Target Details
| UniProt AC | P49336 |
|---|---|
| Gene Symbol | CDK8 |
| Protein Name | Cyclin-dependent kinase 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 886
- Clinical molecules 10
- Avg pChEMBL 7.54
Associated Diseases (1)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HIFKRZORZOSOFC
|
9.7 | IC50 | 4 | — | |
RUNGUDNTFGOPRL
|
9.7 | IC50 | 2 | — | |
YFLGXECHDXSDGM
|
9.7 | IC50 | 2 | — | |
AFQAFERZBGFZRQ
|
9.6 | IC50 | 4 | — | |
QXPHUXPNTWFKOR
|
9.6 | IC50 | 4 | — | |
FFNTZJOKBZFDQL
|
9.5 | IC50 | 4 | — | |
XALHKECHUOZBNB
|
9.5 | IC50 | 3 | — | |
ZKUPHELZBDXDNL
|
9.4 | IC50 | 2 | — | |
BOEKPVCGEJPQQI
|
9.4 | IC50 | 2 | — | |
HVEXJKQESNIDLM
|
9.4 | IC50 | 10 | — | |
VFKCKMKPKIUZOF
|
9.4 | IC50 | 2 | — | |
IRVDFMPPZOLHDV
|
9.4 | IC50 | 4 | — | |
AIRVMUGRIFXGRE
|
9.3 | IC50 | 3 | — | |
YHBCYQIXVZFFIV
|
9.3 | IC50 | 4 | — | |
DXZXMWGMIHOZIS
|
9.3 | IC50 | 2 | — | |
VWCSZVWZRTZNCH
|
9.3 | IC50 | 8 | — | |
IBDRMDVDKFGXHV
|
9.3 | IC50 | 2 | — | |
CUSUZSREAOLZQQ
|
9.3 | IC50 | 3 | — | |
BKXGAUBREGVJQM
|
9.2 | IC50 | 3 | — | |
LFUBEMFSRYUGLW
|
9.2 | IC50 | 3 | — | |
MIRNBYWEECOSRO
|
9.2 | IC50 | 3 | — | |
QJIOPOJQZXHHEW
|
9.2 | IC50 | 2 | — | |
RDJKDXOOXNKSCO
|
9.2 | IC50 | 2 | — | |
WGVVTSMURAVCGU
|
9.2 | IC50 | 2 | — | |
RUFKAIQMVPWHCQ
|
9.2 | IC50 | 4 | — | |
IXRCZLGBPPMVSP
|
9.2 | IC50 | 9 | — | |
OWZWPBNBNAGTCG
|
9.2 | IC50 | 2 | — | |
PQVDKUZOKMCUSV
|
9.2 | IC50 | 3 | — | |
FUMCKNCUEAQHCV
|
9.1 | Ki | 103 | — | |
SPRWPVWJJFDDRK
|
9.1 | IC50 | 2 | — | |
MUDJOIVQYIMGDK
|
9.1 | IC50 | 2 | — | |
DFYVDBLGPYTIAT
|
9.1 | IC50 | 2 | — | |
RJTQBPCQZQSZFF
|
9.1 | IC50 | 9 | — | |
FWXRRJODQJLGKY
|
9.0 | IC50 | 3 | — | |
CDVRWNCFJKEAKY
|
9.0 | IC50 | 3 | — | |
LMIPCDJYZXYYLQ
|
9.0 | IC50 | 5 | — | |
NBSJZWFDNFWQDN
|
9.0 | IC50 | 29 | — | |
RDLVYLCFTGIOIP
|
9.0 | IC50 | 2 | — | |
ZHMXUOBSYMVTBS
|
9.0 | IC50 | 2 | — | |
ALVRKNONSXJKLX
|
9.0 | IC50 | 2 | — | |
CNIOXRPTZYLDHI
|
9.0 | IC50 | 3 | — | |
SSFIJHKAGFQDEJ
|
9.0 | IC50 | 2 | — | |
ULMZCAWRPCELOE
|
9.0 | IC50 | 3 | — | |
UODXTGBFBIFREQ
|
9.0 | IC50 | 8 | Yes | |
WULUGQONDYDNKY
|
9.0 | IC50 | 5 | — | |
ZOOJEBLXLLZVIR
|
9.0 | IC50 | 4 | — | |
JTKNAVYDXHDJAQ
|
8.9 | IC50 | 2 | — | |
LGJRNXYDSYLXSJ
|
8.9 | IC50 | 2 | — | |
PBJOOQQRNPULJG
|
8.9 | IC50 | 2 | — | |
VEWOEDYMHKDFEL
|
8.9 | IC50 | 2 | — |