Target Details
| UniProt AC | P48736 |
|---|---|
| Gene Symbol | PIK3CG |
| Protein Name | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF19710 (PIK3CG_ABD) |
Summary
- Multi-target molecules 2,398
- Clinical molecules 104
- Avg pChEMBL 7.16
KEGG Pathways (14)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Inositol phosphate metabolism
- Kaposi sarcoma-associated herpesvirus infection
- Metabolic pathways
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Salmonella infection
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (2,398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UGXHPLJCSWLUIK
|
7.7 | Ki | 3 | — | |
UVJBPMCZKOGSIP
|
7.7 | IC50 | 4 | — | |
VCBZVSWEFHPAJX
|
7.7 | IC50 | 2 | — | |
VHNNKJCKILGDNA
|
7.7 | IC50 | 5 | — | |
XOVOMIOHGLZGJN
|
7.7 | IC50 | 5 | — | |
YICAXAAHZCUKRE
|
7.7 | IC50 | 2 | — | |
YTFVFLULFAFNTO
|
7.7 | IC50 | 4 | — | |
ZWEJBXXYQYTACR
|
7.7 | Ki | 6 | — | |
AKFJKRXXJVIFOI
|
7.7 | IC50 | 3 | — | |
ALMGVNBNMXRCQV
|
7.7 | IC50 | 8 | — | |
ALYMJMACGKTBIZ
|
7.7 | IC50 | 4 | — | |
CFTQLFMYQDWTPI
|
7.7 | IC50 | 5 | — | |
DDOGMZTWQKWDBQ
|
7.7 | Ki | 5 | — | |
DFTRUCNLZXQDKU
|
7.7 | IC50 | 2 | — | |
HJMSDMFCCDZFIX
|
7.7 | Ki | 4 | — | |
HUIOREQGDCWTAK
|
7.7 | Ki | 5 | — | |
IHWMYZQUTPMTII
|
7.7 | IC50 | 5 | — | |
ISLVPOPCAGBKHP
|
7.7 | IC50 | 8 | — | |
LFNUJWZBIXHQJT
|
7.7 | Ki | 5 | — | |
PLUDSXLHMVRUKP
|
7.7 | IC50 | 2 | — | |
RERZXCUAKWVHPD
|
7.7 | IC50 | 3 | — | |
RERZXCUAKWVHPD
|
7.7 | IC50 | 4 | — | |
RGCKLULZGWBAOV
|
7.7 | IC50 | 2 | — | |
RIQACLQMPHPJFB
|
7.7 | IC50 | 3 | — | |
RYCGEXLWAPGHHN
|
7.7 | IC50 | 3 | — | |
UINYBYLWBAMMPE
|
7.7 | IC50 | 8 | — | |
VNLWAKVFNKVUJI
|
7.7 | IC50 | 3 | — | |
WLWNPIXCZPZWEA
|
7.7 | IC50 | 2 | — | |
XOKZXNOZHXOLDH
|
7.7 | IC50 | 3 | — | |
ZYVPTSVWIYTTDD
|
7.7 | IC50 | 4 | — | |
LXKCPGRADZOFQP
|
7.7 | IC50 | 3 | — | |
RGVKBHWXKPSTNQ
|
7.7 | IC50 | 3 | — | |
XANZNPICXVINSW
|
7.7 | IC50 | 3 | — | |
ZDRCETALOQGAMM
|
7.7 | IC50 | 4 | — | |
CAAMXUUCNDCFFK
|
7.7 | IC50 | 3 | — | |
DNAKNIPQHSVMLE
|
7.7 | IC50 | 3 | — | |
FYGDHTMAQTVJIR
|
7.7 | IC50 | 8 | — | |
GLNUMAOLJXQNNC
|
7.7 | IC50 | 2 | — | |
KKPQTTPNOXAYBC
|
7.7 | IC50 | 4 | — | |
LWEIOXGOXUSRJQ
|
7.7 | Ki | 2 | — | |
MPALXKOTYONGSD
|
7.7 | IC50 | 4 | — | |
MVOGBVAVCQDEHO
|
7.7 | IC50 | 5 | — | |
NWZPJXVCMJVRCW
|
7.7 | IC50 | 3 | — | |
SEMFARBMXOASOD
|
7.7 | IC50 | 3 | — | |
VBYCMVGPGAGETD
|
7.7 | Ki | 4 | — | |
VRGFZOXHCPIFTF
|
7.7 | IC50 | 3 | — | |
XAANLSVGMMQAAB
|
7.7 | IC50 | 3 | — | |
XILYGSAROZNXNT
|
7.7 | Ki | 4 | — | |
YCMPAJXRYQKAKZ
|
7.7 | IC50 | 5 | — | |
YGVFZWRVQCNDLQ
|
7.7 | IC50 | 3 | — |