Target Details
| UniProt AC | P48729 |
|---|---|
| Gene Symbol | CSNK1A1 |
| Protein Name | Casein kinase I isoform alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 470
- Clinical molecules 11
- Avg pChEMBL 7.5
KEGG Pathways (9)
Active Molecules (470)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CDUQLOKKQHDIFD
|
8.5 | IC50 | 2 | — | |
XKQBNZMXBOTZTP
|
8.5 | IC50 | 2 | — | |
GUNUORYXEAKXIM
|
8.5 | IC50 | 2 | — | |
QSOOWYJFQWRIAY
|
8.5 | IC50 | 3 | — | |
TVWCCJYWNNRHHQ
|
8.5 | IC50 | 2 | — | |
WBKHTUIWPNHAAL
|
8.5 | IC50 | 3 | — | |
KURMGXLJUFMRKC
|
8.4 | IC50 | 2 | — | |
LDHDORYQIJLGSC
|
8.4 | IC50 | 2 | — | |
URINSVMRQHIEGL
|
8.4 | IC50 | 2 | — | |
ATJMVWABXWLODR
|
8.4 | IC50 | 2 | — | |
IOTPYKAXEUJUIX
|
8.4 | IC50 | 2 | — | |
MUOKSQABCJCOPU
|
8.4 | IC50 | 36 | — | |
UHKJLPKHZOTEFL
|
8.4 | IC50 | 2 | — | |
VKLWOKCJHQIGOC
|
8.4 | IC50 | 2 | — | |
GWSYESFVOIPTOQ
|
8.4 | IC50 | 2 | — | |
HTDCNRIYLUVMQJ
|
8.4 | IC50 | 2 | — | |
PWHOGQARTNTIPD
|
8.4 | IC50 | 2 | — | |
SFEXHRDDQCDUFA
|
8.4 | IC50 | 2 | — | |
AFYHNCHUOWUSBR
|
8.4 | IC50 | 2 | — | |
DIPYWXZZVYYRSW
|
8.4 | IC50 | 2 | — | |
FMHGUBGXYPCKCK
|
8.4 | IC50 | 2 | — | |
NDTQLXWONKRJGN
|
8.4 | IC50 | 3 | — | |
SILIXJIYAFGFLO
|
8.4 | IC50 | 2 | — | |
VYXVLVRSUJXBDP
|
8.4 | IC50 | 2 | — | |
BLAQSCXKTBCBTO
|
8.4 | IC50 | 2 | — | |
HINDFIKMXAKSSM
|
8.4 | IC50 | 2 | — | |
CAOVBAQHBWKZJG
|
8.3 | IC50 | 3 | — | |
QBGYCMODWQDKCX
|
8.3 | IC50 | 2 | — | |
UJTVNGWILMVGHV
|
8.3 | IC50 | 2 | — | |
UYAQWCZWVIFRCN
|
8.3 | IC50 | 2 | — | |
AAANQOJVZBRGRH
|
8.3 | IC50 | 3 | — | |
BALRJMDHDGPHTH
|
8.3 | IC50 | 3 | — | |
JIIUKZNINHUSRU
|
8.3 | IC50 | 2 | — | |
QWRVRFNSEGHCBL
|
8.3 | IC50 | 2 | — | |
CUOVQWSQXJWUPZ
|
8.3 | IC50 | 2 | — | |
KEZOOBHJFUUXAY
|
8.3 | IC50 | 2 | — | |
VTTNWVNGYMKTFA
|
8.3 | IC50 | 2 | — | |
ZIJTUQQBFTXSRP
|
8.3 | IC50 | 2 | — | |
HWQQHGYFYYEJPD
|
8.3 | IC50 | 2 | — | |
CTPZTYYKWXJYMT
|
8.3 | IC50 | 2 | — | |
OUQRCKNQVHENIF
|
8.3 | IC50 | 2 | — | |
SYOXQXNUFXRNKH
|
8.3 | IC50 | 3 | — | |
ZOFPTOHAYCZFGK
|
8.3 | IC50 | 3 | — | |
GKHICIJKBRWUCL
|
8.3 | IC50 | 3 | — | |
MXKTVDFRBVSJHZ
|
8.3 | IC50 | 2 | — | |
HQMKZJLJBDXPIZ
|
8.3 | IC50 | 3 | — | |
RVZJFCNYSSUDCU
|
8.3 | IC50 | 7 | — | |
RVZJFCNYSSUDCU
|
8.3 | Kd | 2 | — | |
SRQKZTUWCVJTDC
|
8.3 | IC50 | 2 | — | |
WOJAWRJOQHZDRX
|
8.3 | IC50 | 2 | — |