Target Details
| UniProt AC | P49137 |
|---|---|
| Gene Symbol | MAPKAPK2 |
| Protein Name | MAP kinase-activated protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 124
- Clinical molecules 11
- Avg pChEMBL 6.99
KEGG Pathways (8)
Active Molecules (124)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MIKAKZKNMYZLDX
|
7.1 | Ki | 42 | — | |
RLAJOHAIIACFAM
|
7.1 | IC50 | 13 | Yes | |
ZLCBGFVBDKXPBZ
|
7.1 | IC50 | 2 | — | |
ZQUFPLLWPVGSOW
|
7.1 | IC50 | 2 | — | |
DIJIJDANNOSBAG
|
7.0 | IC50 | 2 | — | |
URPBNNONUNUVHW
|
7.0 | IC50 | 2 | — | |
VWNROJWIQIWFSP
|
7.0 | IC50 | 2 | — | |
VVVVSXKJECZPRY
|
6.9 | IC50 | 2 | — | |
WWFURUYYQWIHRV
|
6.8 | IC50 | 2 | — | |
HJSVRZBFKFCGAZ
|
6.8 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
6.8 | IC50 | 408 | — | |
QAQKNZRNOQBKRE
|
6.8 | IC50 | 2 | — | |
USORQDCKXRFILP
|
6.8 | IC50 | 2 | — | |
YLQOELRYUQBERL
|
6.7 | IC50 | 2 | — | |
GWODBBFDCZIKBY
|
6.7 | IC50 | 2 | — | |
FISPOMCKBOYLEG
|
6.7 | IC50 | 2 | — | |
NKGLJTITEFZKAN
|
6.7 | Ki | 35 | — | |
XWXSNJQHZKOICN
|
6.7 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
6.6 | Kd | 289 | Yes | |
JCFJQIHDZHHMQT
|
6.6 | Ki | 42 | — | |
UDFDIIVNIYWXDM
|
6.6 | Ki | 74 | — | |
VSHQPGVRRHIKDU
|
6.6 | IC50 | 2 | — | |
ZJFVUVKJGZKTKC
|
6.6 | IC50 | 2 | — | |
XJJYJNMNYDNXNO
|
6.6 | IC50 | 23 | — | |
DUGXSNHFGBPCPM
|
6.6 | IC50 | 2 | — | |
KCXYHUJEGPMBKM
|
6.6 | IC50 | 2 | — | |
QAQKNZRNOQBKRE
|
6.5 | IC50 | 2 | — | |
ZGBAJMQHJDFTQJ
|
6.5 | Kd | 15 | — | |
GIEOFRPQGSGOLC
|
6.5 | IC50 | 2 | — | |
MMWVUKRVNHSCOU
|
6.5 | IC50 | 2 | — | |
PGQVIPWLMNSOCQ
|
6.5 | IC50 | 2 | — | |
SBFPHSVZEXSHTL
|
6.5 | Ki | 62 | — | |
VFESYYJORSLMBC
|
6.5 | IC50 | 2 | — | |
GPXKVULNYYNGDP
|
6.4 | IC50 | 4 | — | |
LYADGAGFYYXXIO
|
6.4 | IC50 | 82 | — | |
DQHGXHGUNOSYSE
|
6.4 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
6.4 | IC50 | 49 | Yes | |
NVNJXYOVWGMPAO
|
6.4 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
6.4 | Kd | 599 | — | |
DKXHSOUZPMHNIZ
|
6.3 | IC50 | 51 | Yes | |
PHXJVRSECIGDHY
|
6.3 | Kd | 59 | — | |
DKNUPRMJNUQNHR
|
6.3 | Kd | 33 | — | |
BQPLWJRDSDNGNE
|
6.3 | Ki | 16 | — | |
BZQVWTDKMSTNBU
|
6.3 | IC50 | 2 | — | |
LCBAQTCTQXHTJG
|
6.3 | IC50 | 9 | — | |
NYZNNKMKRXQWHA
|
6.3 | IC50 | 2 | — | |
NYZNNKMKRXQWHA
|
6.3 | IC50 | 2 | — | |
ZBNZXTGUTAYRHI
|
6.3 | Kd | 102 | Yes | |
HLFUJFUWDSXIPK
|
6.2 | IC50 | 2 | — | |
JTRXEPCDEVNYPE
|
6.2 | IC50 | 5 | — |