Target Details
| UniProt AC | P48729 |
|---|---|
| Gene Symbol | CSNK1A1 |
| Protein Name | Casein kinase I isoform alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 470
- Clinical molecules 11
- Avg pChEMBL 7.5
KEGG Pathways (9)
Active Molecules (470)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CNPLAHBKWSNADG
|
6.7 | IC50 | 3 | — | |
BIDPCEXNMCKHCG
|
6.7 | IC50 | 3 | — | |
CFDCGXXHXUZSNP
|
6.7 | Kd | 4 | — | |
CYLDJPVEBVIXNB
|
6.6 | Kd | 6 | — | |
QNABDSWBQJKBHK
|
6.6 | IC50 | 45 | — | |
WINHZLLDWRZWRT
|
6.6 | Kd | 201 | Yes | |
BEJCLDKQCNVTQR
|
6.6 | Ki | 16 | — | |
DPEXRCOBPACFOO
|
6.6 | Ki | 36 | — | |
GMIKNOQZLHKCFH
|
6.6 | IC50 | 3 | — | |
MCBPNFWHHNJTGN
|
6.6 | IC50 | 5 | — | |
MLDQJTXFUGDVEO
|
6.6 | IC50 | 85 | Yes | |
PDBPUXLUVDSLML
|
6.6 | Ki | 14 | — | |
QKUFEXGLTQADSA
|
6.6 | Ki | 5 | — | |
SBFPHSVZEXSHTL
|
6.6 | Ki | 62 | — | |
UDFDIIVNIYWXDM
|
6.6 | Ki | 74 | — | |
XUFLBSMTYMFOQH
|
6.6 | Ki | 43 | — | |
YGKFZWJWKPZPQM
|
6.6 | Ki | 13 | — | |
UBPYILGKFZZVDX
|
6.5 | Kd | 130 | Yes | |
WHSIXKUPQCKWBY
|
6.5 | IC50 | 6 | — | |
DPDZHVCKYBCJHW
|
6.5 | IC50 | 11 | — | |
CHTMRWQLNNRRFJ
|
6.5 | Ki | 70 | — | |
DDDPTRGZLJPPQR
|
6.5 | Ki | 6 | — | |
DVWFMBFZDOBWAD
|
6.5 | Ki | 8 | — | |
KKWLJUDRBFHJPA
|
6.5 | Ki | 3 | — | |
KRIUNPBAQZGFQA
|
6.5 | Ki | 76 | — | |
MHWHPWMWKYXCRJ
|
6.5 | Ki | 32 | — | |
PROLIXHVRCJEFH
|
6.5 | Ki | 46 | — | |
SRONQUHCRFZABC
|
6.5 | Ki | 28 | — | |
SEZFNTZQMWJIAI
|
6.5 | Ki | 22 | — | |
MFAQYJIYDMLAIM
|
6.4 | Kd | 130 | Yes | |
FVNNTRZFDXTUGO
|
6.4 | IC50 | 3 | — | |
OQUWTJLQOZIRFA
|
6.4 | IC50 | 8 | — | |
CTNPALGJUAXMMC
|
6.4 | Kd | 151 | — | |
LCHCSKHPVCDXAU
|
6.4 | Ki | 30 | — | |
LPILBMJJRGTKOQ
|
6.4 | Ki | 27 | — | |
LRESELHEXSUQGE
|
6.4 | Ki | 10 | — | |
OULGHWYAFYSZGK
|
6.4 | Ki | 2 | — | |
QZPFUALVXZAFDD
|
6.4 | Ki | 10 | — | |
VTQQYBGURNVVFE
|
6.4 | Ki | 17 | — | |
WIRUYYYAAJOIKO
|
6.4 | Ki | 4 | — | |
XNWKXXIGSPPPBH
|
6.4 | Ki | 31 | — | |
YPDWGKSFVMASOZ
|
6.4 | Ki | 5 | — | |
ZGZVRPRSFXRGCF
|
6.4 | Ki | 76 | — | |
WZMIWVZGYMKUDV
|
6.4 | IC50 | 3 | — | |
WYOFSHLAFWJJAZ
|
6.4 | IC50 | 3 | — | |
DTEKTGDVSARYDS
|
6.3 | IC50 | 11 | — | |
XBAIEEJJCJHBDL
|
6.3 | Ki | 17 | — | |
BSFNGHCTZDCQBF
|
6.3 | Ki | 93 | — | |
GCBJDOWIQHMCMR
|
6.3 | Ki | 84 | — | |
OTQSCDWPCPZRIU
|
6.3 | Ki | 4 | — |