Target Details
| UniProt AC | P48736 |
|---|---|
| Gene Symbol | PIK3CG |
| Protein Name | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF19710 (PIK3CG_ABD) |
Summary
- Multi-target molecules 2,398
- Clinical molecules 104
- Avg pChEMBL 7.16
KEGG Pathways (14)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Inositol phosphate metabolism
- Kaposi sarcoma-associated herpesvirus infection
- Metabolic pathways
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Salmonella infection
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (2,398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AYRHYIQWAHXGQS
|
7.5 | IC50 | 8 | — | |
BHUCXTFJLHAUGW
|
7.5 | IC50 | 2 | — | |
BNYGDAZWSZFPFR
|
7.5 | IC50 | 2 | — | |
JVORBSYGQBGRCY
|
7.5 | IC50 | 3 | — | |
NYHQXLSMSMLVGN
|
7.5 | Ki | 4 | — | |
OCDGTZUIGBFFHU
|
7.5 | IC50 | 2 | — | |
OYYVWNDMOQPMGE
|
7.5 | IC50 | 5 | — | |
RYLZKJJWQWEHSZ
|
7.5 | IC50 | 3 | — | |
UBELCIYBIARHIU
|
7.5 | IC50 | 5 | — | |
AEZTZVXEQNZMAV
|
7.5 | IC50 | 4 | — | |
CCGUJYVWXLUTIA
|
7.5 | IC50 | 3 | — | |
DTTGBWQUOGWGMZ
|
7.5 | IC50 | 4 | — | |
MPWLFBVAYNHZHQ
|
7.5 | IC50 | 8 | — | |
NRNPLKNQEHSDHU
|
7.5 | Ki | 5 | — | |
NSZMXUXTPZEXIU
|
7.5 | IC50 | 3 | — | |
UHAHZARPMJULFU
|
7.5 | IC50 | 3 | — | |
UUWCILLLYRVXIW
|
7.5 | IC50 | 4 | — | |
WARUZPFHLRLCHE
|
7.5 | IC50 | 7 | — | |
XOMIVKVWJYDNPK
|
7.5 | IC50 | 2 | — | |
ZCCMLCRXWWFYEG
|
7.5 | IC50 | 4 | — | |
CPDASYVBDNZTSW
|
7.5 | Ki | 4 | — | |
FUMQATBGDGLOKH
|
7.5 | IC50 | 8 | — | |
GVCOXBXPKBZDEG
|
7.5 | IC50 | 4 | — | |
NUGMMEMSYIUTGA
|
7.5 | IC50 | 5 | — | |
VYXZSLJQQXROKX
|
7.5 | IC50 | 4 | — | |
WCZUQCRTCZORNK
|
7.5 | IC50 | 3 | — | |
XNXYCERJHJYNDT
|
7.5 | IC50 | 3 | — | |
YVFBCMVHJYQPKJ
|
7.5 | IC50 | 2 | — | |
AUNMZFMPIXHYCD
|
7.5 | IC50 | 3 | — | |
GDDSKZQKRFOXKP
|
7.5 | IC50 | 2 | — | |
GIJQCKAFIZEMCM
|
7.5 | IC50 | 3 | — | |
GJLUGKQXXSECIU
|
7.5 | IC50 | 3 | — | |
HDXDQPRPFRKGKZ
|
7.5 | IC50 | 2 | — | |
IFJYYBZHFXCMOD
|
7.5 | IC50 | 3 | — | |
JEHTXQHLTKVUGY
|
7.5 | IC50 | 4 | — | |
JEJWVLIMIXHYDW
|
7.5 | IC50 | 3 | — | |
JXCSRHVITGYTRY
|
7.5 | IC50 | 2 | — | |
KXIQRMIPXPVUID
|
7.5 | IC50 | 3 | — | |
OPVRUFKBBKOABM
|
7.5 | IC50 | 4 | — | |
QRYDPOHAXNITJN
|
7.5 | IC50 | 3 | — | |
QTTBCYFVRARNAY
|
7.5 | Ki | 6 | — | |
AHAJAAGFYQHYMQ
|
7.5 | IC50 | 8 | — | |
AMEKXJGPLKONNT
|
7.5 | IC50 | 2 | — | |
BDQJIUXJPAJLOX
|
7.5 | IC50 | 8 | — | |
BTHPXDNRFHNRDI
|
7.5 | Ki | 5 | — | |
FJZPGNVKNOFELP
|
7.5 | IC50 | 3 | — | |
FUMQATBGDGLOKH
|
7.5 | IC50 | 8 | — | |
LMXYZMNDIFPRCF
|
7.5 | IC50 | 5 | — | |
LNFWSNQWRMMEBJ
|
7.5 | IC50 | 4 | — | |
LWSJQJQMKYBWTR
|
7.5 | IC50 | 3 | — |