Target Details
| UniProt AC | P49137 |
|---|---|
| Gene Symbol | MAPKAPK2 |
| Protein Name | MAP kinase-activated protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 124
- Clinical molecules 11
- Avg pChEMBL 6.99
KEGG Pathways (8)
Active Molecules (124)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LYZZMBVBMJMPFE
|
6.2 | IC50 | 2 | — | |
NJPWCTYVEJIQBM
|
6.2 | Ki | 72 | — | |
USHMNZBDAOGLMB
|
6.2 | Ki | 26 | — | |
KJDMOEPAJHJNBM
|
6.2 | IC50 | 2 | — | |
FNHKPVJBJVTLMP
|
6.2 | Kd | 29 | — | |
ADMFLILDQJSEIK
|
6.1 | Ki | 72 | — | |
JFGACSUTAMZDKC
|
6.1 | Ki | 2 | — | |
JMCCHRFGZMNODA
|
6.1 | IC50 | 2 | — | |
MLGGUGPIWDHBAI
|
6.1 | Ki | 33 | — | |
RKKIDHHGKNGTQI
|
6.1 | Ki | 28 | — | |
XIOOJUQFJYPVLA
|
6.1 | Ki | 17 | — | |
ULXXDDBFHOBEHA
|
6.1 | Kd | 15 | Yes | |
VUQDZGWRLHHYTB
|
6.1 | IC50 | 2 | — | |
YQKSNDNARJQAHP
|
6.1 | Ki | 12 | — | |
BCBAEHQTYTYENT
|
6.0 | IC50 | 2 | — | |
JKFQIDJSSIINNY
|
6.0 | IC50 | 2 | — | |
LQVXSNNAFNGRAH
|
6.0 | IC50 | 33 | Yes | |
IBGLGMOPHJQDJB
|
6.0 | Kd | 8 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JMCCHRFGZMNODA
|
6.0 | IC50 | 2 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
LKUJDAHYLPICSE
|
6.0 | Ki | 24 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
SZMOXKFQHCNMQZ
|
6.0 | IC50 | 2 | — |