Target Details
| UniProt AC | P48736 |
|---|---|
| Gene Symbol | PIK3CG |
| Protein Name | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF19710 (PIK3CG_ABD) |
Summary
- Multi-target molecules 2,398
- Clinical molecules 104
- Avg pChEMBL 7.16
KEGG Pathways (14)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Inositol phosphate metabolism
- Kaposi sarcoma-associated herpesvirus infection
- Metabolic pathways
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Salmonella infection
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (2,398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JNQFWBSHMGXTQX
|
8.2 | IC50 | 6 | — | |
KUGIFHQBIIHRIZ
|
8.2 | Ki | 5 | — | |
NQCGNJZLLGMACO
|
8.2 | IC50 | 4 | — | |
NRQJNWMHLPKGKI
|
8.2 | Ki | 2 | — | |
NSTFOXCDXMJUGH
|
8.2 | IC50 | 3 | — | |
OHZHBEQIRGURAO
|
8.2 | Ki | 5 | — | |
QQBVZBSMGUVONA
|
8.2 | IC50 | 5 | — | |
SUGVMHZDZMFCQJ
|
8.1 | IC50 | 2 | — | |
ZEZJZRDUSAWOET
|
8.1 | IC50 | 2 | — | |
XDXZHIQVJAQRGY
|
8.1 | IC50 | 5 | — | |
XWTGOBYAMGRVHH
|
8.1 | IC50 | 2 | — | |
YHUNTIUERLPKIG
|
8.1 | IC50 | 5 | — | |
RTXWPOABAGXULX
|
8.1 | IC50 | 6 | — | |
DQEGKWHMQYJUKR
|
8.1 | IC50 | 5 | — | |
DSBJBOOMYLWTSO
|
8.1 | IC50 | 4 | — | |
GUXYVZVGGMEFRP
|
8.1 | IC50 | 3 | — | |
HWQOBXLEMHPNMF
|
8.1 | IC50 | 2 | — | |
IMXXTFKFHMPFMA
|
8.1 | Ki | 4 | — | |
JBMPVRPUGHDUOL
|
8.1 | IC50 | 2 | — | |
LJLOTRKTBODGRQ
|
8.1 | Ki | 4 | — | |
NAIYZJSIJREIKA
|
8.1 | IC50 | 4 | — | |
NGGCUTXLGFVQRS
|
8.1 | IC50 | 3 | — | |
NXMKJFZABAEHHG
|
8.1 | IC50 | 4 | — | |
OZKKRHXRCMWNID
|
8.1 | IC50 | 3 | — | |
QDYDLDKGDBEEOL
|
8.1 | IC50 | 3 | — | |
RCBNWWLBZCYILT
|
8.1 | IC50 | 5 | — | |
SQWZFLMPDUSYGV
|
8.1 | IC50 | 11 | — | |
SQWZFLMPDUSYGV
|
8.1 | IC50 | 8 | — | |
SYUHGFRIKWMPPV
|
8.1 | Ki | 5 | — | |
WNLWNUNVLRWGBW
|
8.1 | Ki | 4 | — | |
XESSMGMYMDVIMA
|
8.1 | IC50 | 3 | — | |
XFGGNFBJRMXYAG
|
8.1 | IC50 | 4 | — | |
XTHMHKVQVQAVJS
|
8.1 | IC50 | 3 | — | |
GWNBFGJNUNUOOI
|
8.1 | IC50 | 17 | — | |
RTARVPHTCQRSDW
|
8.1 | IC50 | 7 | Yes | |
TVUPSIBSWDXJGQ
|
8.1 | IC50 | 4 | — | |
BLFHBZZOKOBYDV
|
8.1 | IC50 | 3 | — | |
DKVYWIZHXFHHNQ
|
8.1 | IC50 | 5 | — | |
PESHAFCSMREEAN
|
8.1 | IC50 | 6 | — | |
QVQLSVCCQONRIO
|
8.1 | IC50 | 4 | — | |
XHMVOBSFHGIYQZ
|
8.1 | IC50 | 4 | — | |
OJFOWKCXUALRQN
|
8.1 | IC50 | 5 | — | |
RCQPOVDRJDMKAO
|
8.1 | IC50 | 3 | — | |
YBCNWDQUEDROIU
|
8.1 | IC50 | 3 | — | |
MYIWJCONSHUYIA
|
8.1 | IC50 | 4 | — | |
XDXZHIQVJAQRGY
|
8.1 | IC50 | 5 | — | |
DLFVITASTHEQDC
|
8.1 | Ki | 4 | — | |
DYLZJJGYKQIVGK
|
8.1 | Ki | 4 | — | |
DZRQGNOLDZNGKA
|
8.1 | Ki | 5 | — | |
FUDRVRQHDVLJRT
|
8.1 | IC50 | 3 | — |