Target Details
| UniProt AC | P49336 |
|---|---|
| Gene Symbol | CDK8 |
| Protein Name | Cyclin-dependent kinase 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 886
- Clinical molecules 10
- Avg pChEMBL 7.54
Associated Diseases (1)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RMOAHCIFLAJLMD
|
7.6 | IC50 | 2 | — | |
UKVIZZGJDGTFIV
|
7.6 | IC50 | 2 | — | |
UXLMSZCUDFXGFP
|
7.6 | IC50 | 3 | — | |
HUKBDNROCCIOGK
|
7.6 | IC50 | 4 | — | |
MKEABIJFHUEATP
|
7.6 | IC50 | 2 | — | |
RPEUBLICACLKCM
|
7.6 | Ki | 2 | — | |
UEMDLSOAXRVEIR
|
7.6 | IC50 | 2 | — | |
APIRNJQTJSYXTA
|
7.6 | IC50 | 2 | — | |
FFCFHBVSGILIJY
|
7.6 | Ki | 17 | — | |
HXESDBWWDYJEJQ
|
7.6 | Ki | 10 | — | |
JCQUAZDMEAWOOT
|
7.6 | IC50 | 3 | — | |
JONQOCAQOVHFAQ
|
7.6 | IC50 | 2 | — | |
PLHUMPJXRHMFFR
|
7.6 | Ki | 28 | — | |
RJAXDQYMJMBDCF
|
7.6 | IC50 | 4 | — | |
UYGYYOIUVFMGKQ
|
7.6 | Ki | 30 | — | |
AMPPIJHFLHITHG
|
7.6 | IC50 | 4 | — | |
MTZSGYFLSTWNDM
|
7.6 | Ki | 2 | — | |
XTBBKBBXJPQUKJ
|
7.6 | Ki | 2 | — | |
AXGBNOWDDQXXDR
|
7.6 | IC50 | 3 | — | |
CPFVIABLSKKULA
|
7.6 | IC50 | 2 | — | |
FKZUVZAFVLLRHB
|
7.6 | IC50 | 2 | — | |
WWGYFGUZQDCDTE
|
7.6 | IC50 | 2 | — | |
XSNUKOJSTFODBN
|
7.6 | IC50 | 2 | — | |
CYLDJPVEBVIXNB
|
7.6 | IC50 | 6 | — | |
DJTZJKJIHWUBGI
|
7.6 | IC50 | 2 | — | |
DXUYKSZGHSMVNI
|
7.5 | IC50 | 2 | — | |
MIELHCGANGLYOP
|
7.5 | IC50 | 2 | — | |
ODUDYGGNMIYVLI
|
7.5 | IC50 | 2 | — | |
PAUXJRUOCRBJHR
|
7.5 | IC50 | 6 | — | |
GQOIDSKRGWWFDU
|
7.5 | IC50 | 2 | — | |
HTOZHWWXFWCYGA
|
7.5 | IC50 | 4 | — | |
OHNXBYACIOVGBQ
|
7.5 | IC50 | 2 | — | |
YCHHLNUILPSKGG
|
7.5 | IC50 | 3 | — | |
MLTSNXSYHSYGAM
|
7.5 | IC50 | 2 | — | |
XHVYRNHFNKLZPA
|
7.5 | IC50 | 4 | — | |
JYHNLDQTJYGLIQ
|
7.5 | IC50 | 2 | — | |
OBXJXHURJISADY
|
7.5 | IC50 | 2 | — | |
PBUIDECYWOLPBK
|
7.5 | Ki | 2 | — | |
DEXAFBASLBZBIA
|
7.5 | IC50 | 2 | — | |
IVMAILZOXLZXTB
|
7.5 | IC50 | 4 | — | |
SUUOJCKRZPQUHP
|
7.5 | IC50 | 2 | — | |
UELJIJLPGZIWDX
|
7.5 | IC50 | 2 | — | |
ASXKBNMXEWJZGS
|
7.5 | IC50 | 2 | — | |
BGVLCUOYRCTJCU
|
7.5 | IC50 | 2 | — | |
DGWFLRMBMMLPMA
|
7.5 | IC50 | 3 | — | |
DQPHCRJDVQHPSA
|
7.5 | Ki | 2 | — | |
GJOXRIYWDHESDF
|
7.5 | Ki | 27 | — | |
JJTYLBBKGQOISV
|
7.5 | Ki | 15 | — | |
QAJPIJHWTGPUNZ
|
7.5 | Ki | 37 | — | |
TZFYFJYOXYWJIK
|
7.5 | IC50 | 4 | — |