Target Details
| UniProt AC | P49336 |
|---|---|
| Gene Symbol | CDK8 |
| Protein Name | Cyclin-dependent kinase 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 886
- Clinical molecules 10
- Avg pChEMBL 7.54
Associated Diseases (1)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FXPJXSGYDSEBFL
|
8.1 | IC50 | 3 | — | |
MEFSUICXZJQPFL
|
8.1 | IC50 | 2 | — | |
BREHUJBZTIHZHE
|
8.1 | IC50 | 2 | — | |
CKYHGLQQZNNTMG
|
8.1 | IC50 | 2 | — | |
LQZKADWTXZGRQF
|
8.1 | IC50 | 2 | — | |
NQHGDUGVQSAKOR
|
8.1 | IC50 | 3 | — | |
FNIZWTONUSWDQJ
|
8.1 | IC50 | 4 | — | |
HAEDHIQEQOEOHP
|
8.1 | IC50 | 2 | — | |
HGGIFNLRPYEBQB
|
8.1 | IC50 | 2 | — | |
IIIQUEYXCDAEGD
|
8.1 | IC50 | 2 | — | |
MTLHRGZTWNKSBV
|
8.1 | Ki | 5 | — | |
RTYCSOHJUAWUAK
|
8.1 | IC50 | 3 | — | |
XTKSMYZRQMTSMS
|
8.1 | IC50 | 3 | — | |
FXPMUAXYMIDCCK
|
8.0 | IC50 | 3 | — | |
FZKLIVJJIDYMJT
|
8.0 | IC50 | 2 | — | |
PVYAJYQKDXIVSJ
|
8.0 | IC50 | 3 | — | |
BAXXRIGYAIVSDC
|
8.0 | IC50 | 3 | — | |
MXPUHLQPJSPPAS
|
8.0 | IC50 | 4 | — | |
NAVWVDFKHIIIDK
|
8.0 | IC50 | 2 | — | |
WSHKPIHTYDQNDK
|
8.0 | IC50 | 3 | — | |
HUJOQYSJVADDBN
|
8.0 | IC50 | 3 | — | |
HUKOPIUVSYNTMX
|
8.0 | IC50 | 2 | — | |
ISZRWOBBNIOIMU
|
8.0 | IC50 | 3 | — | |
UXSVDQPKNXQICD
|
8.0 | IC50 | 3 | — | |
ZLPZSHJTTWBCCD
|
8.0 | IC50 | 2 | — | |
AKMUJHSPPZVLAJ
|
8.0 | IC50 | 2 | — | |
AUXBXQOZTPVFRD
|
8.0 | IC50 | 2 | — | |
CFJWYFBHISDVGI
|
8.0 | Ki | 2 | — | |
DKXHSOUZPMHNIZ
|
8.0 | Ki | 51 | Yes | |
FAAVFBBBVCMQSM
|
8.0 | IC50 | 3 | — | |
KPJPEYWXGRKBQF
|
8.0 | IC50 | 2 | — | |
LSZGQBKMSJOVAW
|
8.0 | IC50 | 2 | — | |
NAMIJFMAPMJBGN
|
8.0 | Ki | 2 | — | |
NTCPUSCJDOSUEX
|
8.0 | Kd | 2 | — | |
VDZNZFZOXXXJPD
|
8.0 | Ki | 2 | — | |
OTDAVQICJQMEMA
|
8.0 | IC50 | 2 | — | |
FRILIGULNDONDJ
|
8.0 | IC50 | 2 | — | |
FGWWXXXOMYTMPD
|
8.0 | IC50 | 2 | — | |
GLDUWDZPOUGRKS
|
8.0 | IC50 | 2 | — | |
LOOFFGPDPOEAMT
|
8.0 | IC50 | 2 | — | |
NLYNEHVCNWNHNP
|
8.0 | IC50 | 2 | — | |
ORKBDPRQJKIQTC
|
8.0 | IC50 | 3 | — | |
PQCODRGUOJKOCC
|
8.0 | IC50 | 2 | — | |
VVABWBULVNCYQT
|
8.0 | IC50 | 3 | — | |
XEKMGJCVLWWIGJ
|
8.0 | IC50 | 2 | — | |
AIOQFYKTFBMYKM
|
8.0 | IC50 | 2 | — | |
OUOQXEFHIIUYNW
|
8.0 | IC50 | 2 | — | |
UYMBYVWSBPECIF
|
7.9 | IC50 | 2 | — | |
CUQBBHUITNFLKO
|
7.9 | IC50 | 2 | — | |
DQGVTHXNAGEYRW
|
7.9 | IC50 | 3 | — |