Target Details
| UniProt AC | P48736 |
|---|---|
| Gene Symbol | PIK3CG |
| Protein Name | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF19710 (PIK3CG_ABD) |
Summary
- Multi-target molecules 2,398
- Clinical molecules 104
- Avg pChEMBL 7.16
KEGG Pathways (14)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Inositol phosphate metabolism
- Kaposi sarcoma-associated herpesvirus infection
- Metabolic pathways
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Salmonella infection
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (2,398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XJQPXTWNTSKISQ
|
7.8 | IC50 | 8 | — | |
YEOFKDOQMIILQR
|
7.8 | IC50 | 4 | — | |
IRTAFDFALCVEOW
|
7.8 | Ki | 6 | — | |
ITXYPAQDIOJYSR
|
7.8 | IC50 | 3 | — | |
PJLCSHAJFXTJCY
|
7.8 | IC50 | 2 | — | |
SMYKBETUHPQRLG
|
7.8 | IC50 | 3 | — | |
ZXGQCEYIWIQYRV
|
7.8 | IC50 | 3 | — | |
CBLXFJOGYFFYFS
|
7.8 | IC50 | 8 | — | |
CDBZWHCUAHJXIC
|
7.8 | IC50 | 8 | — | |
YRDHKIFCGOZTGD
|
7.8 | IC50 | 21 | — | |
AXHJCTAXCZSLFA
|
7.7 | Ki | 4 | — | |
BJAFXPJUBHYAHR
|
7.7 | IC50 | 3 | — | |
KXOKJGLSRORVTQ
|
7.7 | IC50 | 2 | — | |
MSLMLOUWBRFGOO
|
7.7 | IC50 | 3 | — | |
NSWURHBWYFQRSK
|
7.7 | IC50 | 4 | — | |
OPNRYAQJSHIIBL
|
7.7 | IC50 | 3 | — | |
QKDLMWZHWDLIHJ
|
7.7 | IC50 | 5 | — | |
SGEUNORSOZVTOL
|
7.7 | Ki | 6 | — | |
SPXPFOZHHLWRME
|
7.7 | IC50 | 3 | — | |
WAOBNLUKXUNDIU
|
7.7 | IC50 | 3 | — | |
WSLSYHQEXCFTLS
|
7.7 | IC50 | 3 | — | |
YPUUKLQYBLWUEU
|
7.7 | IC50 | 4 | — | |
ZJAVHOMVDCMAMF
|
7.7 | IC50 | 9 | — | |
VPLAAHHOBJVHMP
|
7.7 | IC50 | 3 | — | |
ANYFGHOATOBSFY
|
7.7 | IC50 | 5 | — | |
FYUBLRKIOOXTNB
|
7.7 | IC50 | 4 | — | |
MLTPTUWQLMSDBQ
|
7.7 | IC50 | 4 | — | |
MNORRMOFQMRDOH
|
7.7 | IC50 | 4 | — | |
PHAJRAXPUGWQRH
|
7.7 | IC50 | 8 | — | |
PXUUDOHYGXJCDO
|
7.7 | IC50 | 4 | — | |
RBFZKUBWJMBTHB
|
7.7 | IC50 | 5 | — | |
UTIUYGXIWRQSMG
|
7.7 | IC50 | 4 | — | |
XHYCVVZBZFPLDA
|
7.7 | IC50 | 4 | — | |
FWYXLDROMMGZKZ
|
7.7 | IC50 | 3 | — | |
ADDKHACIHJBWDD
|
7.7 | IC50 | 8 | — | |
BTHPXDNRFHNRDI
|
7.7 | Ki | 5 | — | |
BVAIASCEGGMUQD
|
7.7 | IC50 | 2 | — | |
DTJDTFBMPVOAPF
|
7.7 | IC50 | 3 | — | |
GGOACBRVBFQTCO
|
7.7 | IC50 | 4 | — | |
HJYSQORNBGTBRJ
|
7.7 | IC50 | 4 | — | |
HXQFBOHIYKLZRJ
|
7.7 | IC50 | 3 | — | |
IRYPRNBFNRSBFQ
|
7.7 | IC50 | 5 | — | |
JDUUUKXVZOZLSS
|
7.7 | IC50 | 5 | — | |
JLOYLMZLENULHD
|
7.7 | IC50 | 8 | — | |
KDCLKSQWABSKKF
|
7.7 | IC50 | 2 | — | |
LJIZLMDWRRLKJV
|
7.7 | IC50 | 2 | — | |
NLAFCFUVNPEKMI
|
7.7 | IC50 | 3 | — | |
OPIOWYFBJZWXNE
|
7.7 | IC50 | 4 | — | |
SAKNYPNGZWVPOL
|
7.7 | IC50 | 3 | — | |
TYLTZPAGUBOPCU
|
7.7 | IC50 | 3 | — |