Target Details
| UniProt AC | P48736 |
|---|---|
| Gene Symbol | PIK3CG |
| Protein Name | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF19710 (PIK3CG_ABD) |
Summary
- Multi-target molecules 2,398
- Clinical molecules 104
- Avg pChEMBL 7.16
KEGG Pathways (14)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Inositol phosphate metabolism
- Kaposi sarcoma-associated herpesvirus infection
- Metabolic pathways
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Salmonella infection
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (2,398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YWWOQYKAYFXXAB
|
7.7 | IC50 | 8 | — | |
QPRMAEKTXODJGJ
|
7.7 | IC50 | 3 | — | |
ZYJKXKZHIIVJEB
|
7.7 | IC50 | 2 | — | |
FUKVQYDAJUEJHW
|
7.6 | IC50 | 3 | — | |
IJAVTPLMQUWYCR
|
7.6 | IC50 | 3 | — | |
JTAQBMNOEJZXPF
|
7.6 | IC50 | 2 | — | |
KBOCINOJPQBJHY
|
7.6 | IC50 | 8 | — | |
MQMKRQLTIWPEDM
|
7.6 | IC50 | 4 | — | |
OBMONDJKDAOWHR
|
7.6 | Ki | 5 | — | |
WPSIRTUKJQGAMQ
|
7.6 | IC50 | 3 | — | |
ACCFLVVUVBJNGT
|
7.6 | IC50 | 5 | — | |
FACINUDEPGDOCE
|
7.6 | IC50 | 2 | — | |
FJHIWTMAONNZST
|
7.6 | IC50 | 2 | — | |
IVWMPAOBMMXESU
|
7.6 | IC50 | 5 | — | |
JBUVDLRLXPANJI
|
7.6 | Ki | 4 | — | |
JJRKQAAMIWSSRQ
|
7.6 | Ki | 4 | — | |
LYSPEQLEBUPCJX
|
7.6 | IC50 | 3 | — | |
MLKLYQDMHYWKGW
|
7.6 | Ki | 5 | — | |
NYRRAVJTVDFZLN
|
7.6 | IC50 | 8 | — | |
PJSOHQYOAVQLMP
|
7.6 | IC50 | 4 | — | |
ULTJBQSQKZDTRU
|
7.6 | IC50 | 2 | — | |
VDKPPWNYXRVYDM
|
7.6 | IC50 | 8 | — | |
WNMCVILJGJDETC
|
7.6 | IC50 | 3 | — | |
IVYWKCAOPCHVMX
|
7.6 | IC50 | 3 | — | |
KAAMQZKICBFHHV
|
7.6 | IC50 | 3 | — | |
KLBQEMTZKYSAER
|
7.6 | IC50 | 3 | — | |
BDQJIUXJPAJLOX
|
7.6 | IC50 | 8 | — | |
FEAZPCVGCIRWDR
|
7.6 | IC50 | 7 | — | |
GABNZMRCOCJMDX
|
7.6 | IC50 | 3 | — | |
GXPJIBZBTOUYII
|
7.6 | IC50 | 4 | — | |
HRZFUMGOVROJJL
|
7.6 | IC50 | 2 | — | |
IMIPCVCEURKASE
|
7.6 | IC50 | 4 | — | |
IQDBKFTVYYBTJD
|
7.6 | IC50 | 5 | — | |
KFYHKGHTVWFWKP
|
7.6 | IC50 | 4 | — | |
LFYHKOFPAUGDBK
|
7.6 | IC50 | 4 | — | |
LKRMPKDNVLEEJI
|
7.6 | IC50 | 5 | — | |
LUKHPIFOJUBBBW
|
7.6 | IC50 | 8 | — | |
MAVPREISACEICP
|
7.6 | IC50 | 8 | — | |
MDBIXUKQOSSWPT
|
7.6 | IC50 | 2 | — | |
MMPZSLSWQVQLJD
|
7.6 | IC50 | 7 | — | |
NLZNQTSAEGRBEQ
|
7.6 | IC50 | 8 | — | |
OVGAOZHAOVZSBT
|
7.6 | IC50 | 4 | — | |
PRNOUMSQOOBTIW
|
7.6 | IC50 | 3 | — | |
QTUZUSSFUQCQFS
|
7.6 | IC50 | 5 | — | |
QYBGBLQCOOISAR
|
7.6 | IC50 | 9 | — | |
RBSFIASCXZWSQM
|
7.6 | IC50 | 2 | — | |
RXRZPHQBTHQXSV
|
7.6 | IC50 | 2 | — | |
UBLOHCIYTDRGJH
|
7.6 | IC50 | 4 | — | |
UCZZPKDXRPXEAF
|
7.6 | IC50 | 5 | — | |
UISOZEPWNXYPCK
|
7.6 | IC50 | 4 | — |