Target Details
| UniProt AC | P48736 |
|---|---|
| Gene Symbol | PIK3CG |
| Protein Name | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF19710 (PIK3CG_ABD) |
Summary
- Multi-target molecules 2,398
- Clinical molecules 104
- Avg pChEMBL 7.16
KEGG Pathways (14)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Inositol phosphate metabolism
- Kaposi sarcoma-associated herpesvirus infection
- Metabolic pathways
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Salmonella infection
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (2,398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NLRPOLHEDYFDBC
|
8.0 | IC50 | 3 | — | |
MPVZERIWUAYICQ
|
8.0 | IC50 | 3 | — | |
AWKBWQVKZBUMPV
|
8.0 | IC50 | 3 | — | |
BGNRHJBZCKJOLD
|
8.0 | IC50 | 3 | — | |
CGJYZCCLUUIRAJ
|
8.0 | Ki | 4 | — | |
CYAPSTHKVSVUQB
|
8.0 | IC50 | 2 | — | |
DEYMNPBPRBGNRS
|
8.0 | IC50 | 3 | — | |
DWZAEMINVBZMHQ
|
8.0 | IC50 | 6 | — | |
FCNPPPJJIYEWFA
|
8.0 | IC50 | 4 | — | |
GZWUFUZDDITKGF
|
8.0 | IC50 | 6 | — | |
IFPHRQQBRZZIOQ
|
8.0 | Kd | 8 | — | |
IZHWRLKLKIUFPI
|
8.0 | IC50 | 4 | — | |
JQSQDPXQHCJTQC
|
8.0 | IC50 | 4 | — | |
KZFJGEOZCGZDAA
|
8.0 | IC50 | 3 | — | |
MWXOKLKTIOEEPK
|
8.0 | IC50 | 3 | — | |
NIWBUWMZKOEJTN
|
8.0 | IC50 | 7 | — | |
NLZNQTSAEGRBEQ
|
8.0 | IC50 | 8 | — | |
QLGKYVWPTGEGNH
|
8.0 | IC50 | 4 | — | |
RGNZNWVPZKJPFW
|
8.0 | IC50 | 5 | — | |
VDOAMMJTSVNAQH
|
8.0 | IC50 | 4 | — | |
VSYBLIHWVCIUHC
|
8.0 | IC50 | 3 | — | |
YWFOHQFLGQVFIB
|
8.0 | IC50 | 9 | — | |
MMLRSHHXXNXWTM
|
8.0 | Ki | 4 | — | |
NBADQPVOAILYHQ
|
7.9 | IC50 | 3 | — | |
NJXDVWJTIOHBGS
|
7.9 | IC50 | 2 | — | |
XEGNSLLNQAWKBA
|
7.9 | IC50 | 3 | — | |
CICFFAJMTOTWDF
|
7.9 | IC50 | 5 | — | |
FFRDFQZNAIEKKG
|
7.9 | IC50 | 3 | — | |
FSPSBPWQYZGGSM
|
7.9 | IC50 | 2 | — | |
HFDGVAZLABKEEV
|
7.9 | IC50 | 4 | — | |
HMCXLHKQRBBRRQ
|
7.9 | Ki | 5 | — | |
ILHMXWRSMGUCKC
|
7.9 | IC50 | 4 | — | |
ITUBWSOGJQVWCJ
|
7.9 | Ki | 5 | — | |
JDTLYBGUQBBSSW
|
7.9 | IC50 | 3 | — | |
MAXHGWQUDVMRJX
|
7.9 | IC50 | 4 | — | |
OFOXQNICEHYXRI
|
7.9 | IC50 | 2 | — | |
PRMGBZXKGUBORE
|
7.9 | IC50 | 3 | — | |
REQOWEPXNXAPLK
|
7.9 | IC50 | 2 | — | |
SYUHGFRIKWMPPV
|
7.9 | Ki | 5 | — | |
SYUHGFRIKWMPPV
|
7.9 | Ki | 5 | — | |
XQDCEYRYQNFRMX
|
7.9 | IC50 | 4 | — | |
XSYSZSQGLRMKHF
|
7.9 | IC50 | 5 | — | |
YPMWYFVHFHAVSY
|
7.9 | IC50 | 5 | — | |
YXRVSHHKBCULEI
|
7.9 | Ki | 5 | — | |
JCVPRCJMVAWOBT
|
7.9 | IC50 | 3 | — | |
RLHVVFZFOUAZRI
|
7.9 | IC50 | 3 | — | |
URYMFNIQUUIFIY
|
7.9 | IC50 | 3 | — | |
MMOOFFFQYJLTLQ
|
7.9 | IC50 | 3 | — | |
UHSGKZKFUUFRPH
|
7.9 | IC50 | 4 | — | |
VHCSLWRCKYDLOT
|
7.9 | IC50 | 4 | — |