Target Details
| UniProt AC | P48736 |
|---|---|
| Gene Symbol | PIK3CG |
| Protein Name | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF19710 (PIK3CG_ABD) |
Summary
- Multi-target molecules 2,398
- Clinical molecules 104
- Avg pChEMBL 7.16
KEGG Pathways (14)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Inositol phosphate metabolism
- Kaposi sarcoma-associated herpesvirus infection
- Metabolic pathways
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Salmonella infection
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (2,398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JCXVWMWEFKRQCE
|
8.9 | IC50 | 3 | — | |
KRJCGMRLWBVONG
|
8.9 | IC50 | 4 | — | |
KVKANZTYGYFKQY
|
8.9 | IC50 | 3 | — | |
LSPJWTULWKYRTQ
|
8.9 | IC50 | 6 | — | |
YLPQMLSKPUQHLB
|
8.9 | IC50 | 6 | — | |
YXDZBGGLBWHPEB
|
8.9 | IC50 | 4 | — | |
ZAWKCTQNKKDNMQ
|
8.9 | IC50 | 4 | — | |
ZTXDHUWPUMVZCM
|
8.9 | IC50 | 4 | — | |
BLNZPYYVWACTDG
|
8.9 | IC50 | 2 | — | |
CZHFAPKIYABWLB
|
8.9 | IC50 | 2 | — | |
GQPHDBXDJOKWED
|
8.9 | IC50 | 3 | — | |
PKEPKQMDLXYSKW
|
8.9 | IC50 | 2 | — | |
QYVUEMYLTHEUNN
|
8.9 | IC50 | 3 | — | |
SDQPODDUDFEPDG
|
8.9 | IC50 | 3 | — | |
BHFJVMZATJXYCO
|
8.9 | IC50 | 3 | — | |
FEHPMLVVSQNYOF
|
8.9 | IC50 | 7 | — | |
HTSSZLURDMBMPC
|
8.9 | IC50 | 2 | — | |
JHCGWQGKIHGVDU
|
8.9 | IC50 | 4 | — | |
JRWUQSVWSWEGLW
|
8.9 | IC50 | 3 | — | |
KDYQDNYXUAAXIW
|
8.9 | IC50 | 3 | — | |
RQZYVAOSDVOURA
|
8.9 | IC50 | 4 | — | |
RZMAPGTVSWFYCK
|
8.9 | IC50 | 5 | — | |
XCOQTFFMFTWVMC
|
8.9 | IC50 | 4 | — | |
ZWZBXYCUIUOCOO
|
8.9 | IC50 | 4 | — | |
CBDQDYXZWIQXDD
|
8.9 | IC50 | 3 | — | |
ZHBRIUFPBZTXAU
|
8.9 | IC50 | 2 | — | |
AICUMEFERAKQDF
|
8.8 | IC50 | 3 | — | |
HZKFGLSKAKKBBZ
|
8.8 | IC50 | 3 | — | |
PZHYYDQKVVSTEG
|
8.8 | IC50 | 4 | — | |
QWPSEEVUQYTULG
|
8.8 | IC50 | 4 | — | |
TWMIPMSAUTYVGK
|
8.8 | IC50 | 4 | — | |
VAZGJQAKGVIDTE
|
8.8 | IC50 | 2 | — | |
VRJUJTMBOARYOG
|
8.8 | IC50 | 3 | — | |
DYIDODGTFZZZOS
|
8.8 | IC50 | 4 | — | |
KPHKHHHLIKEDLQ
|
8.8 | IC50 | 5 | — | |
NMZOQFREGVBPSH
|
8.8 | IC50 | 6 | — | |
RQLVMAYHFPSXMR
|
8.8 | IC50 | 4 | — | |
XLRIOJGDWOEVMT
|
8.8 | IC50 | 4 | — | |
ZGOADLIMIODLBG
|
8.8 | IC50 | 3 | — | |
CPUXOJVJEJZOSP
|
8.8 | IC50 | 6 | — | |
RAJKNXSUPLWLOY
|
8.8 | IC50 | 3 | — | |
XDLYKKIQACFMJG
|
8.8 | Ki | 6 | — | |
ZSEKNBCKQHQTBI
|
8.8 | IC50 | 4 | — | |
BDCVYSXEEZFOSI
|
8.8 | IC50 | 2 | — | |
IVCWAKFADVSCLD
|
8.8 | IC50 | 2 | — | |
GFOJWGYPLGSKOJ
|
8.8 | Ki | 2 | — | |
IEDGFXCUFJCEAP
|
8.8 | IC50 | 6 | — | |
LCVQUFNGYSNDJN
|
8.8 | IC50 | 5 | — | |
KSQGUTYIJILXDH
|
8.7 | IC50 | 8 | — | |
FHOXICOTPQTJOQ
|
8.7 | Ki | 6 | Yes |