Target Details
| UniProt AC | P48736 |
|---|---|
| Gene Symbol | PIK3CG |
| Protein Name | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF19710 (PIK3CG_ABD) |
Summary
- Multi-target molecules 2,398
- Clinical molecules 104
- Avg pChEMBL 7.16
KEGG Pathways (14)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Inositol phosphate metabolism
- Kaposi sarcoma-associated herpesvirus infection
- Metabolic pathways
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Salmonella infection
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (2,398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BNXOEOMQSLPCKM
|
9.1 | IC50 | 3 | — | |
FZLQVDKBOUEZHS
|
9.1 | IC50 | 4 | — | |
IUKKLFSDRNELCN
|
9.1 | IC50 | 4 | — | |
LLUGOCWVLNJQNI
|
9.1 | IC50 | 4 | — | |
NHFRWRZPNNFBRN
|
9.1 | IC50 | 3 | — | |
PDUCWDNFFQBFEQ
|
9.1 | IC50 | 4 | — | |
RNKHOYDAZIEJFF
|
9.1 | IC50 | 4 | — | |
TWLBPEXRIJIDLQ
|
9.1 | IC50 | 3 | — | |
UCWFGTHMIDAVDE
|
9.1 | IC50 | 4 | — | |
VLRSVMBPXWKSNE
|
9.1 | IC50 | 4 | — | |
XDWSNPNGAFALHJ
|
9.1 | IC50 | 4 | — | |
YAOHUGMVFAJBNE
|
9.1 | IC50 | 4 | — | |
DNWLWWRXENCXEL
|
9.0 | Ki | 4 | — | |
DVLVYFPEVHXTKT
|
9.0 | IC50 | 6 | — | |
BEUQXVWXFDOSAQ
|
9.0 | Ki | 8 | — | |
IKUIGBXUTOOMRZ
|
9.0 | Ki | 6 | — | |
CYXPQVSTQNRNSH
|
9.0 | IC50 | 3 | — | |
DHEKPZQWFVQYSO
|
9.0 | IC50 | 3 | — | |
HXALBTBBYYKFPZ
|
9.0 | IC50 | 2 | — | |
IIZVKFYZFQTGEB
|
9.0 | Ki | 2 | — | |
KLMZZLVCEDUTEA
|
9.0 | Ki | 6 | — | |
KRJCGMRLWBVONG
|
9.0 | IC50 | 4 | — | |
KUGIFHQBIIHRIZ
|
9.0 | Ki | 5 | — | |
LQTYGHZRBUVRMR
|
9.0 | IC50 | 6 | — | |
MFYQUMRHYXKIOO
|
9.0 | IC50 | 4 | — | |
NKNADNLRHUVIAR
|
9.0 | IC50 | 2 | — | |
NTZMWNKORQPPBL
|
9.0 | IC50 | 4 | — | |
QVMAMHTWFZGLDH
|
9.0 | IC50 | 2 | — | |
SFTPPASPRIXXIN
|
9.0 | IC50 | 4 | — | |
SMSOEZUYBOCTCT
|
9.0 | IC50 | 4 | — | |
TYTHLOGWHWLWET
|
9.0 | IC50 | 4 | — | |
UCWFGTHMIDAVDE
|
9.0 | IC50 | 4 | — | |
UUXKXNLWIZYSGT
|
9.0 | IC50 | 4 | — | |
UVTRLGWLUDWQGP
|
9.0 | IC50 | 2 | — | |
VGBZVXNIRCSRBK
|
9.0 | IC50 | 3 | — | |
XPHSYMMHKWHMBV
|
9.0 | IC50 | 2 | — | |
YXGZTQDPLYDOCC
|
9.0 | IC50 | 4 | — | |
YZBYWHCDBQFVFZ
|
9.0 | IC50 | 2 | — | |
ZCRLGLTZPXORIX
|
9.0 | IC50 | 2 | — | |
AHNACMAJVLLNSG
|
9.0 | Ki | 4 | — | |
FLUPYHUXCIWKAE
|
9.0 | IC50 | 4 | — | |
GFTIJVHUHAMPLS
|
9.0 | IC50 | 4 | — | |
NHOGIGRHHZKFTF
|
9.0 | IC50 | 4 | — | |
RVJDAOWTYAVAHK
|
9.0 | IC50 | 4 | — | |
TZUURZCAUFJVTJ
|
9.0 | IC50 | 4 | — | |
WKECSELYDBZHQV
|
9.0 | IC50 | 5 | — | |
OWTOSKMKJXQHMU
|
8.9 | IC50 | 3 | — | |
DHEKPZQWFVQYSO
|
8.9 | IC50 | 4 | — | |
IKNJUYUINPOVDE
|
8.9 | IC50 | 4 | — | |
IKNJUYUINPOVDE
|
8.9 | IC50 | 4 | — |