Target Details
| UniProt AC | P49137 |
|---|---|
| Gene Symbol | MAPKAPK2 |
| Protein Name | MAP kinase-activated protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 124
- Clinical molecules 11
- Avg pChEMBL 6.99
KEGG Pathways (8)
Active Molecules (124)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FYSRKRZDBHOFAY
|
9.5 | Kd | 8 | — | |
CZJALLIMKKSCNX
|
9.0 | IC50 | 2 | — | |
MJQUKUIDCUNAAB
|
8.7 | IC50 | 4 | — | |
BTFCCPKDGZFGPR
|
8.4 | IC50 | 3 | — | |
BEYORXSIIKUPCA
|
8.3 | IC50 | 2 | — | |
TXYKBKYDFZQOCB
|
8.3 | IC50 | 2 | — | |
UQQRUYAIZCVJMP
|
8.3 | IC50 | 2 | — | |
ZRAANXMCPIIUKV
|
8.3 | IC50 | 2 | — | |
CMWRPDHVGMHLSZ
|
8.3 | IC50 | 22 | — | |
XQRUWZMHPKNIDA
|
8.2 | IC50 | 2 | — | |
FLEAYYMORDPWAJ
|
8.2 | Ki | 90 | — | |
SAZVRXTVWZAHBI
|
8.2 | IC50 | 4 | — | |
YDELNSXADYPQGS
|
8.2 | IC50 | 15 | Yes | |
BKMFUDJYEMHEKH
|
8.2 | IC50 | 2 | — | |
SBVVPLRDGQGTMO
|
8.2 | IC50 | 2 | — | |
ISLMQWLFRPLLLI
|
8.1 | IC50 | 2 | — | |
VZGXJTZKPDEJGJ
|
8.1 | IC50 | 2 | — | |
OWFLADWRSCINST
|
8.1 | IC50 | 30 | — | |
RDCWVMUIPUMVKS
|
8.0 | IC50 | 2 | — | |
RGWMWOOWHJUGFL
|
8.0 | IC50 | 2 | — | |
VQQDOYPJOLNJQP
|
8.0 | IC50 | 2 | — | |
ZYTDQGRQFPNBGA
|
7.9 | IC50 | 2 | — | |
FRZMEKOENCSLON
|
7.8 | IC50 | 2 | — | |
OVJIHFBAXJKTRF
|
7.8 | IC50 | 2 | — | |
BEMNJULZEQTDJY
|
7.8 | Kd | 8 | — | |
JPOSFPUHBHRUAX
|
7.7 | IC50 | 40 | Yes | |
ZMELOYOKMZBMRB
|
7.7 | Kd | 4 | — | |
FEAAGBKEHOIVOC
|
7.7 | IC50 | 2 | — | |
SBRNUAKQBCFNDP
|
7.7 | IC50 | 2 | — | |
FQPQMJULRZINPV
|
7.7 | IC50 | 2 | — | |
IJNGXROUMFEKDB
|
7.6 | Ki | 39 | — | |
KKYABQBFGDZVNQ
|
7.6 | Kd | 4 | — | |
MFPICHSQTLJIFK
|
7.5 | IC50 | 2 | — | |
JJQNDXCUJRPPDT
|
7.5 | IC50 | 2 | — | |
TUZYUHMHEXTLNB
|
7.5 | IC50 | 2 | — | |
WJYGDQYYYZYICM
|
7.5 | IC50 | 2 | — | |
LRZYYIZFBXFSJB
|
7.5 | IC50 | 69 | — | |
MWKSRKSEWLRPBL
|
7.4 | Kd | 1075 | — | |
FGQLPUTYZYTKLO
|
7.4 | IC50 | 2 | — | |
CJLVRCRBVMSXBQ
|
7.4 | IC50 | 2 | — | |
LVKGEKFNCBTKTM
|
7.4 | IC50 | 2 | — | |
AWZFCQRICMFIES
|
7.3 | IC50 | 9 | Yes | |
RAVOJDKMDLUTLW
|
7.2 | IC50 | 2 | — | |
DIVVQJIIRBQSMU
|
7.2 | IC50 | 2 | — | |
WOSKHXYHFSIKNG
|
7.2 | Kd | 24 | — | |
NNQMSHWOTYMSDC
|
7.2 | IC50 | 3 | — | |
LNMRSSIMGCDUTP
|
7.2 | Kd | 13 | — | |
WKRRYRSXQAPECL
|
7.1 | IC50 | 2 | — | |
DXXJDEVFDVVIGG
|
7.1 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.1 | Ki | 118 | — |