Target Details
| UniProt AC | P48736 |
|---|---|
| Gene Symbol | PIK3CG |
| Protein Name | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF00794 (PI3K_rbd) PF00613 (PI3Ka) PF19710 (PIK3CG_ABD) |
Summary
- Multi-target molecules 2,398
- Clinical molecules 104
- Avg pChEMBL 7.16
KEGG Pathways (14)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Inositol phosphate metabolism
- Kaposi sarcoma-associated herpesvirus infection
- Metabolic pathways
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Salmonella infection
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (2,398)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GACQNUHFDBEIQH
|
10.0 | Ki | 4 | — | |
WHJIHZSXTQRCNX
|
9.8 | Ki | 10 | — | |
WVFAKEBPNFHPRY
|
9.8 | IC50 | 2 | — | |
ZLIOLJNSOUWXQU
|
9.6 | IC50 | 2 | — | |
PWYFLFWGSIDZCZ
|
9.5 | IC50 | 2 | — | |
XUMALORDVCFWKV
|
9.5 | IC50 | 7 | — | |
DHYKCYPTCMJMTA
|
9.5 | IC50 | 4 | — | |
IUQWLTSZFLUELP
|
9.5 | IC50 | 4 | — | |
RXZWDJAMFHLGND
|
9.5 | IC50 | 5 | — | |
JANGZKOHBDPUSU
|
9.4 | Ki | 2 | — | |
ILXAWHFQWWTBNG
|
9.4 | Ki | 4 | — | |
LPJAKJUVEMSSSX
|
9.4 | Ki | 9 | — | |
HLXBXWCMJQLPHD
|
9.3 | IC50 | 3 | — | |
JOOQGACJDJKFPA
|
9.3 | IC50 | 5 | — | |
CGBJSGAELGCMKE
|
9.3 | IC50 | 11 | — | |
YZIQNVDBRMRXLM
|
9.3 | Ki | 4 | — | |
DUUVJFLCJKWQTO
|
9.2 | IC50 | 4 | — | |
FTAOKGSTPLDORD
|
9.2 | IC50 | 5 | — | |
QXEBUDGMCKMQGM
|
9.2 | IC50 | 4 | — | |
CEANWFYTBJIQQX
|
9.2 | IC50 | 3 | — | |
KOSIBWHRFICAMX
|
9.2 | IC50 | 2 | — | |
HSISPDIJGGZDQA
|
9.2 | IC50 | 2 | — | |
RMZMULPZUXWJGE
|
9.2 | IC50 | 3 | — | |
YKKDQSUXCTZICT
|
9.2 | IC50 | 2 | — | |
RVHGXIUOUJYWPJ
|
9.2 | IC50 | 5 | — | |
ATRNPHJIZBECNS
|
9.2 | IC50 | 5 | — | |
AYLIBFXIKSYUIG
|
9.2 | IC50 | 5 | — | |
DBBKLJOYGVTYCR
|
9.2 | IC50 | 5 | — | |
KGNNMSGRBVKSQP
|
9.2 | IC50 | 3 | — | |
LAOPBSKJOXMHRY
|
9.2 | IC50 | 5 | — | |
WLKYZGMFQZHXRQ
|
9.2 | IC50 | 3 | — | |
SLVDFWRJWQJSRW
|
9.1 | IC50 | 5 | — | |
AQYTWWQAZAOONP
|
9.1 | IC50 | 5 | — | |
BMEVMMHSZQHXGB
|
9.1 | IC50 | 4 | — | |
CRXLXOVZGMTILX
|
9.1 | IC50 | 2 | — | |
DMIIPYYADLDKAX
|
9.1 | IC50 | 4 | — | |
FLNSZPSGBYDYIC
|
9.1 | IC50 | 2 | — | |
GMKBCIVCVYKVBE
|
9.1 | IC50 | 3 | — | |
GSXKIGLWEFFMTG
|
9.1 | IC50 | 2 | — | |
KWHLMLQDUKNHBO
|
9.1 | IC50 | 3 | — | |
LHKIAELCKQHVBI
|
9.1 | IC50 | 3 | — | |
LOYIOALZAFIRRM
|
9.1 | IC50 | 4 | — | |
MZRYOHCLXSQOIU
|
9.1 | IC50 | 4 | — | |
NDSSKUUMDINTDG
|
9.1 | IC50 | 3 | — | |
PAQUFWFUOVDUIO
|
9.1 | IC50 | 4 | — | |
SDQPODDUDFEPDG
|
9.1 | IC50 | 3 | — | |
VFBCXKOMIUXVNH
|
9.1 | IC50 | 4 | — | |
WEMBXYLJGBGCSQ
|
9.1 | IC50 | 3 | — | |
YXGZTQDPLYDOCC
|
9.1 | IC50 | 4 | — | |
ZGQXHYGEONUMTE
|
9.1 | IC50 | 7 | — |