Target Details
| UniProt AC | P48729 |
|---|---|
| Gene Symbol | CSNK1A1 |
| Protein Name | Casein kinase I isoform alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 470
- Clinical molecules 11
- Avg pChEMBL 7.5
KEGG Pathways (9)
Active Molecules (470)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JBJYTZXCZDNOJW
|
6.0 | IC50 | 2 | — | |
JZTOUVBEZONDKA
|
6.0 | Ki | 80 | — | |
KBFBKKNSHPUFET
|
6.0 | Ki | 5 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
LBVKEEFIPBQIMD
|
6.0 | Ki | 27 | — | |
LSLPDHNUWRDOGC
|
6.0 | Ki | 25 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NLUPJKQOKWBWFC
|
6.0 | Ki | 69 | — | |
OUSFTKFNBAZUKL
|
6.0 | Kd | 58 | Yes | |
OWFLADWRSCINST
|
6.0 | Ki | 30 | — | |
PYQFQGXOARMGAQ
|
6.0 | IC50 | 11 | — | |
QHKYPYXTTXKZST
|
6.0 | Ki | 28 | — | |
RGOPHVZLEMGMBZ
|
6.0 | Ki | 20 | — | |
SVUIYNKSDCANAY
|
6.0 | Ki | 16 | — | |
VBIYDORVDCFKHM
|
6.0 | Ki | 13 | — | |
VRIFJAKXSBXYFZ
|
6.0 | Ki | 8 | — | |
XPHWIERLJBFPFV
|
6.0 | Ki | 69 | — | |
XTVULKIROSNNTG
|
6.0 | Ki | 29 | — | |
YMIJUBCSOKSFRU
|
6.0 | Ki | 87 | — | |
YNUMBZPWLHDVEX
|
6.0 | Ki | 6 | — |