Target Details
| UniProt AC | P49336 |
|---|---|
| Gene Symbol | CDK8 |
| Protein Name | Cyclin-dependent kinase 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 886
- Clinical molecules 10
- Avg pChEMBL 7.54
Associated Diseases (1)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QHMOZKVAGIEXJR
|
8.3 | IC50 | 2 | — | |
WSCCAHKPFOILSF
|
8.3 | IC50 | 2 | — | |
IKWJMCVFMQHZBD
|
8.3 | IC50 | 2 | — | |
IZRGMKQUICGMNO
|
8.3 | IC50 | 2 | — | |
NCIRPZWSTPFOGW
|
8.3 | IC50 | 2 | — | |
QLMIHYKKDODCRC
|
8.3 | IC50 | 3 | — | |
MMTZCTUXVCJRSF
|
8.2 | IC50 | 2 | — | |
MUQRYGJXSGWQNK
|
8.2 | IC50 | 3 | — | |
QBMVSTFFMINBKY
|
8.2 | IC50 | 2 | — | |
CALOLERUXQBROP
|
8.2 | IC50 | 4 | — | |
OJIQEAIHEGJBFE
|
8.2 | IC50 | 3 | — | |
ZDQFWXPJQYVSMT
|
8.2 | IC50 | 3 | — | |
CBSAOWNMAJFXSH
|
8.2 | IC50 | 2 | — | |
LUSRSUWSGVIMEM
|
8.2 | IC50 | 2 | — | |
ONVYPVVYNXLFQK
|
8.2 | IC50 | 4 | — | |
MRSAAOGDVNDADH
|
8.2 | IC50 | 2 | — | |
RTMDKYGKOKLIFN
|
8.2 | IC50 | 3 | — | |
BUGVQNZMIPEMTK
|
8.2 | IC50 | 3 | — | |
GADFZYLJRACWPZ
|
8.2 | IC50 | 3 | — | |
OZZYAWZFNLQDDK
|
8.2 | IC50 | 2 | — | |
RONMYLLIYUXIFC
|
8.2 | IC50 | 3 | — | |
SONQRTMFYJXMDT
|
8.2 | IC50 | 2 | — | |
SPFRZBQLMQBEJM
|
8.2 | IC50 | 2 | — | |
UXENHMYWTQJELH
|
8.2 | IC50 | 2 | — | |
VTROAQBXWNPBTF
|
8.2 | IC50 | 2 | — | |
ZHXAYCNHSHNBBO
|
8.2 | IC50 | 2 | — | |
PAPUAQAWYXMVQI
|
8.2 | IC50 | 2 | — | |
FLCVCISWDBTPRS
|
8.2 | IC50 | 2 | — | |
IKRSLQINMKBFSM
|
8.2 | IC50 | 2 | — | |
BUVVQUOSYFAZRC
|
8.2 | Ki | 2 | — | |
JXXSSUSJGPUFLD
|
8.2 | IC50 | 2 | — | |
PWPUINQCPPKTQG
|
8.2 | IC50 | 3 | — | |
TYCOTTAYUVNCMS
|
8.2 | IC50 | 3 | — | |
VYEMYSAPQYFLBU
|
8.2 | IC50 | 3 | — | |
AGXNDPDCEGWAIY
|
8.1 | IC50 | 2 | — | |
YRNKBHIBUTYIHE
|
8.1 | IC50 | 3 | — | |
ZYLCPTQVVVTGSL
|
8.1 | IC50 | 2 | — | |
CESJOILAQXASKZ
|
8.1 | IC50 | 2 | — | |
CRKQBJZCCHKEGI
|
8.1 | Ki | 20 | — | |
DCBOUGQYASVENA
|
8.1 | Ki | 2 | — | |
GJKVMXDBPDDFHI
|
8.1 | Ki | 27 | — | |
HZPACYSNLOCDLW
|
8.1 | Ki | 48 | — | |
LBFYQISQYCGDDW
|
8.1 | IC50 | 7 | — | |
MJQYFYSOJQOQNT
|
8.1 | IC50 | 2 | — | |
NMCZSPLOTVSBEU
|
8.1 | IC50 | 2 | — | |
ODRITQGYYWHQGM
|
8.1 | IC50 | 4 | — | |
PBCVBUZBZRHMQH
|
8.1 | Ki | 2 | — | |
RHIYLWIQYIFQGZ
|
8.1 | IC50 | 2 | — | |
BIPBLKIGJHZBND
|
8.1 | IC50 | 2 | — | |
CMEFLKIFRPLMJK
|
8.1 | IC50 | 5 | — |