Target Details
| UniProt AC | P48549 |
|---|---|
| Gene Symbol | KCNJ3 |
| Protein Name | G protein-activated inward rectifier potassium channel 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01007 (IRK) PF17655 (IRK_C) |
Summary
- Multi-target molecules 143
- Clinical molecules 0
- Avg pChEMBL 6.87
KEGG Pathways (10)
Active Molecules (143)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WZJJOHJIKKADBA
|
8.7 | IC50 | 2 | — | |
XSTIKDBUFTWNNB
|
8.1 | IC50 | 2 | — | |
DBRBZVDPIWOVAV
|
8.1 | Ki | 3 | — | |
VJWMFGICJZJHAO
|
8.1 | IC50 | 2 | — | |
YBFIRRLWTMWYQM
|
8.1 | IC50 | 2 | — | |
PPOFRZAMNFVMDG
|
8.0 | IC50 | 2 | — | |
XTBUAANEULFASN
|
8.0 | IC50 | 2 | — | |
NEIITZWACZSJEY
|
7.9 | IC50 | 2 | — | |
XYYWOQHYDUCWCD
|
7.9 | IC50 | 2 | — | |
XYYWOQHYDUCWCD
|
7.8 | IC50 | 2 | — | |
LBUKDMRMXBBNPX
|
7.8 | IC50 | 2 | — | |
SCIZOVDYSFRBNZ
|
7.8 | IC50 | 2 | — | |
QGZGTAVFFSLXOZ
|
7.8 | IC50 | 2 | — | |
XYYWOQHYDUCWCD
|
7.8 | IC50 | 2 | — | |
LHOYPFIGBFSNOS
|
7.7 | IC50 | 2 | — | |
HCTCNUKJFUGPRV
|
7.6 | IC50 | 2 | — | |
WDGVFWSLMYEAGZ
|
7.6 | IC50 | 2 | — | |
GJTKABAAPMNUMC
|
7.6 | IC50 | 2 | — | |
LBCVNBYMBREQQW
|
7.6 | IC50 | 2 | — | |
XNEUDCWKNMCPIY
|
7.6 | IC50 | 2 | — | |
WDTOLNJBENUFBQ
|
7.6 | IC50 | 2 | — | |
SJJQFMZJSMAXHL
|
7.5 | IC50 | 2 | — | |
TUKPJFKLDJTXDD
|
7.5 | IC50 | 2 | — | |
OZAPVCJGIULPCZ
|
7.5 | IC50 | 2 | — | |
SNMWXWMIXVAIPH
|
7.5 | IC50 | 2 | — | |
BSKNWGRELQKJMA
|
7.5 | IC50 | 2 | — | |
BAKFDWZBSGAYAR
|
7.5 | IC50 | 2 | — | |
ZXTLKJYZTUFSID
|
7.5 | IC50 | 2 | — | |
QHACNFMTZPBWRL
|
7.5 | IC50 | 2 | — | |
BMSQSCMJMBTGSK
|
7.5 | IC50 | 2 | — | |
LJRVXPVZQPEPBW
|
7.4 | IC50 | 2 | — | |
HLIDCCUMHXLIRM
|
7.4 | IC50 | 2 | — | |
MGUUTBZGBKDYFF
|
7.4 | IC50 | 2 | — | |
KWKBWPLUKPGJCR
|
7.4 | IC50 | 2 | — | |
FJNDSSQBHOYCSW
|
7.4 | IC50 | 2 | — | |
MHWBUIZVNLFKEP
|
7.4 | IC50 | 2 | — | |
YLYMIVSKYAHRGN
|
7.3 | IC50 | 2 | — | |
SYWRDVNCTMJCFH
|
7.3 | IC50 | 2 | — | |
AWQZXHDLUBADMM
|
7.3 | IC50 | 2 | — | |
CHQGILRQWLEPAK
|
7.3 | IC50 | 3 | — | |
AIIUGOHGPMBKHX
|
7.3 | IC50 | 2 | — | |
DCKMLYPIFNABIX
|
7.3 | IC50 | 2 | — | |
XTTWQOXKGSVQSX
|
7.2 | IC50 | 2 | — | |
ITPBWSUVZDXXGH
|
7.2 | IC50 | 2 | — | |
QTLNAOKNMRRSKL
|
7.2 | IC50 | 2 | — | |
MHXJMDYNADZPBS
|
7.2 | IC50 | 2 | — | |
FWXGVUPQGGYNPO
|
7.2 | IC50 | 2 | — | |
XDLLFWSQHBDIIK
|
7.2 | IC50 | 2 | — | |
PGJVAYQMCYJFFH
|
7.1 | IC50 | 2 | — | |
WUOZKIDPSWHTMY
|
7.1 | IC50 | 2 | — |