Target Details
| UniProt AC | P49336 |
|---|---|
| Gene Symbol | CDK8 |
| Protein Name | Cyclin-dependent kinase 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 886
- Clinical molecules 10
- Avg pChEMBL 7.54
Associated Diseases (1)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FZQAZSRDRZGHTP
|
7.9 | IC50 | 3 | — | |
GTCHOWGVVHHKBH
|
7.9 | IC50 | 3 | — | |
KSGZCKSNTAJOJS
|
7.9 | IC50 | 5 | — | |
KSGZCKSNTAJOJS
|
7.9 | IC50 | 2 | — | |
MRPGRAKIAJJGMM
|
7.9 | IC50 | 11 | — | |
QCGCKUCRBUABID
|
7.9 | IC50 | 2 | — | |
RZPBTCAZCIFOKZ
|
7.9 | IC50 | 3 | — | |
VTYUGUKLRVNFAA
|
7.9 | IC50 | 2 | — | |
WLTRIWCDHOZNRP
|
7.9 | IC50 | 14 | — | |
DTNDZQHUJGBYAQ
|
7.9 | IC50 | 4 | — | |
YDCAIQGKZSEZJE
|
7.9 | IC50 | 2 | — | |
CHTMRWQLNNRRFJ
|
7.9 | Ki | 70 | — | |
DQPYZHUAILXFJI
|
7.9 | Ki | 27 | — | |
SRONQUHCRFZABC
|
7.9 | Ki | 28 | — | |
UMTWTCVTRDYHQQ
|
7.9 | Ki | 56 | — | |
BBLKGBHRBXFWHD
|
7.9 | IC50 | 2 | — | |
BDVKKXRTQYBQFJ
|
7.9 | IC50 | 2 | — | |
GEANABGVEPQZHT
|
7.9 | IC50 | 2 | — | |
VWJSHXLEQJGMPN
|
7.9 | IC50 | 2 | — | |
FKSAHKFFMSBYIJ
|
7.9 | IC50 | 4 | — | |
YENIGUGPROEFFL
|
7.9 | IC50 | 3 | — | |
AIOXFJJODLAAIZ
|
7.8 | IC50 | 2 | — | |
DFXPOARIQXPDMN
|
7.8 | Ki | 2 | — | |
FSBMCTDYWXIBLM
|
7.8 | IC50 | 22 | — | |
ILMHDRGZABQLEW
|
7.8 | Ki | 5 | — | |
IQJKHKMDUAVVBY
|
7.8 | IC50 | 4 | — | |
JZJJXQLMEJTQNR
|
7.8 | Ki | 2 | — | |
OVBNODUHLULOMH
|
7.8 | IC50 | 2 | — | |
OYCPRMBVNKLWJN
|
7.8 | IC50 | 2 | — | |
PHXJVRSECIGDHY
|
7.8 | IC50 | 59 | — | |
PMWYYXJYUKFILR
|
7.8 | Ki | 2 | — | |
CYUUDYXCDKUQSM
|
7.8 | IC50 | 2 | — | |
HIHDNOVBJSCLBP
|
7.8 | IC50 | 4 | — | |
WBHQPLISMLDBLH
|
7.8 | IC50 | 4 | — | |
HOFCDHUGGVZPCY
|
7.8 | IC50 | 2 | — | |
MSMMOWGLNAZZPB
|
7.8 | IC50 | 2 | — | |
WAKJOUVIVRSNKI
|
7.8 | IC50 | 3 | — | |
BGVARKGXOUTVCM
|
7.8 | IC50 | 2 | — | |
BWDARHFPTQIHIU
|
7.8 | IC50 | 2 | — | |
DFFPNDMXOZUGLU
|
7.8 | IC50 | 4 | — | |
FVBDIBZJXLGYED
|
7.8 | Ki | 2 | — | |
GHHDMQJYDMQTDY
|
7.8 | IC50 | 2 | — | |
IWZSHWBGHQBIML
|
7.8 | IC50 | 2 | — | |
JLTBOCSFMNSLFH
|
7.8 | Ki | 9 | — | |
LHIUZPIDLZYPRL
|
7.8 | IC50 | 8 | — | |
MUKGYZFIZLFCGL
|
7.8 | IC50 | 3 | — | |
RKUKAACYUCUJEE
|
7.8 | Ki | 58 | — | |
WGBUCZXTNTVPDM
|
7.8 | IC50 | 2 | — | |
XUFLBSMTYMFOQH
|
7.8 | Ki | 43 | — | |
YSBNRVRADYMQNP
|
7.8 | Ki | 2 | — |