Target Details
| UniProt AC | P48736 |
|---|---|
| Gene Symbol | PIK3CG |
| Protein Name | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF19710 (PIK3CG_ABD) |
Summary
- Multi-target molecules 2,398
- Clinical molecules 104
- Avg pChEMBL 7.16
KEGG Pathways (14)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Inositol phosphate metabolism
- Kaposi sarcoma-associated herpesvirus infection
- Metabolic pathways
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Salmonella infection
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (2,398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XDMHYCMFWUAUQG
|
7.9 | IC50 | 3 | — | |
XLCBQUCCOPILIO
|
7.9 | IC50 | 5 | — | |
AIGSGJXYLHDMBA
|
7.9 | IC50 | 6 | — | |
ALFGGTAMJAANKH
|
7.9 | IC50 | 4 | — | |
CKYACLUDESDZDP
|
7.9 | IC50 | 5 | — | |
CVJYZNKVAFBTDT
|
7.9 | IC50 | 8 | — | |
DQZLROXWLDKQMA
|
7.9 | IC50 | 2 | — | |
FFIJKEOXPCFSSY
|
7.9 | Ki | 2 | — | |
FGJSGEOFFFKFLV
|
7.9 | IC50 | 8 | — | |
FRHKVIMTLRQAGG
|
7.9 | IC50 | 3 | — | |
IJIRLVRZBZFXKE
|
7.9 | IC50 | 4 | — | |
INYPLABHSCEPJW
|
7.9 | IC50 | 3 | — | |
JNDYHRYIYXJWHN
|
7.9 | IC50 | 3 | — | |
LHLRTOZIMJUPET
|
7.9 | IC50 | 6 | — | |
LROPHDOTMYDOGU
|
7.9 | IC50 | 2 | — | |
LYZVYVLSMGRTPB
|
7.9 | IC50 | 5 | — | |
MABMRCWHKCPRMW
|
7.9 | IC50 | 5 | — | |
MRGAOHCEZOSOKZ
|
7.9 | IC50 | 3 | — | |
MSEBGSRJRAODPC
|
7.9 | IC50 | 5 | — | |
MVPHPMFJESRQLE
|
7.9 | IC50 | 5 | — | |
NORWTLLCOTYPQA
|
7.9 | IC50 | 8 | — | |
PGUDWAVWKFMVMF
|
7.9 | IC50 | 2 | — | |
QATDLTPQGNUUQD
|
7.9 | IC50 | 4 | — | |
RWYIHTNRCHCINH
|
7.9 | IC50 | 2 | — | |
WEHWXEIMYUDVOQ
|
7.9 | IC50 | 4 | — | |
ZNFDDMXBLQLUCC
|
7.9 | IC50 | 5 | — | |
ZTVMJVCYGUPZPC
|
7.9 | IC50 | 2 | — | |
MGQDDAHTGNTYQE
|
7.9 | IC50 | 3 | — | |
XNCXYRRIKXUUBE
|
7.9 | IC50 | 3 | — | |
YZAXUUNTFHQIHS
|
7.9 | IC50 | 3 | — | |
AVPAAQMVQVGYGP
|
7.8 | IC50 | 8 | — | |
CRRFQVURAQJNGW
|
7.8 | IC50 | 2 | — | |
FUMQATBGDGLOKH
|
7.8 | IC50 | 8 | — | |
ICGMCBFTEXPBTK
|
7.8 | IC50 | 3 | — | |
IICBFVCHOUCXJI
|
7.8 | IC50 | 5 | — | |
JLLNJCLPXQOWFX
|
7.8 | IC50 | 4 | — | |
LPQNHUUMWHCKNU
|
7.8 | Ki | 5 | — | |
OJHSROFLMBEBRH
|
7.8 | IC50 | 5 | — | |
XKONQDZYNDBPBD
|
7.8 | IC50 | 3 | — | |
XMUMBKFOUOBSOO
|
7.8 | IC50 | 5 | — | |
YOVVNQKCSKSHKT
|
7.8 | IC50 | 15 | — | |
YOVVNQKCSKSHKT
|
7.8 | IC50 | 5 | — | |
YVAOMSDQXISTTH
|
7.8 | IC50 | 5 | — | |
ZHHKIDAEQSNMOI
|
7.8 | IC50 | 4 | — | |
IXMCVAWUFQXLOS
|
7.8 | IC50 | 3 | — | |
MIPSHXJPVYIDDC
|
7.8 | IC50 | 3 | — | |
SGRQFHRGTVOPPV
|
7.8 | IC50 | 3 | — | |
DUFOKEKRNQSOSS
|
7.8 | IC50 | 4 | — | |
AKKCGLXULFRAET
|
7.8 | IC50 | 7 | — | |
AZDQPKKYASUZCZ
|
7.8 | IC50 | 5 | — |