Target Details
| UniProt AC | P48736 |
|---|---|
| Gene Symbol | PIK3CG |
| Protein Name | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF19710 (PIK3CG_ABD) |
Summary
- Multi-target molecules 2,398
- Clinical molecules 104
- Avg pChEMBL 7.16
KEGG Pathways (14)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Inositol phosphate metabolism
- Kaposi sarcoma-associated herpesvirus infection
- Metabolic pathways
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Salmonella infection
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (2,398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MZVFITYKDVDNGL
|
7.5 | IC50 | 3 | — | |
VARVHYOTVXHELT
|
7.5 | IC50 | 5 | — | |
XGTSXSXOYSMLKN
|
7.5 | IC50 | 2 | — | |
BRNCLSYLICSNRO
|
7.5 | IC50 | 2 | — | |
CUMZRJYMUMFVHW
|
7.5 | IC50 | 2 | — | |
DSLTXRYHANMRCS
|
7.5 | IC50 | 3 | — | |
HFXBHLPRJMROSI
|
7.5 | IC50 | 3 | — | |
ORCYHNDWPXEHBN
|
7.5 | IC50 | 2 | — | |
SLVOAUDZJJTTLJ
|
7.5 | IC50 | 2 | — | |
VPOMGPGTRWISIU
|
7.5 | IC50 | 4 | — | |
XIGIJFUSWMTGMS
|
7.5 | IC50 | 6 | — | |
MFGUSQRABAVVFV
|
7.5 | IC50 | 4 | — | |
JEGHXKRHKHPBJD
|
7.4 | IC50 | 4 | — | |
KHJNCYCXAKBENU
|
7.4 | IC50 | 4 | — | |
SSALYFTWJFAWDV
|
7.4 | IC50 | 4 | — | |
XDNGIZBMMIZNGD
|
7.4 | IC50 | 8 | — | |
XJQPXTWNTSKISQ
|
7.4 | IC50 | 8 | — | |
GNRMZIZVRFJSOD
|
7.4 | IC50 | 5 | — | |
IPVLXKJQJCLTKU
|
7.4 | IC50 | 3 | — | |
IQDLOUNBMCMZPG
|
7.4 | IC50 | 2 | — | |
NOXQEXHGLFKCLC
|
7.4 | IC50 | 5 | — | |
VFNUYVJFDQOTNJ
|
7.4 | IC50 | 6 | — | |
XLPQUBPSCCBYDH
|
7.4 | IC50 | 3 | — | |
AVYIJPUHWYOVRO
|
7.4 | IC50 | 8 | — | |
GJYCAYLNRYZYBQ
|
7.4 | IC50 | 2 | — | |
HJBUXSYRSZQEGF
|
7.4 | IC50 | 3 | — | |
HVYJBSUHDFURHA
|
7.4 | IC50 | 4 | — | |
KJYMUGDPPRMHGD
|
7.4 | IC50 | 3 | — | |
MJQGMYGGZLZWDH
|
7.4 | IC50 | 2 | — | |
QXQIOGDLSRWGPA
|
7.4 | IC50 | 2 | — | |
RTTVESHNTCUEOK
|
7.4 | IC50 | 3 | — | |
WKDBRCUUDXLTIM
|
7.4 | IC50 | 4 | — | |
YJIUXGKGVIYTOQ
|
7.4 | IC50 | 3 | — | |
YVBUTAWXLPEFFD
|
7.4 | IC50 | 5 | — | |
YWWOQYKAYFXXAB
|
7.4 | IC50 | 8 | — | |
ZMLQYUGCULYVRF
|
7.4 | IC50 | 3 | — | |
CMZIHVRMPLWUAZ
|
7.4 | IC50 | 2 | — | |
DZTLWKBUHSDUNK
|
7.4 | IC50 | 3 | — | |
IRENWYOEYVTIRD
|
7.4 | Ki | 2 | — | |
LBXKRIWHCRXGHJ
|
7.4 | IC50 | 8 | — | |
MFRGGAROFRXKRT
|
7.4 | IC50 | 10 | Yes | |
RFIVDWZOZZKRLA
|
7.4 | IC50 | 2 | — | |
ZBJQUHYYXNXALJ
|
7.4 | IC50 | 3 | — | |
AZAIEPRPFYJUGI
|
7.4 | IC50 | 4 | — | |
BXPJPICORRAXTC
|
7.4 | IC50 | 3 | — | |
FEXTUSFUMVYBFH
|
7.4 | IC50 | 2 | — | |
FPDKFSHCGOROGZ
|
7.4 | Ki | 4 | — | |
HAWIAVPLXUYCRU
|
7.4 | IC50 | 4 | — | |
KPFIPJMXDOSFKZ
|
7.4 | IC50 | 8 | — | |
LFYHKOFPAUGDBK
|
7.4 | IC50 | 4 | — |