Target Details
| UniProt AC | P48736 |
|---|---|
| Gene Symbol | PIK3CG |
| Protein Name | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF19710 (PIK3CG_ABD) |
Summary
- Multi-target molecules 2,398
- Clinical molecules 104
- Avg pChEMBL 7.16
KEGG Pathways (14)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Inositol phosphate metabolism
- Kaposi sarcoma-associated herpesvirus infection
- Metabolic pathways
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Salmonella infection
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (2,398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QVCHABKSWSKVFX
|
8.7 | IC50 | 4 | — | |
TYTHLOGWHWLWET
|
8.7 | IC50 | 4 | — | |
XDLYKKIQACFMJG
|
8.7 | Ki | 6 | — | |
DZBXWGPFVTUJJO
|
8.7 | Ki | 4 | — | |
CTMXQXVWTYALGC
|
8.7 | IC50 | 4 | — | |
CVSBXKYUXXFEGL
|
8.7 | IC50 | 4 | — | |
DOBMLLWIKWJZDR
|
8.7 | IC50 | 4 | — | |
FGZCLHINZBWLRN
|
8.7 | IC50 | 2 | — | |
IFIUXKIVTAKIHT
|
8.7 | Ki | 4 | — | |
KYZLRDASIUNFBY
|
8.7 | IC50 | 5 | — | |
LCMHSLJJLJYDPS
|
8.7 | Ki | 2 | — | |
LOBJMCQPMNBKQW
|
8.7 | IC50 | 4 | — | |
TZFMCSSETKBUSI
|
8.7 | IC50 | 5 | — | |
VYPWROGLWNYKDD
|
8.7 | Ki | 2 | — | |
ZMFSLMFEFNPUMJ
|
8.7 | IC50 | 5 | — | |
HLTLYKPFSSMNIF
|
8.7 | IC50 | 6 | — | |
BHEMPSVJQFJQIN
|
8.7 | Ki | 5 | — | |
DJWGTNCIAUYYCQ
|
8.7 | IC50 | 4 | — | |
KFNBJCXUFADQNW
|
8.7 | IC50 | 4 | — | |
OCQKCCHSJMAUAS
|
8.7 | IC50 | 2 | — | |
KFBBYMDWDSZYSP
|
8.7 | IC50 | 2 | — | |
ASXTXORHWGOEKM
|
8.6 | IC50 | 4 | — | |
QBNCLHVZCGFCOS
|
8.6 | IC50 | 4 | — | |
RPSYNNOLAXEZAD
|
8.6 | IC50 | 2 | — | |
BCYRIDCXNMUOGH
|
8.6 | IC50 | 2 | — | |
MYQDIPJMQYEWIZ
|
8.6 | Ki | 5 | — | |
YKIWXNATSYCOKT
|
8.6 | IC50 | 7 | Yes | |
YKPMNBJYASHWAN
|
8.6 | IC50 | 5 | — | |
BITYGNDFPWCLCP
|
8.6 | IC50 | 2 | — | |
BLCVYWUNXXAHGY
|
8.6 | Ki | 4 | — | |
CTMJHHLZQLYKLF
|
8.6 | IC50 | 4 | — | |
HYIDZNMZGFEUTQ
|
8.6 | IC50 | 4 | — | |
KDSLANAJQYLHMO
|
8.6 | IC50 | 7 | — | |
OMXQWLDNOXGCSM
|
8.6 | IC50 | 2 | — | |
VAEUIPVISAJITP
|
8.6 | IC50 | 2 | — | |
CBZPCOUPBNLTKW
|
8.6 | IC50 | 4 | — | |
VFRMCSHREULMEB
|
8.6 | IC50 | 4 | — | |
BBRINJUWZRLWKK
|
8.6 | IC50 | 5 | — | |
ZOKVMFNJBPBZCE
|
8.6 | IC50 | 7 | — | |
WBYSXNKZTPYYPM
|
8.5 | IC50 | 3 | — | |
CXTUBZFXIDPAQC
|
8.5 | IC50 | 5 | — | |
DJGGTMUWVGIFOX
|
8.5 | IC50 | 2 | — | |
DPHFLPMHQWTKGY
|
8.5 | IC50 | 3 | — | |
PJBHWJZJLJZHAY
|
8.5 | IC50 | 4 | — | |
QCMFYOKICDMTNU
|
8.5 | IC50 | 4 | — | |
QVDJLIIRGGPQQJ
|
8.5 | IC50 | 2 | — | |
YPRWSTYMGINCCO
|
8.5 | IC50 | 2 | — | |
JUMHBOXYBKXAMA
|
8.5 | IC50 | 3 | — | |
PRXYMLOSAFSKGK
|
8.5 | IC50 | 2 | — | |
YQGHFKNCOZCKKN
|
8.5 | IC50 | 5 | — |