Target Details
| UniProt AC | P49336 |
|---|---|
| Gene Symbol | CDK8 |
| Protein Name | Cyclin-dependent kinase 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 886
- Clinical molecules 10
- Avg pChEMBL 7.54
Associated Diseases (1)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RDVHTWWUICGUOA
|
8.5 | IC50 | 3 | — | |
NKRTZXOPWXKKJM
|
8.5 | IC50 | 2 | — | |
QDMGVWHKVHTJPB
|
8.5 | IC50 | 2 | — | |
BNCMMIOUWWXGGZ
|
8.4 | IC50 | 2 | — | |
OOWVGRDBRZFHTD
|
8.4 | IC50 | 2 | — | |
RLVURTZJQZIODI
|
8.4 | IC50 | 2 | — | |
XGWLARMAWLGPNP
|
8.4 | IC50 | 2 | — | |
DMIAAAUSYPPGHE
|
8.4 | IC50 | 3 | — | |
LVQICVKIHBQMRT
|
8.4 | IC50 | 4 | — | |
PIMQWRZWLQKKBJ
|
8.4 | IC50 | 36 | — | |
UIMLSKNJMYHPHO
|
8.4 | IC50 | 2 | — | |
ZLJBWVWHTDCWFO
|
8.4 | IC50 | 3 | — | |
CLEGDJQQHUTCOW
|
8.4 | Ki | 43 | — | |
HEIMUHPANNQRGV
|
8.4 | IC50 | 2 | — | |
KTWBYGUSEYSRND
|
8.4 | Ki | 28 | — | |
SUJFSWHSHYPYRU
|
8.4 | IC50 | 2 | — | |
YRFOQHHFWYWAST
|
8.4 | IC50 | 22 | — | |
KOZWDURZSCBPDP
|
8.4 | IC50 | 4 | — | |
SOGOUJPVOZWDFQ
|
8.4 | IC50 | 2 | — | |
XJFPWEGWVPIYIH
|
8.4 | IC50 | 2 | — | |
YXVVCWWWIWRJKH
|
8.4 | IC50 | 2 | — | |
CPYTXFOZVKULHY
|
8.4 | IC50 | 2 | — | |
FPCNFWJGROIGLW
|
8.4 | IC50 | 2 | — | |
ISQMHRGAJWVQET
|
8.4 | IC50 | 4 | — | |
NFUKLMJHYQPDNT
|
8.4 | IC50 | 3 | — | |
NALGKDPHSMQYFA
|
8.3 | IC50 | 3 | — | |
QXGOBEONKUXLNG
|
8.3 | IC50 | 4 | — | |
TUIAGTUBZBTEHN
|
8.3 | IC50 | 2 | — | |
YSULJPQXWIYNMJ
|
8.3 | IC50 | 2 | — | |
ZYRJLEBRYYKEIM
|
8.3 | IC50 | 2 | — | |
FXSAYAHGTCKXRP
|
8.3 | IC50 | 2 | — | |
JCBMNKGAZMDVPY
|
8.3 | IC50 | 3 | — | |
ASBSOCYVAYZKGS
|
8.3 | IC50 | 3 | — | |
KVXMBXJEXMWXLQ
|
8.3 | IC50 | 4 | — | |
VNKGRMAIKMWRDN
|
8.3 | IC50 | 2 | — | |
WJORYPIALAWPKB
|
8.3 | IC50 | 2 | — | |
ZFKIMLOZPZTQJP
|
8.3 | IC50 | 2 | — | |
OARDWOBZBKIVNO
|
8.3 | IC50 | 2 | — | |
XGPSXEHFMOUIKO
|
8.3 | IC50 | 2 | — | |
DNQPOMIKYILRSQ
|
8.3 | IC50 | 2 | — | |
DWRDPMAVWSBVOL
|
8.3 | IC50 | 3 | — | |
HAMWSFRMPKMULI
|
8.3 | IC50 | 2 | — | |
PGLBZRZEQTVNDN
|
8.3 | IC50 | 2 | — | |
PTVQSGXLKJJLML
|
8.3 | IC50 | 2 | — | |
RJZUGXNAXUOKRX
|
8.3 | IC50 | 3 | — | |
TYGRNYUURMQGDD
|
8.3 | Ki | 2 | — | |
VPJXPDLMACOGIZ
|
8.3 | IC50 | 3 | — | |
WDARYLSSWBWVCU
|
8.3 | Ki | 49 | — | |
WNVQODMEPIULDK
|
8.3 | IC50 | 3 | — | |
ZBGLBBSOTJOVJO
|
8.3 | IC50 | 5 | — |