Target Details
| UniProt AC | P48736 |
|---|---|
| Gene Symbol | PIK3CG |
| Protein Name | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF19710 (PIK3CG_ABD) |
Summary
- Multi-target molecules 2,398
- Clinical molecules 104
- Avg pChEMBL 7.16
KEGG Pathways (14)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Inositol phosphate metabolism
- Kaposi sarcoma-associated herpesvirus infection
- Metabolic pathways
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Salmonella infection
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (2,398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SVSSPHFLEURYPE
|
7.3 | IC50 | 3 | — | |
UDDJJHILDQDTBM
|
7.3 | IC50 | 8 | — | |
UIAOVNUDKCZSHU
|
7.3 | IC50 | 2 | — | |
UOORQSPLBHUQDQ
|
7.3 | IC50 | 4 | — | |
XBZDKDNYELJFTM
|
7.3 | IC50 | 5 | — | |
AYAJXNDPUHQQND
|
7.3 | IC50 | 2 | — | |
DDNDFDDGMCJGHM
|
7.3 | IC50 | 2 | — | |
FGCNFUVIPKIWLZ
|
7.3 | IC50 | 2 | — | |
ONJSIGPCPAOGNJ
|
7.3 | Ki | 4 | — | |
WUZRDHWCBDKJTL
|
7.3 | IC50 | 3 | — | |
XUWNECGLJFPCFS
|
7.3 | IC50 | 2 | — | |
ZNOQCQOSJQSWLD
|
7.3 | IC50 | 3 | — | |
ZNOQCQOSJQSWLD
|
7.3 | IC50 | 3 | — | |
AQPXZIOUXMMPJH
|
7.3 | IC50 | 3 | — | |
BLLWLBULZYSIAH
|
7.3 | IC50 | 4 | — | |
GFPPJADRSAPASM
|
7.3 | IC50 | 2 | — | |
JUEPBEIBFLRQSU
|
7.3 | IC50 | 4 | — | |
KHDSNMCNVGLJEF
|
7.3 | IC50 | 2 | — | |
WJXACEILBUSAPK
|
7.3 | IC50 | 3 | — | |
XVCFFNKOIUPASX
|
7.3 | IC50 | 2 | — | |
AJRVMUXGCPDPOT
|
7.3 | IC50 | 8 | — | |
CQPIITBUFCLJQW
|
7.3 | IC50 | 8 | — | |
FYSONCGCYHZETE
|
7.3 | IC50 | 2 | — | |
JDZSJMYXUCQNLL
|
7.3 | IC50 | 3 | — | |
LGRMHOXGTNEFAW
|
7.3 | IC50 | 3 | — | |
LUEFAVVZVXRANQ
|
7.3 | IC50 | 2 | — | |
UATSBNOGNFUSGY
|
7.3 | IC50 | 3 | — | |
VMLVXCSOPRPIDI
|
7.3 | IC50 | 3 | — | |
FBFHUGMVRQBPIQ
|
7.3 | IC50 | 4 | — | |
HGVNLRPZOWWDKD
|
7.3 | IC50 | 7 | — | |
KCNCCZCAVYLQAH
|
7.3 | IC50 | 3 | — | |
KXKADLQRHDFGBR
|
7.3 | IC50 | 8 | — | |
LEWJWUJNURRNQY
|
7.3 | IC50 | 4 | — | |
OVMBAIROGFJDTQ
|
7.3 | IC50 | 3 | — | |
UPQKAJYEZWCPJY
|
7.3 | IC50 | 3 | — | |
XBGGERTXBDEQIK
|
7.3 | IC50 | 3 | — | |
XEBRAMSBPJUGET
|
7.3 | Ki | 5 | — | |
YOGHJOPHCBCAKS
|
7.3 | IC50 | 3 | — | |
ZXONVJJRRBXWDX
|
7.3 | IC50 | 3 | — | |
ADLJEZREHNJMCU
|
7.3 | IC50 | 6 | — | |
BIFBJBYMVYPTPW
|
7.3 | IC50 | 4 | — | |
DISXGKPKWGNTKB
|
7.3 | IC50 | 4 | — | |
DSQJVZCCWLGHTH
|
7.3 | IC50 | 2 | — | |
FDJSQHVHCVOQLN
|
7.3 | IC50 | 3 | — | |
HYZJEDZJBWGLFY
|
7.3 | IC50 | 3 | — | |
JLAZWUFUZDVBSK
|
7.3 | IC50 | 2 | — | |
LIUSADRVCKXVIA
|
7.3 | Ki | 5 | — | |
PJPYMAJZJCYLKR
|
7.3 | IC50 | 3 | — | |
SUIQWWVKWMJPIF
|
7.3 | IC50 | 2 | — | |
UIHWUCKQDZWWKN
|
7.3 | IC50 | 2 | — |