Target Details
| UniProt AC | P49336 |
|---|---|
| Gene Symbol | CDK8 |
| Protein Name | Cyclin-dependent kinase 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 886
- Clinical molecules 10
- Avg pChEMBL 7.54
Associated Diseases (1)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZZZRHFQPNAABMT
|
7.8 | IC50 | 2 | — | |
GLZNPLDOIXFNBU
|
7.8 | IC50 | 2 | — | |
IUIMXKRFPHOPLB
|
7.8 | IC50 | 2 | — | |
TZUKIYSPMHRCBN
|
7.8 | IC50 | 2 | — | |
KZPBPRPGCUHTER
|
7.8 | IC50 | 2 | — | |
UVFPZSQALDIFOG
|
7.8 | IC50 | 2 | — | |
LVIYMOOJJGCMCP
|
7.8 | IC50 | 2 | — | |
OSUSJQOYNWQHEC
|
7.8 | IC50 | 2 | — | |
WVPWJZVPSPEJCP
|
7.8 | IC50 | 2 | — | |
NMTSFNXTUCLDKF
|
7.8 | Ki | 2 | — | |
PWYKURSOQPCEIO
|
7.8 | IC50 | 2 | — | |
RXQSXUFJBOKCAT
|
7.8 | IC50 | 3 | — | |
WWSYRAJTUUAHEC
|
7.8 | IC50 | 2 | — | |
XZWGYUDHWRFVLU
|
7.8 | IC50 | 2 | — | |
JZQQXYWMBCHJDE
|
7.7 | IC50 | 2 | — | |
OMXPPLKRCNPLSE
|
7.7 | Kd | 2 | — | |
TVIGYYOJLHHHKZ
|
7.7 | IC50 | 3 | — | |
BJTUXMKSSKKZAW
|
7.7 | Ki | 2 | — | |
GBEUJGXZRJILPH
|
7.7 | IC50 | 2 | — | |
GIVLDIIPJXUCNE
|
7.7 | IC50 | 2 | — | |
GTJWTPSHGINPNN
|
7.7 | IC50 | 2 | — | |
PEUOHMPBTLQKMK
|
7.7 | IC50 | 2 | — | |
WPOFKPTYRRBVST
|
7.7 | IC50 | 3 | — | |
FNIZWTONUSWDQJ
|
7.7 | IC50 | 3 | — | |
AYXVSCVVQIADBF
|
7.7 | Ki | 10 | — | |
BSOKQZFUZVLTAW
|
7.7 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.7 | Ki | 118 | — | |
IKNDNTIDNPFLAC
|
7.7 | IC50 | 2 | — | |
RVKNONNXSNALJV
|
7.7 | IC50 | 21 | — | |
SWANEGKPPCJDTE
|
7.7 | IC50 | 2 | — | |
VCFDMLBPASGZTP
|
7.7 | Ki | 38 | — | |
XNWKXXIGSPPPBH
|
7.7 | Ki | 31 | — | |
ZICLKVKKMGHHDX
|
7.7 | IC50 | 4 | — | |
GRRIIMXGYIQXDB
|
7.7 | IC50 | 2 | — | |
IZIZTVUBBXGCPR
|
7.7 | IC50 | 2 | — | |
WFJJLBVYQIIGHG
|
7.7 | IC50 | 2 | — | |
BOXRYRKZIFAJDP
|
7.7 | Ki | 2 | — | |
MOARLOGPIPTREO
|
7.7 | IC50 | 2 | — | |
PKNQYZOKNCUDHE
|
7.7 | IC50 | 2 | — | |
PXSGYNYFXCHNNR
|
7.7 | IC50 | 2 | — | |
VYWUTAQQVFMHBW
|
7.7 | IC50 | 3 | — | |
KMJBSZNZTUBEMD
|
7.7 | IC50 | 4 | — | |
JIUIKAWQGWJUAQ
|
7.7 | Ki | 2 | — | |
LTDHSYFBXJACGM
|
7.7 | IC50 | 3 | — | |
RHPNLUKAYGCIIG
|
7.7 | Ki | 2 | — | |
VZOLINZYKOLXAC
|
7.7 | IC50 | 2 | — | |
VZOLINZYKOLXAC
|
7.7 | IC50 | 2 | — | |
YBNHQEFUOGXZRC
|
7.7 | Ki | 2 | — | |
IICSXHYHGAAWBA
|
7.6 | IC50 | 3 | — | |
OEHBLKFWGKSFLY
|
7.6 | IC50 | 3 | — |