Target Details
| UniProt AC | P48729 |
|---|---|
| Gene Symbol | CSNK1A1 |
| Protein Name | Casein kinase I isoform alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 470
- Clinical molecules 11
- Avg pChEMBL 7.5
KEGG Pathways (9)
Active Molecules (470)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XBQQDPWXSKKKQL
|
8.1 | IC50 | 2 | — | |
BUTAQMUMZATNRF
|
8.1 | IC50 | 2 | — | |
CNNUFNBSGQUOFZ
|
8.1 | IC50 | 2 | — | |
CVDSGACKMHURND
|
8.1 | IC50 | 2 | — | |
DPXSVWSOUOLCJN
|
8.1 | IC50 | 2 | — | |
LBCTWIUPHHIYNO
|
8.1 | IC50 | 3 | — | |
MPNYXYMZXMXPMG
|
8.1 | IC50 | 3 | — | |
RBSCAZUMOUDJAV
|
8.1 | IC50 | 3 | — | |
OJTLEZVQEGWXAH
|
8.1 | IC50 | 2 | — | |
SXZJJMQIEVMLRL
|
8.1 | IC50 | 2 | — | |
CIUATZJWGJGLPW
|
8.1 | IC50 | 4 | — | |
DAVLHGUDTGYPHJ
|
8.1 | IC50 | 2 | — | |
KDFAUZONCVHIQC
|
8.0 | IC50 | 3 | — | |
KIAWAHJOKQOSAO
|
8.0 | IC50 | 3 | — | |
OCJNACKDBJHBPG
|
8.0 | IC50 | 2 | — | |
VBCYKNRNAQCIRZ
|
8.0 | IC50 | 2 | — | |
SWZLQQMKDWLWKC
|
8.0 | IC50 | 2 | — | |
XQNREAZQMGMBMX
|
8.0 | IC50 | 2 | — | |
BYINJOSWODJSOV
|
8.0 | IC50 | 2 | — | |
YSPIHUWHLMNFOV
|
8.0 | Kd | 2 | — | |
LOTGQVOARVITHH
|
8.0 | IC50 | 2 | — | |
MRRGNSSCHWNURS
|
8.0 | IC50 | 3 | — | |
OVWHGYZCHAOSFL
|
8.0 | IC50 | 3 | — | |
RUBGULKMMNPVRT
|
8.0 | IC50 | 2 | — | |
XJDSDBTWZHZYJT
|
8.0 | IC50 | 2 | — | |
AZBIOIRZHDKQJI
|
8.0 | IC50 | 2 | — | |
HBKRAHRIWQMIJU
|
8.0 | IC50 | 3 | — | |
NAIIXKKQMASUIR
|
8.0 | IC50 | 2 | — | |
ATJVIGPUJQKPPP
|
8.0 | IC50 | 2 | — | |
DUYUPVFZOHBSBS
|
8.0 | IC50 | 2 | — | |
FAIXFRDVCIWZOZ
|
8.0 | IC50 | 3 | — | |
WJNUSNNYLBLXMQ
|
8.0 | IC50 | 3 | — | |
YWWLWBUGJCBTOP
|
8.0 | IC50 | 2 | — | |
IJUJMMPOXXBQCM
|
8.0 | IC50 | 3 | — | |
UYAQWCZWVIFRCN
|
8.0 | IC50 | 2 | — | |
BGYLKQWHNHTXJA
|
7.9 | IC50 | 3 | — | |
LPYBJNPKBPALQQ
|
7.9 | IC50 | 3 | — | |
ZSGYTKAQRWJXFD
|
7.9 | IC50 | 2 | — | |
QCSBVNWGWVHGRR
|
7.9 | IC50 | 2 | — | |
CEDLEAIGKVAXEE
|
7.9 | IC50 | 3 | — | |
CESMQOAMBJTRME
|
7.9 | IC50 | 2 | — | |
GDPJYLRERIWTKI
|
7.9 | IC50 | 2 | — | |
IKATWWUGCJFQJV
|
7.9 | IC50 | 2 | — | |
IOKYXCFBOLCWNW
|
7.9 | IC50 | 2 | — | |
SXBIWPGTSITBPU
|
7.9 | IC50 | 3 | — | |
UASMATGCQULMCR
|
7.9 | IC50 | 3 | — | |
VTHDNDMZUMSBFW
|
7.9 | IC50 | 3 | — | |
KTQMBTHJIRDISH
|
7.9 | IC50 | 2 | — | |
USMHWTKVCMQLRC
|
7.9 | IC50 | 2 | — | |
VSPFURGQAYMVAN
|
7.9 | Ki | 17 | — |