Target Details
| UniProt AC | P48729 |
|---|---|
| Gene Symbol | CSNK1A1 |
| Protein Name | Casein kinase I isoform alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 470
- Clinical molecules 11
- Avg pChEMBL 7.5
KEGG Pathways (9)
Active Molecules (470)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PUYIXDDMOUMMRR
|
6.3 | Ki | 27 | — | |
UCOWZARZLHNDKP
|
6.3 | Ki | 8 | — | |
XXSPHNFKLDJDAK
|
6.3 | Ki | 26 | — | |
ZPXPEKQMLOAPLT
|
6.3 | Ki | 15 | — | |
ZQUSFAUAYSEREK
|
6.3 | Ki | 7 | — | |
ZQUSFAUAYSEREK
|
6.3 | Ki | 9 | Yes | |
VCUXVXLUOHDHKK
|
6.3 | IC50 | 6 | — | |
PRPGMEHVPYNUSF
|
6.2 | IC50 | 3 | — | |
KQWTXAWKBUUOMU
|
6.2 | IC50 | 20 | Yes | |
UVOREYMEAFPJPX
|
6.2 | IC50 | 9 | — | |
FAIHBCXQSBIRIL
|
6.2 | Ki | 22 | — | |
LYNBNVBMAGDJRW
|
6.2 | Ki | 81 | — | |
NGDXEOHYWJHBTJ
|
6.2 | IC50 | 5 | — | |
PBBRWFOVCUAONR
|
6.2 | Ki | 26 | Yes | |
SPYHMOFSJGTUNP
|
6.2 | Ki | 9 | — | |
SXBYKNSSEVQWPL
|
6.2 | Ki | 4 | — | |
UEFCSGDOOJJXTN
|
6.2 | IC50 | 46 | — | |
UPYHVTCMTMZKAX
|
6.2 | Ki | 12 | — | |
VSVWQTDDGQSGHP
|
6.2 | Ki | 51 | — | |
VXYDJXMHISGSDA
|
6.2 | Ki | 59 | — | |
ZGGIYFOLDBTZIL
|
6.2 | Ki | 27 | — | |
XEOVWJYINDYNSM
|
6.2 | Ki | 6 | — | |
RURHVWQWTJYUPS
|
6.2 | IC50 | 9 | — | |
CQNCHLJHIGRPDA
|
6.2 | IC50 | 6 | — | |
KNGBZHZRBXFQLV
|
6.1 | IC50 | 3 | — | |
JTVBXQAYBIJXRP
|
6.1 | Kd | 20 | — | |
AEYLJTAIDDIOBA
|
6.1 | Ki | 53 | — | |
FFQQZBOORWKWDZ
|
6.1 | Ki | 3 | — | |
FLEAYYMORDPWAJ
|
6.1 | Ki | 90 | — | |
GCYXEGSPUDSZJY
|
6.1 | Ki | 82 | — | |
IILNBGZKSQQREW
|
6.1 | Ki | 6 | — | |
JLTBOCSFMNSLFH
|
6.1 | Ki | 9 | — | |
PDTYLGXVBIWRIM
|
6.1 | Ki | 7 | — | |
PEEMSUJXJVLHFP
|
6.1 | Ki | 4 | — | |
RYAVJHIPOWNWDE
|
6.1 | Ki | 38 | — | |
ULSIWAGDPRIVCH
|
6.1 | Ki | 3 | — | |
WIHAOLDOGQOGIU
|
6.1 | Ki | 5 | — | |
WZMIWVZGYMKUDV
|
6.1 | IC50 | 3 | — | |
MSJODEOZODDVGW
|
6.1 | IC50 | 10 | — | |
UJIAQDJKSXQLIT
|
6.1 | Kd | 38 | — | |
AUMDBEHGJRZSOO
|
6.1 | IC50 | 3 | — | |
UJBJWYNPUOLFIZ
|
6.1 | IC50 | 49 | — | |
DKZYXHCYPUVGAF
|
6.0 | Kd | 112 | — | |
HKSZLNNOFSGOKW
|
6.0 | Kd | 408 | — | |
HOYRWTWZUFFACV
|
6.0 | Ki | 28 | — | |
HUXSWYWELGEQNC
|
6.0 | Ki | 5 | — | |
HZPACYSNLOCDLW
|
6.0 | Ki | 48 | — | |
IUEBPIPDFMCSTP
|
6.0 | Ki | 29 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JBJYTZXCZDNOJW
|
6.0 | IC50 | 3 | — |