Target Details
| UniProt AC | P48729 |
|---|---|
| Gene Symbol | CSNK1A1 |
| Protein Name | Casein kinase I isoform alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 470
- Clinical molecules 11
- Avg pChEMBL 7.5
KEGG Pathways (9)
Active Molecules (470)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FSLUVRSRENLUCL
|
8.3 | IC50 | 2 | — | |
DXOCGCLMPFHJFY
|
8.3 | IC50 | 2 | — | |
UGFJLMYCKZVPQW
|
8.3 | IC50 | 2 | — | |
PXIYPQXFGIMIKA
|
8.2 | IC50 | 2 | — | |
RBEKAJBCTQVXNP
|
8.2 | IC50 | 2 | — | |
UGZCBAQQMBKAOK
|
8.2 | IC50 | 2 | — | |
CCGPGRFPBJBQBH
|
8.2 | IC50 | 3 | — | |
HZBBZBIWSKGLLH
|
8.2 | IC50 | 2 | — | |
NIZDUIYCSULLSX
|
8.2 | IC50 | 2 | — | |
NQIKPWAJXBQQRO
|
8.2 | IC50 | 2 | — | |
ACSUKGRGGMZYHI
|
8.2 | IC50 | 3 | — | |
BCIMKEWMLAXRHD
|
8.2 | IC50 | 2 | — | |
JMADTDZBMULVHU
|
8.2 | IC50 | 2 | — | |
NEKWBIWCDRCGTN
|
8.2 | IC50 | 2 | — | |
HBGWEQADNDNBRS
|
8.2 | IC50 | 2 | — | |
KTTODKFIHICJMH
|
8.2 | IC50 | 2 | — | |
UNQVLUNGEAHZPW
|
8.2 | IC50 | 2 | — | |
VVCVNUUHMZMIBR
|
8.2 | IC50 | 2 | — | |
XPNJMLZYFXKLLR
|
8.2 | IC50 | 2 | — | |
BHTXWBUTVJYLAD
|
8.2 | IC50 | 2 | — | |
CKWPZOKUIUDWSA
|
8.2 | IC50 | 2 | — | |
JOXAVXOYZIYVPW
|
8.2 | IC50 | 2 | — | |
YXAZIXFVTZLQCR
|
8.2 | IC50 | 2 | — | |
SHHZYLAVDLPYJO
|
8.2 | IC50 | 2 | — | |
YDOZYQCKMQHHAB
|
8.2 | IC50 | 2 | — | |
NXZVSYWCPKVCRD
|
8.2 | IC50 | 2 | — | |
CVDHDXBBGDUUGC
|
8.2 | IC50 | 2 | — | |
LHIQTHDBSXSQTG
|
8.2 | IC50 | 3 | — | |
GVIDEIQDBDMNLC
|
8.2 | IC50 | 2 | — | |
VMRHBZTUDNJLEK
|
8.2 | IC50 | 2 | — | |
ARCIXQNVMWOXFO
|
8.1 | IC50 | 2 | — | |
SWOIFXHMBKFCRM
|
8.1 | IC50 | 4 | — | |
VVCVNUUHMZMIBR
|
8.1 | IC50 | 2 | — | |
DZZMTEOZQNBZDN
|
8.1 | IC50 | 2 | — | |
HIVSWSGDGRIDSN
|
8.1 | IC50 | 2 | — | |
IWCAAHBDNLJZOI
|
8.1 | IC50 | 3 | — | |
QNOANZOPMMGGQK
|
8.1 | IC50 | 2 | — | |
YDQUYBVEFYYJTD
|
8.1 | IC50 | 2 | — | |
YMWSWWLCKGGUCS
|
8.1 | IC50 | 2 | — | |
CQDQSVXDMSYUGR
|
8.1 | IC50 | 3 | — | |
CUSGCSBOGPVLNM
|
8.1 | IC50 | 2 | — | |
DPBBZVZOGCLXDJ
|
8.1 | IC50 | 2 | — | |
WPBKIQLDOLQVHG
|
8.1 | IC50 | 3 | — | |
WXFWDDXWJIXSSH
|
8.1 | IC50 | 2 | — | |
BTNLDKCTJOLQLU
|
8.1 | IC50 | 3 | — | |
MCKPYPWHBUXLEZ
|
8.1 | Ki | 21 | — | |
MXKWSWPSGNBXIT
|
8.1 | IC50 | 2 | — | |
RKUKAACYUCUJEE
|
8.1 | Ki | 58 | — | |
STQCJZAKVWFOTG
|
8.1 | IC50 | 2 | — | |
FAKIWNQURVDPPN
|
8.1 | IC50 | 2 | — |