Target Details
| UniProt AC | P48549 |
|---|---|
| Gene Symbol | KCNJ3 |
| Protein Name | G protein-activated inward rectifier potassium channel 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01007 (IRK) PF17655 (IRK_C) |
Summary
- Multi-target molecules 143
- Clinical molecules 0
- Avg pChEMBL 6.87
KEGG Pathways (10)
Active Molecules (143)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NACUEOVEOGDGII
|
6.5 | IC50 | 2 | — | |
LYJIYGZXENLAPE
|
6.4 | IC50 | 2 | — | |
NACUEOVEOGDGII
|
6.4 | IC50 | 2 | — | |
HWHJLTXOSDACJN
|
6.4 | IC50 | 3 | — | |
LFOZKAQFOKTGII
|
6.4 | IC50 | 2 | — | |
PCMMBCZCYFFFPN
|
6.4 | IC50 | 2 | — | |
KUICHCUXYZKNOO
|
6.3 | IC50 | 3 | — | |
UWRHVPLUUPPQMY
|
6.3 | IC50 | 3 | — | |
FGDZDUOUXXUQNC
|
6.3 | IC50 | 2 | — | |
TVNJCCQHEJCRNN
|
6.3 | IC50 | 2 | — | |
CMPJAGCXBOHFAF
|
6.3 | IC50 | 3 | — | |
PZCYDKAVVVBKMA
|
6.3 | IC50 | 3 | — | |
UVMFWOKHXJEFRH
|
6.3 | IC50 | 3 | — | |
HKOFDZHMCAXCDS
|
6.3 | IC50 | 3 | — | |
YHMZEOXOMITJAP
|
6.3 | IC50 | 2 | — | |
AQQAHAYQAJHXGR
|
6.3 | IC50 | 3 | — | |
ZIQQHOBPJRQYEL
|
6.3 | IC50 | 3 | — | |
IJOJWHSJUNWVSC
|
6.3 | IC50 | 2 | — | |
NYSHIPDVLVFILL
|
6.2 | IC50 | 3 | — | |
FICICJIEUQQPMN
|
6.2 | IC50 | 2 | — | |
JKYYHANCMQDUCZ
|
6.2 | IC50 | 3 | — | |
FSXVXGIXJHYALR
|
6.2 | IC50 | 3 | — | |
JSMYZOGJVLHMQJ
|
6.2 | IC50 | 3 | — | |
LIAFEMWXGYBTML
|
6.2 | IC50 | 2 | — | |
HWFDNIKGXJLHGC
|
6.2 | IC50 | 2 | — | |
OXMXIXOKIIPOHL
|
6.2 | IC50 | 3 | — | |
ILNOCUPRGROOMO
|
6.1 | IC50 | 3 | — | |
WMKOFHYQCJBOLA
|
6.1 | IC50 | 2 | — | |
AHZZRNPXIUXUFU
|
6.1 | IC50 | 3 | — | |
XDFLKJCYHLTIAP
|
6.1 | IC50 | 2 | — | |
CBJBDCXJQSNMSZ
|
6.1 | IC50 | 3 | — | |
BSHNBXWFTGFFHC
|
6.1 | IC50 | 3 | — | |
OPFUTVRZTCWTRC
|
6.1 | IC50 | 3 | — | |
AMCGZCKPUGVFCK
|
6.1 | IC50 | 2 | — | |
LNTOZVGJRVNTIE
|
6.1 | IC50 | 2 | — | |
PZPIHPWBSGLFFH
|
6.1 | IC50 | 2 | — | |
WOOQITHNVSFGKK
|
6.0 | IC50 | 3 | — | |
QEXPFDNRGMLZPW
|
6.0 | IC50 | 3 | — | |
NNVDXVUCNSMWTQ
|
6.0 | IC50 | 2 | — | |
CFHAMFAFVWBLDT
|
6.0 | IC50 | 3 | — | |
QEBMMPNMOSIUKC
|
6.0 | IC50 | 3 | — | |
YRKPFBCMURMWHH
|
6.0 | IC50 | 2 | — | |
XBRDFDHQDNGPAA
|
6.0 | IC50 | 3 | — |