Target Details
| UniProt AC | P49336 |
|---|---|
| Gene Symbol | CDK8 |
| Protein Name | Cyclin-dependent kinase 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 886
- Clinical molecules 10
- Avg pChEMBL 7.54
Associated Diseases (1)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IMJBJHNFFBDGFG
|
8.7 | IC50 | 3 | — | |
KDZLCWBDQVILHC
|
8.7 | IC50 | 2 | — | |
QXNLDTWVURNIRW
|
8.7 | IC50 | 2 | — | |
VVEGARMQKNYDID
|
8.7 | Ki | 24 | — | |
ZPUYWMRULPSNOR
|
8.7 | IC50 | 4 | — | |
CGELUDGKNGUGSC
|
8.7 | IC50 | 2 | — | |
FFAWVGUBSMGFJF
|
8.7 | IC50 | 2 | — | |
FKZUTCUBVKIYSO
|
8.7 | IC50 | 2 | — | |
ZRCRKSJBXVRFPW
|
8.7 | IC50 | 4 | — | |
MPEULGZDXWQEGW
|
8.7 | IC50 | 4 | — | |
GQWMRZZYHJLZFL
|
8.6 | IC50 | 3 | — | |
PJGCBELMRGKAMA
|
8.6 | IC50 | 3 | — | |
ZNMSRFYDOSAZLZ
|
8.6 | IC50 | 3 | — | |
DYILYHVZADZHDJ
|
8.6 | IC50 | 3 | — | |
GBYCDBFSAXCWDG
|
8.6 | IC50 | 2 | — | |
GCMACTQBSNIQGT
|
8.6 | IC50 | 3 | — | |
HCFPJWWQXYFZLK
|
8.6 | IC50 | 2 | — | |
RRAVJRJCTBGPCG
|
8.6 | IC50 | 3 | — | |
SRMSEKPITZQWRD
|
8.6 | IC50 | 3 | — | |
WFXNKOHCSFBJLW
|
8.6 | IC50 | 2 | — | |
CTLOWNSSFKLIFJ
|
8.6 | IC50 | 2 | — | |
MCKPYPWHBUXLEZ
|
8.6 | Ki | 21 | — | |
MOIRAYXVFLWFTA
|
8.6 | IC50 | 2 | — | |
PNURMDJXHPDCNM
|
8.6 | IC50 | 2 | — | |
QOZPYXBSOMOOTN
|
8.6 | IC50 | 2 | — | |
SYYLWEQOPOZEHZ
|
8.6 | IC50 | 2 | — | |
VTQQYBGURNVVFE
|
8.6 | Ki | 17 | — | |
ZHMXUOBSYMVTBS
|
8.6 | IC50 | 2 | — | |
ADNJUAOLUJJJHY
|
8.6 | IC50 | 4 | — | |
BBXDHOXWXXMPLZ
|
8.6 | IC50 | 2 | — | |
YZQXGSFVWSAYFN
|
8.6 | IC50 | 3 | — | |
CBZADZPBIPFAOG
|
8.6 | IC50 | 2 | — | |
FKGDVUYRXAGOSW
|
8.6 | IC50 | 2 | — | |
YQYMAYUQUXDUNP
|
8.6 | IC50 | 3 | — | |
JJIQBYGSBIHLSR
|
8.6 | IC50 | 2 | — | |
UDRFCFLSQTXHOX
|
8.6 | IC50 | 2 | — | |
UWTMXZFDTBHJPH
|
8.6 | IC50 | 3 | — | |
WLNUDRFOSHWBNG
|
8.6 | IC50 | 3 | — | |
FFAWVGUBSMGFJF
|
8.5 | IC50 | 2 | — | |
MOFLRZQOEVPOMU
|
8.5 | IC50 | 3 | — | |
MRWUTTXEVGWLFR
|
8.5 | IC50 | 3 | — | |
NCPSMBVBKJXJPP
|
8.5 | IC50 | 3 | — | |
PWDLXPJQFNVTNL
|
8.5 | IC50 | 3 | — | |
RKTPHHQXNCHBCF
|
8.5 | IC50 | 2 | — | |
SKKRZILJUKYLJS
|
8.5 | Ki | 25 | — | |
CEWROMVZNURIEF
|
8.5 | IC50 | 4 | — | |
ICKPROJHWZPXBO
|
8.5 | IC50 | 2 | — | |
LLNFBSQVFXOHIC
|
8.5 | IC50 | 2 | — | |
BDZJCURBFSRLAZ
|
8.5 | IC50 | 2 | — | |
PSLTXNZIRUGQOG
|
8.5 | IC50 | 3 | — |