Target Details
| UniProt AC | P48736 |
|---|---|
| Gene Symbol | PIK3CG |
| Protein Name | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF19710 (PIK3CG_ABD) |
Summary
- Multi-target molecules 2,398
- Clinical molecules 104
- Avg pChEMBL 7.16
KEGG Pathways (14)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Inositol phosphate metabolism
- Kaposi sarcoma-associated herpesvirus infection
- Metabolic pathways
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Salmonella infection
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (2,398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UOXOWFBZFQTLKZ
|
7.6 | IC50 | 3 | — | |
WHLHMMULLULBDZ
|
7.6 | IC50 | 8 | — | |
XMUQISMCKNWEHC
|
7.6 | IC50 | 3 | — | |
YKJGGEMOMSRCDT
|
7.6 | IC50 | 2 | — | |
ZQEMGSHFLAOJBZ
|
7.6 | IC50 | 3 | — | |
JOGKUKXHTYWRGZ
|
7.6 | IC50 | 28 | — | |
WLYIDVRUQGGLFL
|
7.6 | IC50 | 5 | — | |
DWSBFBNKOHQARX
|
7.6 | IC50 | 4 | — | |
FAELUCQBHSZYDV
|
7.6 | IC50 | 2 | — | |
LKZTUGNQRBBSGT
|
7.6 | IC50 | 4 | — | |
NUVCPSZAUMDZDL
|
7.6 | IC50 | 5 | — | |
ONTJFJBLGNRKST
|
7.6 | IC50 | 2 | — | |
YETISTKVYMZRKN
|
7.6 | IC50 | 4 | — | |
AQPXZIOUXMMPJH
|
7.6 | IC50 | 3 | — | |
BVUXORJTWQTUTI
|
7.6 | IC50 | 3 | — | |
DCBRPTMPTRRLGM
|
7.6 | IC50 | 5 | — | |
DNCJCVADVSHMIZ
|
7.6 | IC50 | 3 | — | |
DNYROFWYJBYUMQ
|
7.6 | IC50 | 8 | — | |
FZJSJVSWAKSDTQ
|
7.6 | IC50 | 4 | — | |
HRNGMKXGIBFNBE
|
7.6 | IC50 | 3 | — | |
IMDGJJWMDCENIG
|
7.6 | IC50 | 2 | — | |
OIFRMGWBMAWZFZ
|
7.6 | Ki | 5 | — | |
SJVQHLPISAIATJ
|
7.6 | IC50 | 5 | — | |
UOPPKPSZIRYWNN
|
7.6 | IC50 | 3 | — | |
BUCWDQXJJGZECG
|
7.6 | IC50 | 3 | — | |
ZMCCTUGKELKLJP
|
7.6 | IC50 | 4 | — | |
DHYADLCEAXMYPS
|
7.5 | IC50 | 9 | Yes | |
FHCPWFJAEYLMGM
|
7.5 | IC50 | 8 | — | |
GSRNNPHHTAAGGS
|
7.5 | IC50 | 3 | — | |
IHXYNQCIZAQJGQ
|
7.5 | Ki | 4 | — | |
JGMSAJQEYJEURV
|
7.5 | IC50 | 8 | — | |
JTACVHJPXOKMTI
|
7.5 | IC50 | 2 | — | |
MQJXZZFGKUKOGM
|
7.5 | IC50 | 4 | — | |
PDXZRWGUWIWZGB
|
7.5 | IC50 | 3 | — | |
QIHCTUXJDIPXKX
|
7.5 | IC50 | 3 | — | |
RXUICGPCVJHIGZ
|
7.5 | IC50 | 4 | — | |
TXHSRGJSQAXDGN
|
7.5 | IC50 | 4 | — | |
WZDLLWUKMJOVAK
|
7.5 | IC50 | 5 | — | |
FVOXAVYMKTXHTN
|
7.5 | IC50 | 3 | — | |
GXTWTBFETNXESR
|
7.5 | IC50 | 8 | — | |
HWGAIJRGZSBQBB
|
7.5 | IC50 | 2 | — | |
JTFVVDMVICDHIG
|
7.5 | IC50 | 3 | — | |
LINCHXKNCSPOKA
|
7.5 | IC50 | 8 | — | |
LMXZAHWOXLADSH
|
7.5 | IC50 | 5 | — | |
NRUOQMAAFHGBEE
|
7.5 | IC50 | 2 | — | |
NYDXFIYKDTZNFF
|
7.5 | IC50 | 3 | — | |
QINPEPAQOBZPOF
|
7.5 | IC50 | 4 | — | |
WJGUPWANJQCMJY
|
7.5 | IC50 | 3 | — | |
XZIRFISMMDAPDH
|
7.5 | Ki | 4 | — | |
RUUJMGODVLGFKM
|
7.5 | IC50 | 2 | — |