Target Details
| UniProt AC | P48729 |
|---|---|
| Gene Symbol | CSNK1A1 |
| Protein Name | Casein kinase I isoform alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 470
- Clinical molecules 11
- Avg pChEMBL 7.5
KEGG Pathways (9)
Active Molecules (470)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ATGVCJYHNOSZEV
|
7.3 | Ki | 23 | — | |
RJZDECGDCKOHBV
|
7.3 | Ki | 70 | — | |
BISBOJVKDYPBTP
|
7.3 | IC50 | 2 | — | |
KOFPMBNUPXOKAY
|
7.3 | IC50 | 3 | — | |
KEEOFKPCOCGLAA
|
7.3 | IC50 | 4 | — | |
BZFZAOWFYOKWDA
|
7.3 | IC50 | 2 | — | |
PPUNDPQNOCBVKW
|
7.3 | IC50 | 2 | — | |
DSVNYHIVOUUYFJ
|
7.2 | IC50 | 2 | — | |
CFRUQBGKKYVHHQ
|
7.2 | IC50 | 2 | — | |
BSAVGANXIAKUQK
|
7.2 | IC50 | 2 | — | |
FUMCKNCUEAQHCV
|
7.2 | Ki | 103 | — | |
HMUYZTPOWOYZKW
|
7.2 | IC50 | 2 | — | |
XGFIIXQAEJTAHR
|
7.1 | IC50 | 2 | — | |
CDMGBJANTYXAIV
|
7.1 | Kd | 34 | Yes | |
PYDWRLNPMMKKCI
|
7.1 | Ki | 7 | — | |
SLKCVFPEQGHNSI
|
7.1 | Ki | 29 | — | |
ATXRBBLJRPAIHG
|
7.1 | IC50 | 2 | — | |
HGZBLFDJBJBFKL
|
7.0 | IC50 | 2 | — | |
IVISHGNTPOVTQM
|
7.0 | IC50 | 2 | — | |
AECVPUDXLSQNOL
|
7.0 | IC50 | 3 | — | |
IJAGJGCELDNCJJ
|
7.0 | IC50 | 2 | — | |
DTMZXHDQZQLTHA
|
7.0 | Ki | 21 | — | |
FHYUGAJXYORMHI
|
7.0 | Ki | 7 | — | |
HDCULFQYOZCWNP
|
7.0 | IC50 | 2 | — | |
HEKAIDKUDLCBRU
|
7.0 | Ki | 20 | — | |
JJJSCYSPSKBQAX
|
7.0 | Ki | 34 | — | |
KHGPYYFCIAISBU
|
7.0 | Ki | 31 | — | |
UVTIDTZUUMJEGM
|
7.0 | IC50 | 2 | — | |
YUGAWPXFORPIGO
|
6.9 | IC50 | 2 | — | |
MGNQNQOSSLCUFP
|
6.9 | Ki | 12 | — | |
NJPWCTYVEJIQBM
|
6.9 | Ki | 72 | — | |
RGNHKJWHFIPHIM
|
6.9 | Ki | 66 | — | |
ZGDYBJXDIXVTLV
|
6.9 | Ki | 54 | — | |
YRFOQHHFWYWAST
|
6.9 | IC50 | 22 | — | |
BMIMXMZRHINYQM
|
6.9 | IC50 | 2 | — | |
VGNSQEJXQARLLC
|
6.8 | IC50 | 3 | — | |
OOYQNTZOMNZRSG
|
6.8 | IC50 | 8 | — | |
FGWOKLCRQJXPPQ
|
6.8 | Ki | 14 | — | |
KTWBYGUSEYSRND
|
6.8 | Ki | 28 | — | |
RPGBQFNDFPEOON
|
6.8 | Ki | 22 | — | |
XZONYYFHQICDAM
|
6.8 | Ki | 19 | — | |
KPGMXAQTPURKMK
|
6.8 | IC50 | 3 | — | |
BIUDJFOTQAVFMN
|
6.7 | IC50 | 9 | — | |
NVZGKHUBLBRWMH
|
6.7 | IC50 | 3 | — | |
JJGSOVIZOMZMCS
|
6.7 | Ki | 35 | — | |
OVKIYZXGCCAIJG
|
6.7 | Ki | 6 | — | |
PLHUMPJXRHMFFR
|
6.7 | Ki | 28 | — | |
UTMRCMCLMBDPNW
|
6.7 | Ki | 10 | — | |
XFWUTMHVDGPWLH
|
6.7 | Ki | 75 | — | |
ZKLJKKASNXVQBZ
|
6.7 | Ki | 27 | — |