Target Details
| UniProt AC | P48735 |
|---|---|
| Gene Symbol | IDH2 |
| Protein Name | Isocitrate dehydrogenase [NADP], mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00180 (Iso_dh) |
Summary
- Multi-target molecules 78
- Clinical molecules 0
- Avg pChEMBL 6.99
KEGG Pathways (8)
Associated Diseases (4)
Active Molecules (78)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZCCPLJOKGAACRT
|
8.7 | Kd | 599 | — | |
GTMXNXATSGQGCH
|
8.4 | IC50 | 2 | — | |
JZZYEUNYLVHGAO
|
8.2 | IC50 | 2 | — | |
NCCNQXYOCGUIQW
|
8.2 | IC50 | 2 | — | |
WFTCEDYVKXKHBE
|
8.2 | IC50 | 2 | — | |
QCZAWDGAVJMPTA
|
8.2 | IC50 | 2 | — | |
QCZAWDGAVJMPTA
|
8.1 | IC50 | 2 | — | |
JWMKUJAOIPXYIG
|
8.1 | IC50 | 2 | — | |
GJNPRCBREKXFRM
|
7.9 | IC50 | 2 | — | |
KNDBYTOOVAJFRN
|
7.9 | IC50 | 2 | — | |
SDVGLHHVYYZRJZ
|
7.8 | IC50 | 2 | — | |
KRSKURCJOGAEOS
|
7.8 | IC50 | 2 | — | |
DWIQMUBNZXFUDC
|
7.7 | IC50 | 2 | — | |
UIBBMCJNFUASJY
|
7.7 | IC50 | 2 | — | |
BHYQNYPMHHWOHO
|
7.5 | IC50 | 2 | — | |
BASWGFWYCDZRSM
|
7.5 | IC50 | 2 | — | |
AFGYODUJVVOZAX
|
7.4 | IC50 | 2 | — | |
GSAWFHLLQMRJAD
|
7.3 | IC50 | 2 | — | |
PKBWNJLBLZQTRD
|
7.3 | IC50 | 2 | — | |
BASWGFWYCDZRSM
|
7.3 | IC50 | 2 | — | |
BHYQNYPMHHWOHO
|
7.2 | IC50 | 2 | — | |
PKBWNJLBLZQTRD
|
7.1 | IC50 | 2 | — | |
PKBWNJLBLZQTRD
|
7.1 | IC50 | 2 | — | |
CNPVZLAVEHNGOP
|
7.1 | IC50 | 2 | — | |
DDVPWDBXRXZEBC
|
7.1 | IC50 | 2 | — | |
HNZFJEZPGBZOCO
|
7.1 | IC50 | 2 | — | |
KBOZWPPHVTYNOC
|
7.1 | IC50 | 2 | — | |
LWUOICMGVABMMB
|
7.1 | IC50 | 2 | — | |
MDCZNBIZILVZSF
|
7.1 | IC50 | 2 | — | |
MMQKYUIBTNHALE
|
7.1 | IC50 | 2 | — | |
MNWAUMZTPYXVGO
|
7.1 | IC50 | 2 | — | |
MVCBBRZTMZDXPK
|
7.1 | IC50 | 2 | — | |
OKFOLQBIBWUZIG
|
7.1 | IC50 | 2 | — | |
PDSKCDIBFYQGCE
|
7.1 | IC50 | 2 | — | |
SDUBFPITPDQUSW
|
7.1 | IC50 | 2 | — | |
SDUBFPITPDQUSW
|
7.1 | IC50 | 2 | — | |
VVDJVXUCSQFDNF
|
7.1 | IC50 | 2 | — | |
VWUHSVAZJFWQPW
|
7.1 | IC50 | 2 | — | |
WTQROKONFNCZLX
|
7.1 | IC50 | 2 | — | |
YNUDPCHEAJUNPU
|
7.1 | IC50 | 2 | — | |
YVNVAIVKELSNHE
|
7.1 | IC50 | 2 | — | |
BHYQNYPMHHWOHO
|
7.1 | IC50 | 2 | — | |
KUNRVODWGULPIF
|
7.1 | IC50 | 2 | — | |
KFKFZAMDAKZTOH
|
7.1 | IC50 | 2 | — | |
LYMZYGUSADHRMY
|
7.0 | IC50 | 2 | — | |
AFGYODUJVVOZAX
|
7.0 | IC50 | 2 | — | |
QCZAWDGAVJMPTA
|
6.9 | IC50 | 2 | — | |
BASWGFWYCDZRSM
|
6.9 | IC50 | 2 | — | |
JQBYMSMAAIFVRP
|
6.7 | IC50 | 2 | — | |
IESPVJDCWDMFAC
|
6.7 | IC50 | 2 | — |