKFA
|
8.2 | pIC50 | 2 | Yes | |
FQLPAFFYSWNCAX
|
8.2 | IC50 | 2 | — | |
GXROPRYKIVOUEO
|
8.2 | pIC50 | 2 | Yes | |
HMBVZGUDIZJMIK
|
8.2 | pIC50 | 3 | Yes | |
HQHGMTIPVQADEA
|
8.2 | pIC50 | 2 | Yes | |
ZMGCFGGMTCMSDP
|
8.2 | pIC50 | 2 | Yes | |
ARBOPWPZIKDYTB
|
8.1 | IC50 | 2 | — | |
DGRIIWOHDOZOIX
|
8.1 | pIC50 | 2 | Yes | |
IENQPUVVSDIXCT
|
8.1 | pIC50 | 3 | Yes | |
JOVWTITYEDGJSM
|
8.1 | pIC50 | 2 | Yes | |
JUTCCKPVWGLSCN
|
8.1 | IC50 | 2 | — | |
OIXTWEGQCSRVEN
|
8.1 | pIC50 | 2 | Yes | |
QLRFEPWQAANFLT
|
8.1 | IC50 | 2 | — | |
RHBHKMYAKIXENB
|
8.1 | pIC50 | 2 | Yes | |
CDXIZXQBISVZMK
|
8.1 | pIC50 | 2 | Yes | |
FJIWDNJPYKXVLG
|
8.1 | pIC50 | 2 | Yes | |
KUOCTSJFVHNDDY
|
8.1 | pIC50 | 2 | Yes | |
MTCBWDAIIYFYNS
|
8.1 | IC50 | 2 | — | |
OEAYYCBXEABVGK
|
8.1 | IC50 | 2 | — | |
PJMSBMNZIBDJOM
|
8.1 | pIC50 | 2 | Yes | |
VESCLSDOPNDLRS
|
8.1 | pIC50 | 2 | Yes | |
BKSIKSJVVZGDPT
|
8.1 | pIC50 | 2 | Yes | |
BMAWJYDMAVDMKG
|
8.1 | pIC50 | 2 | Yes | |
CKUAWXYQQWMTHM
|
8.1 | pIC50 | 3 | Yes | |
HMBVZGUDIZJMIK
|
8.1 | pIC50 | 2 | Yes | |
MDBOTFRSILQXBP
|
8.1 | pIC50 | 2 | Yes | |
MOLIDNVFZBNVNE
|
8.1 | pIC50 | 2 | Yes | |
OMXJXAHPPQYWRS
|
8.1 | pIC50 | 2 | Yes | |
QBDQYYQDOAPAPB
|
8.1 | pIC50 | 2 | Yes | |
RISGGZVWVXRFHC
|
8.1 | pIC50 | 2 | Yes | |
TWNBGUAWTJEEOF
|
8.1 | pIC50 | 2 | Yes | |
UOOPOGXXNZHSPG
|
8.1 | pIC50 | 2 | Yes |