Target Details
| UniProt AC | P48729 |
|---|---|
| Gene Symbol | CSNK1A1 |
| Protein Name | Casein kinase I isoform alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 470
- Clinical molecules 11
- Avg pChEMBL 7.5
KEGG Pathways (9)
Active Molecules (470)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UJJMQXWMFBWWJA
|
7.9 | IC50 | 3 | — | |
KBUFBAQJZKYNEP
|
7.9 | IC50 | 2 | — | |
WTEKKYAHRWEYNN
|
7.9 | IC50 | 2 | — | |
FNUUVPCZCHTPPR
|
7.9 | IC50 | 3 | — | |
RFSUZJIQGIZAAA
|
7.9 | IC50 | 3 | — | |
FHYLCIXGVBYKBV
|
7.9 | IC50 | 2 | — | |
JYJVQAWBZXDVQN
|
7.9 | IC50 | 2 | — | |
LAFYDKMPJZTXHE
|
7.9 | IC50 | 3 | — | |
RFNJXUGGPMXOOK
|
7.9 | IC50 | 2 | — | |
VVCVNUUHMZMIBR
|
7.9 | IC50 | 2 | — | |
XCLVEFQLWKDCDX
|
7.9 | IC50 | 3 | — | |
DQGYZGUWRZBVCE
|
7.8 | IC50 | 2 | — | |
LBQIACDBOWZJEM
|
7.8 | IC50 | 2 | — | |
LWANFAFTTOKZAX
|
7.8 | IC50 | 11 | — | |
LWANFAFTTOKZAX
|
7.8 | IC50 | 3 | — | |
TUSWCHQSBHMNQB
|
7.8 | IC50 | 2 | — | |
UCWZHWFDHODGBP
|
7.8 | IC50 | 2 | — | |
AHTHSKQPKKMYPX
|
7.8 | IC50 | 3 | — | |
ATBIVHXUOKHWSC
|
7.8 | IC50 | 2 | — | |
DIBZPOAEDBOEEZ
|
7.8 | IC50 | 3 | — | |
OPOQBSCRYUUEBT
|
7.8 | IC50 | 2 | — | |
RKWUJVALCBMSHZ
|
7.8 | IC50 | 2 | — | |
ATSAULVLXRFCAQ
|
7.8 | IC50 | 2 | — | |
ILZYLHZIAQJQGN
|
7.8 | IC50 | 2 | — | |
KAPROIFCQLMDFT
|
7.8 | IC50 | 2 | — | |
JQPFYUYZGQPQOZ
|
7.8 | IC50 | 3 | — | |
KBUFBAQJZKYNEP
|
7.8 | IC50 | 2 | — | |
MQRBKUYTZJQBKW
|
7.8 | IC50 | 3 | — | |
PUQQTDNYVKXYIV
|
7.8 | IC50 | 2 | — | |
QAJPIJHWTGPUNZ
|
7.8 | Ki | 37 | — | |
WDARYLSSWBWVCU
|
7.8 | Ki | 49 | — | |
HUWCGRYLNBSQLN
|
7.8 | IC50 | 2 | — | |
HVAVBAIPXDAXHC
|
7.8 | IC50 | 2 | — | |
QHLWRPSEJQXVCM
|
7.8 | IC50 | 2 | — | |
RSMPMJNJRFVSRB
|
7.8 | IC50 | 2 | — | |
CJPUXQCRSOGYND
|
7.8 | IC50 | 2 | — | |
LXTFCMYUAINYQN
|
7.8 | IC50 | 2 | — | |
AKGWIZHTFUPWKX
|
7.7 | IC50 | 2 | — | |
PUKUDMLAYTVLDN
|
7.7 | IC50 | 2 | — | |
GECYDQWEFLTJMM
|
7.7 | IC50 | 2 | — | |
NWLSEQZPIYEHII
|
7.7 | IC50 | 2 | — | |
VEPRLRDIGFBHAG
|
7.7 | IC50 | 3 | — | |
VUVUREKZWANTPW
|
7.7 | IC50 | 4 | — | |
KKRDXOPMQOYAGZ
|
7.7 | IC50 | 2 | — | |
VAMRGLQMNCSXDM
|
7.7 | IC50 | 3 | — | |
VYKBWPLPWBMVTQ
|
7.7 | IC50 | 2 | — | |
WLUDGAUDVDKIOF
|
7.7 | IC50 | 2 | — | |
XZTZFGIZKXWMMU
|
7.7 | IC50 | 3 | — | |
OEXTZXWPZXNIIH
|
7.7 | IC50 | 3 | — | |
JMADTDZBMULVHU
|
7.7 | IC50 | 2 | — |