Target Details
| UniProt AC | P48549 |
|---|---|
| Gene Symbol | KCNJ3 |
| Protein Name | G protein-activated inward rectifier potassium channel 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01007 (IRK) PF17655 (IRK_C) |
Summary
- Multi-target molecules 143
- Clinical molecules 0
- Avg pChEMBL 6.87
KEGG Pathways (10)
Active Molecules (143)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XNUWGAOWLHXYGX
|
7.1 | IC50 | 2 | — | |
KYZSDKSHODHMRD
|
7.0 | IC50 | 3 | — | |
RLBUTVOWGRSOBF
|
7.0 | IC50 | 2 | — | |
AAPHFUNPTFOKHK
|
7.0 | IC50 | 2 | — | |
MEDIMLKAXOOFGC
|
7.0 | IC50 | 2 | — | |
MTKOXTDETDSROF
|
7.0 | IC50 | 2 | — | |
ZFFSQOGPNZWLRZ
|
7.0 | IC50 | 2 | — | |
DDDSGZFENQKDDY
|
7.0 | IC50 | 2 | — | |
PMNIPBGSJIEKQS
|
6.9 | IC50 | 2 | — | |
XDAYAPJRCGNDON
|
6.9 | IC50 | 2 | — | |
OSWNTPIKMGXESA
|
6.9 | IC50 | 2 | — | |
DDDSGZFENQKDDY
|
6.9 | IC50 | 3 | — | |
BUFKMYQMAHJBHT
|
6.9 | IC50 | 2 | — | |
DDDSGZFENQKDDY
|
6.9 | IC50 | 2 | — | |
AKSZPYCQJARRAA
|
6.8 | IC50 | 2 | — | |
ALXTXATYLGFTMA
|
6.8 | IC50 | 2 | — | |
NCMYMRCUTWGGJO
|
6.8 | IC50 | 2 | — | |
DPUOOLDBTIZYJV
|
6.8 | IC50 | 2 | — | |
XDAYAPJRCGNDON
|
6.8 | IC50 | 2 | — | |
XUENZROPARGQNH
|
6.8 | IC50 | 2 | — | |
MGRLWDRGBXQTMU
|
6.8 | IC50 | 3 | — | |
OVOYJHPFWJNUQB
|
6.8 | IC50 | 2 | — | |
HUMITMAJXKZKTO
|
6.8 | IC50 | 2 | — | |
QHACNFMTZPBWRL
|
6.8 | IC50 | 2 | — | |
AINXAXVYSCZWQG
|
6.8 | IC50 | 3 | — | |
IKPDCTPBFIIQRF
|
6.8 | IC50 | 2 | — | |
VXGWLTJUJVHZMV
|
6.8 | IC50 | 2 | — | |
FJJRZFWOCQMGEY
|
6.7 | IC50 | 2 | — | |
MLKRCEWWRVAFRU
|
6.7 | IC50 | 3 | — | |
LYJIYGZXENLAPE
|
6.7 | IC50 | 2 | — | |
CLIYTKDQEKPQQV
|
6.7 | IC50 | 2 | — | |
HUIYSGLQEYEPFI
|
6.7 | IC50 | 3 | — | |
DBYLIOOXAAJUAD
|
6.6 | IC50 | 2 | — | |
OEYIWLUJHKVFFP
|
6.6 | IC50 | 2 | — | |
YFKJAUKINKKAPS
|
6.6 | IC50 | 2 | — | |
CHVSUZLQBVXEQI
|
6.6 | IC50 | 2 | — | |
NOHWRIQJLRSUIM
|
6.6 | IC50 | 3 | — | |
GJDHCQVTACKVML
|
6.6 | IC50 | 2 | — | |
TXBPZBKXZMRZAD
|
6.6 | IC50 | 2 | — | |
BORCZNYMAGQEGS
|
6.6 | IC50 | 3 | — | |
XDAYAPJRCGNDON
|
6.6 | IC50 | 2 | — | |
JEIFFJHSPMANBT
|
6.5 | IC50 | 2 | — | |
JDBLAMMCTHKGTE
|
6.5 | IC50 | 2 | — | |
NACUEOVEOGDGII
|
6.5 | IC50 | 2 | — | |
JDMFEDXJXXQMKN
|
6.5 | IC50 | 2 | — | |
ALRMPHHZEVRXDO
|
6.5 | IC50 | 3 | — | |
IOJQHMDFIWJXLF
|
6.5 | IC50 | 2 | — | |
MREYLDDLEGSHRF
|
6.5 | IC50 | 2 | — | |
RTXJBTFTKDIJGJ
|
6.5 | IC50 | 2 | — | |
LYJIYGZXENLAPE
|
6.5 | IC50 | 2 | — |