Target Details
| UniProt AC | P49336 |
|---|---|
| Gene Symbol | CDK8 |
| Protein Name | Cyclin-dependent kinase 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 886
- Clinical molecules 10
- Avg pChEMBL 7.54
Associated Diseases (1)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
URNZTLZSAVLTIZ
|
8.9 | Ki | 26 | — | |
LYQFHPSZCYRZHH
|
8.9 | IC50 | 2 | — | |
MRADTWDZEMCUJY
|
8.9 | IC50 | 2 | — | |
PBJOOQQRNPULJG
|
8.9 | IC50 | 2 | — | |
ROZDFHHCJWWRPT
|
8.9 | IC50 | 2 | — | |
VEFPQLMCHLYXLM
|
8.9 | IC50 | 2 | — | |
IRVDFMPPZOLHDV
|
8.9 | IC50 | 4 | — | |
BIBOVMGNFAPEJA
|
8.8 | IC50 | 4 | — | |
FNIZWTONUSWDQJ
|
8.8 | IC50 | 4 | — | |
GYCMNQWPVCUOPZ
|
8.8 | IC50 | 3 | — | |
HAUGVIAEKSQIGA
|
8.8 | IC50 | 4 | — | |
HJPLVEAFJZGECM
|
8.8 | IC50 | 2 | — | |
ODPGGGTTYSGTGO
|
8.8 | Kd | 153 | — | |
ORKTZIGUWHVTBU
|
8.8 | IC50 | 2 | — | |
SZLHAVCVTGQMJV
|
8.8 | IC50 | 2 | — | |
URTXFNMSFMYZRA
|
8.8 | IC50 | 4 | — | |
BUWYJLHXEGUSQE
|
8.8 | IC50 | 2 | — | |
GAENHTLOUWWIEL
|
8.8 | IC50 | 2 | — | |
GHUGJYUFZCOUPW
|
8.8 | IC50 | 2 | — | |
LFAHWMOZPVCJAY
|
8.8 | IC50 | 8 | — | |
PNSCLJRKJNHORL
|
8.8 | IC50 | 3 | — | |
QCFROKOAPICCRK
|
8.8 | IC50 | 2 | — | |
RKOMZOWWZMLCAU
|
8.8 | IC50 | 2 | — | |
ZMWFSXAKXCNWGH
|
8.8 | IC50 | 2 | — | |
BGYVWFZMYBWCNY
|
8.8 | Ki | 30 | — | |
FAYAUAZLLLJJGH
|
8.8 | Ki | 36 | Yes | |
IUIDISNVIBKQQL
|
8.8 | IC50 | 3 | — | |
LAYMXNJSUDFINH
|
8.8 | IC50 | 3 | — | |
MNEPGHKCEKEYEZ
|
8.8 | IC50 | 2 | — | |
NJPWCTYVEJIQBM
|
8.8 | Ki | 72 | — | |
RFBPWKMQWSIPEO
|
8.8 | Ki | 28 | — | |
SLKCVFPEQGHNSI
|
8.8 | Ki | 29 | — | |
SOZZTNWQGFCMCH
|
8.8 | IC50 | 2 | — | |
WDBRDGNVWBDCLI
|
8.8 | IC50 | 2 | — | |
YEIMDRLHFGJVBY
|
8.8 | IC50 | 2 | — | |
ZHMXUOBSYMVTBS
|
8.8 | IC50 | 2 | — | |
YLJSAFSDGFNKAC
|
8.8 | IC50 | 4 | — | |
BUWYJLHXEGUSQE
|
8.8 | IC50 | 2 | — | |
JJCQVMCBHSWKAC
|
8.8 | IC50 | 2 | — | |
ZVSGCPGPQNLKLU
|
8.8 | IC50 | 3 | — | |
COZFAYYFONTRSA
|
8.7 | IC50 | 2 | — | |
OQOHDKVDMBADIN
|
8.7 | IC50 | 2 | — | |
ORKTZIGUWHVTBU
|
8.7 | IC50 | 2 | — | |
RUWVXGZGSKEPIG
|
8.7 | IC50 | 2 | — | |
NZIVBHCIRGQSRI
|
8.7 | IC50 | 3 | — | |
YWHDHVUZZPMSQD
|
8.7 | IC50 | 3 | — | |
ITRXYWUAAUJIKA
|
8.7 | IC50 | 4 | — | |
BACOSPUGMHOGST
|
8.7 | IC50 | 2 | — | |
BIIVYFLTOXDAOV
|
8.7 | Ki | 31 | — | |
DOLVPVSWTLFZMQ
|
8.7 | Ki | 17 | — |