Target Details
| UniProt AC | P48736 |
|---|---|
| Gene Symbol | PIK3CG |
| Protein Name | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF19710 (PIK3CG_ABD) |
Summary
- Multi-target molecules 2,398
- Clinical molecules 104
- Avg pChEMBL 7.16
KEGG Pathways (14)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Inositol phosphate metabolism
- Kaposi sarcoma-associated herpesvirus infection
- Metabolic pathways
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Salmonella infection
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (2,398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MHBBEPGMTPLJJK
|
7.4 | IC50 | 4 | — | |
NPCCZSIFYWKTIW
|
7.4 | IC50 | 2 | — | |
OWYNYCCFQVSEKU
|
7.4 | Ki | 4 | — | |
PEIFGMMJOLFHBE
|
7.4 | IC50 | 8 | — | |
PMJUIGQEQOQVFN
|
7.4 | IC50 | 4 | — | |
QTHCAAFKVUWAFI
|
7.4 | IC50 | 23 | — | |
RNJOUVJEMXMEDF
|
7.4 | IC50 | 2 | — | |
UQIUWUJYJBQZBY
|
7.4 | IC50 | 4 | — | |
UVSDWWSWVGVLAM
|
7.4 | IC50 | 3 | — | |
WNFRNSMPYGJUNB
|
7.4 | IC50 | 3 | — | |
GIQAVYAYXZICPG
|
7.4 | IC50 | 8 | — | |
HFXBHLPRJMROSI
|
7.4 | IC50 | 3 | — | |
KHRLDQKYINODSW
|
7.4 | IC50 | 4 | — | |
MZDVYDDLVZYLGV
|
7.4 | Ki | 5 | — | |
OXKACKLTXZOHOG
|
7.4 | IC50 | 3 | — | |
VOZATGBILRZYMT
|
7.4 | IC50 | 3 | — | |
YJIUXGKGVIYTOQ
|
7.4 | IC50 | 3 | — | |
BCKQIDIXDOCRCK
|
7.4 | IC50 | 2 | — | |
BUOSMKAGFRTJKQ
|
7.4 | IC50 | 3 | — | |
IZSUSVHQPBIXPL
|
7.4 | Ki | 5 | — | |
KABBATBNPHTWDK
|
7.4 | IC50 | 4 | — | |
KOBDMZOFSXEFLG
|
7.4 | IC50 | 2 | — | |
MFAQYJIYDMLAIM
|
7.4 | Kd | 130 | Yes | |
NWOGAKBGRRKZPL
|
7.4 | IC50 | 2 | — | |
COAQRADEUYYCDG
|
7.4 | IC50 | 12 | Yes | |
GEZALMMCQYDFML
|
7.4 | IC50 | 15 | Yes | |
HQLYDYYQRFGZDZ
|
7.4 | IC50 | 7 | — | |
JBPFTIQLGQPNCK
|
7.4 | IC50 | 3 | — | |
JOWHQAYXFVOIIS
|
7.4 | IC50 | 4 | — | |
KNRONZUHGXIQLA
|
7.4 | IC50 | 4 | — | |
RFWIWJIKKWYZIY
|
7.4 | IC50 | 3 | — | |
TYJXVOWPGAWAHU
|
7.4 | IC50 | 2 | — | |
YPEHJQSANCKVPH
|
7.4 | IC50 | 3 | — | |
YXFHSKVBWDUQIW
|
7.4 | IC50 | 8 | — | |
ADFBGHLIVBZYKW
|
7.4 | IC50 | 3 | — | |
DGGZIRYFUXUEIQ
|
7.4 | IC50 | 3 | — | |
DZJGDNZVUPCXPX
|
7.4 | IC50 | 8 | — | |
HRRMXIICSWVXIS
|
7.4 | IC50 | 13 | Yes | |
KQQKNWZMZNQWRK
|
7.4 | IC50 | 3 | — | |
SNBBYDABBPIQBU
|
7.4 | IC50 | 4 | — | |
VLNLIVDYHRPHDN
|
7.4 | IC50 | 3 | — | |
VXHZLQYXNABHFH
|
7.4 | IC50 | 3 | — | |
YHKJMQFPJKYQOU
|
7.4 | IC50 | 3 | — | |
YUSWHXYYRGYCHG
|
7.4 | Ki | 6 | — | |
AOFNYCXYCYLTJD
|
7.3 | IC50 | 5 | — | |
HGAJTKWPNZDTRJ
|
7.3 | IC50 | 8 | — | |
KZJLHYQNEJSYNN
|
7.3 | IC50 | 6 | — | |
LVUPFSONRUTLLF
|
7.3 | Ki | 4 | — | |
NGZQIEWQLIAQMG
|
7.3 | IC50 | 4 | — | |
NXHSCEQOULVBJS
|
7.3 | IC50 | 8 | — |