Target Details
| UniProt AC | P49354 |
|---|---|
| Gene Symbol | FNTA |
| Protein Name | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01239 (PPTA) |
Summary
- Multi-target molecules 1,421
- Clinical molecules 1125
- Avg pChEMBL 7.75
KEGG Pathways (1)
Active Molecules (1,421)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ARSPPFOBLHMDFX
|
8.3 | pIC50 | 2 | Yes | |
FLFNSORDYCBQRT
|
8.3 | pIC50 | 2 | Yes | |
IWQXXMWFEZGUPJ
|
8.3 | pIC50 | 2 | Yes | |
JFSBDKASCAKCDV
|
8.3 | pIC50 | 2 | Yes | |
POQMRAAOGZQAAM
|
8.3 | pIC50 | 2 | Yes | |
QMCCVNYWKLFKCQ
|
8.3 | IC50 | 2 | — | |
QRZPLNXYFZWRNQ
|
8.3 | pIC50 | 3 | Yes | |
SWFSUXNVVXEJHD
|
8.3 | pIC50 | 2 | Yes | |
SWVWFVRGBYSYCX
|
8.3 | IC50 | 2 | — | |
UHBVRZRMCWMQGX
|
8.3 | pIC50 | 2 | Yes | |
VCBCUVKYTUDCRS
|
8.3 | IC50 | 4 | — | |
DTKKIBZEICDNGH
|
8.3 | Ki | 2 | — | |
JGXPXXUUXXPAIZ
|
8.3 | pIC50 | 2 | Yes | |
MONZTFSZTWQCKH
|
8.3 | pIC50 | 2 | Yes | |
QBDQYYQDOAPAPB
|
8.3 | pIC50 | 2 | Yes | |
RGXWUSMPBUPQSB
|
8.3 | pIC50 | 2 | Yes | |
UGLKTTMREWKECX
|
8.3 | pIC50 | 2 | Yes | |
YCRWTAAJDYJPGL
|
8.3 | pIC50 | 2 | Yes | |
WPANQPAWMQHJEJ
|
8.3 | pIC50 | 4 | Yes | |
FKXKURNMQKQXKJ
|
8.3 | pIC50 | 2 | Yes | |
NSYTZIOXSOGJFP
|
8.3 | pIC50 | 2 | Yes | |
OAERLEDUYZOGEV
|
8.3 | IC50 | 2 | — | |
TWXSHNQCPSUCSH
|
8.3 | IC50 | 2 | — | |
UZEOMOSDTQNLKZ
|
8.3 | pIC50 | 2 | Yes | |
POTOEJFYCBZWMK
|
8.2 | pIC50 | 2 | Yes | |
HUOQFTKEEWWMLS
|
8.2 | pIC50 | 2 | Yes | |
HWYWVGSBHACYHO
|
8.2 | pIC50 | 2 | Yes | |
KDJOWKLMGPUQBA
|
8.2 | pIC50 | 2 | Yes | |
MRONYHYWJWVKKK
|
8.2 | pIC50 | 2 | Yes | |
DNQNJLLRSCYHPU
|
8.2 | pIC50 | 2 | Yes | |
FGDXJSBOTIKISM
|
8.2 | pIC50 | 2 | Yes | |
BJWZXDNEKWSGQH
|
8.2 | IC50 | 2 | — | |
GIGXNNUVDWTCGJ
|
8.2 | pIC50 | 2 | Yes | |
JFUPLVLXDDNRLK
|
8.2 | pIC50 | 2 | Yes | |
JJNUKHXGSMGYPO
|
8.2 | pIC50 | 2 | Yes | |
KJBINAWDNVGVJU
|
8.2 | pIC50 | 2 | Yes | |
LQAKOQWYSFLBMK
|
8.2 | pIC50 | 2 | Yes | |
MKGYPBDRQKFJKZ
|
8.2 | pIC50 | 2 | Yes | |
QQNBNRKLJSPBKX
|
8.2 | pIC50 | 2 | Yes | |
UKMSOESJBYSCKH
|
8.2 | pIC50 | 2 | Yes | |
WDYGFNPGSTZSNU
|
8.2 | pIC50 | 2 | Yes | |
YDEBODDQKWRXPQ
|
8.2 | pIC50 | 2 | Yes | |
ZYJDBHSEWMJVRV
|
8.2 | pIC50 | 2 | Yes | |
FBAYEMRGZYQUMX
|
8.2 | pIC50 | 2 | Yes | |
NCHZWYVOXHDWLS
|
8.2 | pIC50 | 2 | Yes | |
NMLGTGOKSLHKRQ
|
8.2 | pIC50 | 2 | Yes | |
OAOZPXOXMVMQBZ
|
8.2 | pIC50 | 2 | Yes | |
UNRVWOAQHIHREH
|
8.2 | pIC50 | 2 | Yes | |
DXEBREDQSQBFRD
|
8.2 | IC50 | 2 | — | |
GBZJRDYYHMFEPS
|
8.2 | pIC50 | 2 | Yes |