Target Details
| UniProt AC | P48729 |
|---|---|
| Gene Symbol | CSNK1A1 |
| Protein Name | Casein kinase I isoform alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 470
- Clinical molecules 11
- Avg pChEMBL 7.5
KEGG Pathways (9)
Active Molecules (470)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NCIGMDJBHNIAJD
|
7.7 | IC50 | 2 | — | |
UUSCGSSISCGHIZ
|
7.7 | IC50 | 2 | — | |
ILGBTEPJRFWOFV
|
7.7 | IC50 | 2 | — | |
LWQRCWSAGSPNNW
|
7.7 | IC50 | 2 | — | |
NEOVWVIFEVIRBF
|
7.7 | IC50 | 2 | — | |
ASSQRJJOLODGSX
|
7.6 | IC50 | 2 | — | |
RCHPQGHUPYFPMV
|
7.6 | IC50 | 2 | — | |
AWQFFDDPKOKUOH
|
7.6 | IC50 | 2 | — | |
BSAVGANXIAKUQK
|
7.6 | IC50 | 3 | — | |
JIEXEDGFFBGAIL
|
7.6 | IC50 | 3 | — | |
KVIQZRSTAIWWJF
|
7.6 | IC50 | 2 | — | |
WYFBDHPKVNKMTH
|
7.6 | IC50 | 2 | — | |
QRVYIZSFRSIONY
|
7.6 | IC50 | 2 | — | |
UMQXUQDUPKDQIR
|
7.6 | IC50 | 2 | — | |
HRJDYJVDFILFKO
|
7.6 | IC50 | 2 | — | |
JOJTYLQIUBKNMM
|
7.6 | IC50 | 2 | — | |
RHYSDEXBESYPCB
|
7.6 | IC50 | 3 | — | |
FCDJELCDNCYXQE
|
7.6 | IC50 | 2 | — | |
FSUKRPNMEJYOMM
|
7.5 | IC50 | 2 | — | |
PVCDSODWAKIOMW
|
7.5 | IC50 | 2 | — | |
DKXHSOUZPMHNIZ
|
7.5 | Ki | 51 | Yes | |
DCGFWGFEATUMQK
|
7.5 | IC50 | 2 | — | |
PVVJMBBQASQRAX
|
7.5 | IC50 | 3 | — | |
RYYNYPNIEUPDOA
|
7.5 | IC50 | 2 | — | |
XBJAOZKEXGWEPB
|
7.5 | IC50 | 2 | — | |
MHLPTBJWCVRRPC
|
7.5 | IC50 | 2 | — | |
YCWSXEOEVCQKSE
|
7.5 | IC50 | 2 | — | |
ZPGJWXXQFLAVAY
|
7.5 | IC50 | 2 | — | |
ATBAETXFFCOZOY
|
7.5 | IC50 | 39 | — | |
YIYDFQGZXPQCEL
|
7.5 | IC50 | 2 | — | |
GGXUUYZKIPHVAW
|
7.5 | IC50 | 2 | — | |
DQBAYRJVCNUPBT
|
7.4 | IC50 | 2 | — | |
UYAQWCZWVIFRCN
|
7.4 | IC50 | 2 | — | |
BSAVGANXIAKUQK
|
7.4 | IC50 | 3 | — | |
GQYLIQAEIRWFEC
|
7.4 | IC50 | 2 | — | |
BGYVWFZMYBWCNY
|
7.4 | Ki | 30 | — | |
KBQAVBKOEJZTFM
|
7.4 | IC50 | 2 | — | |
NVRXTLZYXZNATH
|
7.4 | Ki | 47 | Yes | |
OWZSUHGYHPDMLH
|
7.4 | IC50 | 2 | — | |
XZWVOUQIYLZUCJ
|
7.4 | Ki | 23 | — | |
CDPQTBTYURAFME
|
7.4 | IC50 | 2 | — | |
BOQMJAHNAMIBMJ
|
7.4 | IC50 | 2 | — | |
PFYGLKQLEHKJBE
|
7.4 | IC50 | 3 | — | |
RDIZWXHOXKMYHK
|
7.3 | IC50 | 2 | — | |
VZLYECDBMSJTQG
|
7.3 | IC50 | 2 | — | |
HOMKDCYPLCAGBD
|
7.3 | IC50 | 2 | — | |
DBHMJFHKKRRBAC
|
7.3 | IC50 | 3 | — | |
GWTJDEOZCYRULI
|
7.3 | IC50 | 3 | — | |
QEYHZDYWQJEOMC
|
7.3 | IC50 | 2 | — | |
ADMFLILDQJSEIK
|
7.3 | Ki | 72 | — |